MX9700763A - Procedimiento para la preparacion de benzoxazoles y derivados de piridinas utiles en el tratamiento de la diabetes del tipo ii, los benzoxazoles y derivados de piridina obtenidos, composiciones de los mismos y su uso. - Google Patents

Procedimiento para la preparacion de benzoxazoles y derivados de piridinas utiles en el tratamiento de la diabetes del tipo ii, los benzoxazoles y derivados de piridina obtenidos, composiciones de los mismos y su uso.

Info

Publication number
MX9700763A
MX9700763A MX9700763A MX9700763A MX9700763A MX 9700763 A MX9700763 A MX 9700763A MX 9700763 A MX9700763 A MX 9700763A MX 9700763 A MX9700763 A MX 9700763A MX 9700763 A MX9700763 A MX 9700763A
Authority
MX
Mexico
Prior art keywords
pryridine
benzoxazoles
diabetes
treatment
type
Prior art date
Application number
MX9700763A
Other languages
English (en)
Inventor
David Haigh
Harshad Kantilal Rami
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB9415330A external-priority patent/GB9415330D0/en
Priority claimed from GBGB9425599.9A external-priority patent/GB9425599D0/en
Priority claimed from GBGB9509923.0A external-priority patent/GB9509923D0/en
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of MX9700763A publication Critical patent/MX9700763A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

Un compuesto de la formula (I) o una sal farmacéuticamente aceptable del mismo, y/o un solvato farmacéuticamente aceptable del mismo, en donde R?? representa 2-benzoxazolilo o 2-piridilo y R1 representa CH2OCH3 o CF3; un procedimiento para la preparacion de dichos compuestos, una composicion farmacéutica que contiene dichos compuestos y el uso de dichos compuestos y composiciones en medicina.
MX9700763A 1994-07-29 1995-07-28 Procedimiento para la preparacion de benzoxazoles y derivados de piridinas utiles en el tratamiento de la diabetes del tipo ii, los benzoxazoles y derivados de piridina obtenidos, composiciones de los mismos y su uso. MX9700763A (es)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB9415330A GB9415330D0 (en) 1994-07-29 1994-07-29 Novel compounds
GBGB9425599.9A GB9425599D0 (en) 1994-12-19 1994-12-19 Novel compounds
GBGB9509923.0A GB9509923D0 (en) 1995-05-17 1995-05-17 Novel compounds
PCT/GB1995/001323 WO1996004261A1 (en) 1994-07-29 1995-06-07 Benzoxazoles and pryridine derivatives useful in the treatment of the type ii diabetes
PCT/EP1995/003038 WO1996004260A1 (en) 1994-07-29 1995-07-28 Benzoxazoles and pyridine derivatives useful in the treatment of the type ii diabetes

Publications (1)

Publication Number Publication Date
MX9700763A true MX9700763A (es) 1997-05-31

Family

ID=27267309

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9700763A MX9700763A (es) 1994-07-29 1995-07-28 Procedimiento para la preparacion de benzoxazoles y derivados de piridinas utiles en el tratamiento de la diabetes del tipo ii, los benzoxazoles y derivados de piridina obtenidos, composiciones de los mismos y su uso.

Country Status (16)

Country Link
EP (1) EP0772605A1 (es)
AP (1) AP776A (es)
BR (1) BR9508468A (es)
CA (1) CA2196079A1 (es)
CZ (1) CZ25497A3 (es)
DZ (1) DZ1916A1 (es)
FI (1) FI970357A (es)
HU (1) HUT76637A (es)
IL (3) IL114759A (es)
MA (1) MA23632A1 (es)
MX (1) MX9700763A (es)
NO (1) NO307827B1 (es)
OA (1) OA10470A (es)
PL (1) PL318766A1 (es)
SK (1) SK12297A3 (es)
WO (2) WO1996004261A1 (es)

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US6300339B1 (en) 1998-10-21 2001-10-09 Novo Nordisk A/S Compounds, their preparation and use
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Also Published As

Publication number Publication date
CA2196079A1 (en) 1996-02-15
NO970373L (no) 1997-03-18
WO1996004260A1 (en) 1996-02-15
IL114759A0 (en) 1995-12-31
MA23632A1 (fr) 1996-04-01
WO1996004261A1 (en) 1996-02-15
IL125525A0 (en) 1999-03-12
PL318766A1 (en) 1997-07-07
EP0772605A1 (en) 1997-05-14
IL125525A (en) 2000-02-29
NO307827B1 (no) 2000-06-05
FI970357A0 (fi) 1997-01-28
HUT76637A (en) 1997-10-28
DZ1916A1 (fr) 2002-02-17
IL114759A (en) 1999-10-28
BR9508468A (pt) 1997-11-25
AP776A (en) 1999-10-28
NO970373D0 (no) 1997-01-28
SK12297A3 (en) 1997-08-06
FI970357A (fi) 1997-03-26
OA10470A (en) 2002-04-08
AP9700918A0 (en) 1997-01-31
CZ25497A3 (en) 1997-09-17

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