MY143370A - Fused quinoline derivative and use thereof - Google Patents

Fused quinoline derivative and use thereof

Info

Publication number
MY143370A
MY143370A MYPI20051875A MYPI20051875A MY143370A MY 143370 A MY143370 A MY 143370A MY PI20051875 A MYPI20051875 A MY PI20051875A MY PI20051875 A MYPI20051875 A MY PI20051875A MY 143370 A MY143370 A MY 143370A
Authority
MY
Malaysia
Prior art keywords
hydrogen atom
substituent
quinoline derivative
absence
represent
Prior art date
Application number
MYPI20051875A
Other languages
English (en)
Inventor
Masahiro Kajino
Nicholas Williams Hird
Naoki Tarui
Hiroshi Banno
Yasuhiko Kawano
Nobuhiro Inatomi
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of MY143370A publication Critical patent/MY143370A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
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    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • AHUMAN NECESSITIES
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    • A61P9/12Antihypertensives

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Virology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Oncology (AREA)
  • Psychiatry (AREA)
  • Communicable Diseases (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Psychology (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Anesthesiology (AREA)
  • Ophthalmology & Optometry (AREA)
MYPI20051875A 2004-04-28 2005-04-28 Fused quinoline derivative and use thereof MY143370A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2004134705 2004-04-28

Publications (1)

Publication Number Publication Date
MY143370A true MY143370A (en) 2011-04-29

Family

ID=34966886

Family Applications (1)

Application Number Title Priority Date Filing Date
MYPI20051875A MY143370A (en) 2004-04-28 2005-04-28 Fused quinoline derivative and use thereof

Country Status (28)

Country Link
US (4) US7592453B2 (pt)
EP (2) EP1740584B9 (pt)
JP (2) JP4361566B2 (pt)
KR (1) KR20070015598A (pt)
CN (1) CN1976932A (pt)
AT (1) ATE416176T1 (pt)
AU (1) AU2005238388B2 (pt)
BR (1) BRPI0510365A (pt)
CA (1) CA2565018A1 (pt)
CR (1) CR8755A (pt)
CY (1) CY1109222T1 (pt)
DE (1) DE602005011424D1 (pt)
DK (1) DK1740584T5 (pt)
ES (1) ES2318483T4 (pt)
HK (1) HK1099284A1 (pt)
HR (1) HRP20090121T5 (pt)
MX (1) MXPA06012323A (pt)
MY (1) MY143370A (pt)
NO (1) NO20065494L (pt)
NZ (1) NZ550983A (pt)
PL (1) PL1740584T3 (pt)
PT (1) PT1740584E (pt)
RS (1) RS50756B (pt)
RU (1) RU2384571C2 (pt)
SI (1) SI1740584T1 (pt)
TW (1) TW200540155A (pt)
WO (1) WO2005105802A1 (pt)
ZA (1) ZA200609261B (pt)

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US7592453B2 (en) * 2004-04-28 2009-09-22 Takeda Pharmaceutical Company Limited Fused quinoline derivative and use thereof
MXPA06014909A (es) 2004-06-18 2007-02-28 Chiron Corp Derivados de n-(1-(1-bencil -4-fenil-1h -imidazol -2-il)-2, 2-dimetilpropil) benzamida y compuestos relacionados como inhibidores de proteina de huso de cinesina (ksp) para el tratamiento del cancer.
NZ554555A (en) 2004-10-20 2011-09-30 Univ California Cyclohexyl-urea derivatives as improved inhibitors for the soluble epoxide hydrolase
DE102005027170A1 (de) * 2005-06-13 2006-12-14 Merck Patent Gmbh Substituierte Tetrahydrochinoline
GB0522715D0 (en) * 2005-11-08 2005-12-14 Helperby Therapeutics Ltd New use
WO2007074491A1 (en) * 2005-12-28 2007-07-05 Universita Degli Studi Di Siena HETEROTRICYCLIC AMIDE DERIVATIVES AS NEUROKININ-l (NKl) RECEPTOR LIGANDS
JP4509080B2 (ja) * 2006-09-28 2010-07-21 信越化学工業株式会社 シルセスキオキサン系化合物混合物及び加水分解性シラン化合物、その製造方法及びそれを用いたレジスト組成物並びにパターン形成方法及び基板の加工方法
WO2008070994A1 (en) 2006-12-14 2008-06-19 Nps Pharmaceuticals, Inc. Use of d-serine derivatives for the treatment of anxiety disorders
WO2008109991A1 (en) 2007-03-09 2008-09-18 University Health Network Inhibitors of carnitine palmitoyltransferase and treating cancer
DE102007013856A1 (de) 2007-03-20 2008-09-25 Merck Patent Gmbh Substituierte Tetrahydropyrrolochinoline
WO2008153027A1 (ja) * 2007-06-11 2008-12-18 Takeda Pharmaceutical Company Limited ピロロキノリン誘導体およびその用途
US8680282B2 (en) 2007-08-01 2014-03-25 University Health Network Cyclic inhibitors of carnitine palmitoyltransferase and treating cancer
AR069526A1 (es) 2007-12-03 2010-01-27 Takeda Pharmaceutical Compuesto heterociclico que contiene nitrogeno y su uso
TWI498115B (zh) 2007-12-27 2015-09-01 Daiichi Sankyo Co Ltd 咪唑羰基化合物
USRE48334E1 (en) 2008-09-19 2020-12-01 Takeda Pharmaceutical Company Limited Nitrogen-containing heterocyclic compound and use of same
WO2010038434A1 (ja) * 2008-09-30 2010-04-08 武田薬品工業株式会社 光学活性なヘキサヒドロピロロキノリン類の製造法およびその中間体
JP2011256110A (ja) * 2008-09-30 2011-12-22 Takeda Chem Ind Ltd ヘキサヒドロピロロキノリンの製造法
AR075158A1 (es) 2009-01-27 2011-03-16 Takeda Pharmaceutical Derivados de pirrolopirimidinas, composiciones farmaceuticas y usos.
JP2013053070A (ja) 2009-11-06 2013-03-21 Takeda Chem Ind Ltd ジヒドロピロロキノリン誘導体
AU2010339691B2 (en) * 2010-01-07 2015-04-02 Alkermes Pharma Ireland Limited Prodrugs of heteraromatic compounds
FR2974729B1 (fr) * 2011-05-02 2013-04-19 Servier Lab Nouvelle association entre le 4-{3-[cis-hexahydrocyclopenta[c]pyrrol-2(1h)-yl]propoxy}benzamide et un inhibiteur de l'acetylcholinesterase et les compositions pharmaceutiques qui la contiennent
EP2647638A1 (en) * 2012-04-02 2013-10-09 Almirall, S.A. Substituted tricyclic compounds with activity towards ep1 receptors
CN105017266B (zh) * 2015-07-17 2017-07-18 安徽农业大学 手性2‑芳基‑1,2,3,4‑四氢喹啉类化合物及其合成方法
MX2018009759A (es) 2016-02-12 2018-11-29 Astellas Pharma Inc Derivados de tetrahidroisoquinolina.
WO2018085288A1 (en) * 2016-11-01 2018-05-11 President And Fellows Of Harvard College Inhibitors of rna guided nucleases and uses thereof
US11352357B2 (en) 2019-11-27 2022-06-07 Sumitomo Dainippon Pharma Co., Ltd. Cycloalkylurea derivative
CA3157769A1 (en) * 2019-11-27 2021-06-03 Eiji IDEUE Cycloalkyl urea derivative
WO2021150613A1 (en) 2020-01-20 2021-07-29 Incyte Corporation Spiro compounds as inhibitors of kras
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