ZA200609261B - Fused quinoline derivative and use thereof - Google Patents

Fused quinoline derivative and use thereof

Info

Publication number
ZA200609261B
ZA200609261B ZA200609261A ZA200609261A ZA200609261B ZA 200609261 B ZA200609261 B ZA 200609261B ZA 200609261 A ZA200609261 A ZA 200609261A ZA 200609261 A ZA200609261 A ZA 200609261A ZA 200609261 B ZA200609261 B ZA 200609261B
Authority
ZA
South Africa
Prior art keywords
substituent
optionally
group optionally
acyl
hydrogen atom
Prior art date
Application number
ZA200609261A
Other languages
English (en)
Inventor
Kajino Masahiro
Hird Nicholas William
Tarui Naoki
Banno Hiroshi
Kawano Yasuhiko
Inatomi Nobuhiro
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of ZA200609261B publication Critical patent/ZA200609261B/xx

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
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    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Psychiatry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Oncology (AREA)
  • Hospice & Palliative Care (AREA)
  • Communicable Diseases (AREA)
  • Otolaryngology (AREA)
  • Molecular Biology (AREA)
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ZA200609261A 2004-04-28 2005-04-28 Fused quinoline derivative and use thereof ZA200609261B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2004134705 2004-04-28

Publications (1)

Publication Number Publication Date
ZA200609261B true ZA200609261B (en) 2008-08-27

Family

ID=34966886

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200609261A ZA200609261B (en) 2004-04-28 2005-04-28 Fused quinoline derivative and use thereof

Country Status (28)

Country Link
US (4) US7592453B2 (xx)
EP (2) EP1740584B9 (xx)
JP (2) JP4361566B2 (xx)
KR (1) KR20070015598A (xx)
CN (1) CN1976932A (xx)
AT (1) ATE416176T1 (xx)
AU (1) AU2005238388B2 (xx)
BR (1) BRPI0510365A (xx)
CA (1) CA2565018A1 (xx)
CR (1) CR8755A (xx)
CY (1) CY1109222T1 (xx)
DE (1) DE602005011424D1 (xx)
DK (1) DK1740584T5 (xx)
ES (1) ES2318483T4 (xx)
HK (1) HK1099284A1 (xx)
HR (1) HRP20090121T5 (xx)
MX (1) MXPA06012323A (xx)
MY (1) MY143370A (xx)
NO (1) NO20065494L (xx)
NZ (1) NZ550983A (xx)
PL (1) PL1740584T3 (xx)
PT (1) PT1740584E (xx)
RS (1) RS50756B (xx)
RU (1) RU2384571C2 (xx)
SI (1) SI1740584T1 (xx)
TW (1) TW200540155A (xx)
WO (1) WO2005105802A1 (xx)
ZA (1) ZA200609261B (xx)

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RS50756B (sr) * 2004-04-28 2010-08-31 Takeda Pharmaceutical Company Limited Fuzionisani derivati hinolina i njegova upotreba
EP1765789B1 (en) * 2004-06-18 2013-02-27 Novartis AG N-(1-(1-benzyl-4-phenyl-1h-imidazol-2-yl)-2,2-dimethylpropyl)benzamide derivatives and related compounds as kinesin spindle protein (ksp) inhibitors for the treatment of cancer
CA2584342C (en) 2004-10-20 2013-04-30 The Regents Of The University Of California Improved inhibitors for the soluble epoxide hydrolase
DE102005027170A1 (de) * 2005-06-13 2006-12-14 Merck Patent Gmbh Substituierte Tetrahydrochinoline
GB0522715D0 (en) 2005-11-08 2005-12-14 Helperby Therapeutics Ltd New use
WO2007074491A1 (en) * 2005-12-28 2007-07-05 Universita Degli Studi Di Siena HETEROTRICYCLIC AMIDE DERIVATIVES AS NEUROKININ-l (NKl) RECEPTOR LIGANDS
JP4509080B2 (ja) * 2006-09-28 2010-07-21 信越化学工業株式会社 シルセスキオキサン系化合物混合物及び加水分解性シラン化合物、その製造方法及びそれを用いたレジスト組成物並びにパターン形成方法及び基板の加工方法
CA2672494A1 (en) 2006-12-14 2008-06-19 Nps Pharmaceuticals, Inc. Use of d-serine derivatives for the treatment of anxiety disorders
WO2008109991A1 (en) 2007-03-09 2008-09-18 University Health Network Inhibitors of carnitine palmitoyltransferase and treating cancer
DE102007013856A1 (de) 2007-03-20 2008-09-25 Merck Patent Gmbh Substituierte Tetrahydropyrrolochinoline
WO2008153027A1 (ja) * 2007-06-11 2008-12-18 Takeda Pharmaceutical Company Limited ピロロキノリン誘導体およびその用途
WO2009015485A1 (en) * 2007-08-01 2009-02-05 University Health Network Cyclic inhibitors of carnitine palmitoyltransferase and treating cancer
TW200930713A (en) 2007-12-03 2009-07-16 Takeda Pharmaceutical Nitrogen-containing heterocyclic compound and use thereof
TWI498115B (zh) 2007-12-27 2015-09-01 Daiichi Sankyo Co Ltd 咪唑羰基化合物
USRE49686E1 (en) 2008-09-19 2023-10-10 Takeda Pharmaceutical Company Limited Nitrogen-containing heterocyclic compound and use of same
JP2011256110A (ja) * 2008-09-30 2011-12-22 Takeda Chem Ind Ltd ヘキサヒドロピロロキノリンの製造法
WO2010038434A1 (ja) * 2008-09-30 2010-04-08 武田薬品工業株式会社 光学活性なヘキサヒドロピロロキノリン類の製造法およびその中間体
US20100190747A1 (en) 2009-01-27 2010-07-29 Hideo Suzuki Fused ring compound and use thereof
JP2013053070A (ja) * 2009-11-06 2013-03-21 Takeda Chem Ind Ltd ジヒドロピロロキノリン誘導体
WO2011084848A2 (en) * 2010-01-07 2011-07-14 Alkermes, Inc. Prodrugs of heteraromatic compounds
FR2974729B1 (fr) * 2011-05-02 2013-04-19 Servier Lab Nouvelle association entre le 4-{3-[cis-hexahydrocyclopenta[c]pyrrol-2(1h)-yl]propoxy}benzamide et un inhibiteur de l'acetylcholinesterase et les compositions pharmaceutiques qui la contiennent
EP2647638A1 (en) * 2012-04-02 2013-10-09 Almirall, S.A. Substituted tricyclic compounds with activity towards ep1 receptors
CN105017266B (zh) * 2015-07-17 2017-07-18 安徽农业大学 手性2‑芳基‑1,2,3,4‑四氢喹啉类化合物及其合成方法
TWI773118B (zh) * 2016-02-12 2022-08-01 美商細胞動力學股份有限公司 四氫異喹啉衍生物
US11787795B2 (en) 2016-11-01 2023-10-17 President And Fellows Of Harvard College Inhibitors of RNA guided nucleases and uses thereof
US11352357B2 (en) 2019-11-27 2022-06-07 Sumitomo Dainippon Pharma Co., Ltd. Cycloalkylurea derivative
MX2022006422A (es) * 2019-11-27 2022-08-25 Sumitomo Pharma Co Ltd Derivado de cicloalquilurea.
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