MX2016011771A - Compuestos de amida, metodos de preparacion y uso de los mismos como agentes para el tratamiento y prevención de enfermedades ocasionadas por virus que contienen arn y/o adn y enfermedades concomitantes. - Google Patents

Compuestos de amida, metodos de preparacion y uso de los mismos como agentes para el tratamiento y prevención de enfermedades ocasionadas por virus que contienen arn y/o adn y enfermedades concomitantes.

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Publication number
MX2016011771A
MX2016011771A MX2016011771A MX2016011771A MX2016011771A MX 2016011771 A MX2016011771 A MX 2016011771A MX 2016011771 A MX2016011771 A MX 2016011771A MX 2016011771 A MX2016011771 A MX 2016011771A MX 2016011771 A MX2016011771 A MX 2016011771A
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Mexico
Prior art keywords
treatment
genus
prophylaxis
containing viruses
rna
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MX2016011771A
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English (en)
Inventor
Tatyana Alexandrovna Kromova
Evgenievich Nebolsin Vladimir
Original Assignee
Obschestvo S Ogranichennoi Otvetstvennostiyu Pharmenterprises
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Publication of MX2016011771A publication Critical patent/MX2016011771A/es

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    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C07D207/09—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
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Abstract

La presente invención se relaciona con medicina e incluye un método para prevenir y tratar enfermedades causadas por virus que contienen ARN y ADN, y enfermedades concomitantes, en donde el método comprende el uso de una cantidad efectiva de compuestos de la fórmula general I o sales farmacéuticamente aceptables de la misma; la invención también se relaciona con métodos para preparar dichos compuestos, composiciones farmacéuticas para la prevención o tratamiento de enfermedades causadas por virus que contienen ARN y ADN, dichas composiciones comprenden una cantidad efectiva de un compuesto de la fórmula I o una sal farmacéuticamente aceptable del mismo; la invención trata con el objetivo de proporcionar un agente novedoso efectivo en el tratamiento de enfermedades causadas por un virus que contiene ARN perteneciente al género Enterovirus, Metapneumo virus, Pneumovirus, Respirovirus o Alfa-coronavirus, y/o por un virus que contiene ADN perteneciente a la familia Adenoviridae y/o Herpesviridae, y en la prevención y tratamiento de exacerbación de asma, enfermedad pulmonar obstructiva crónica, mucoviscidosis, conjuntivitis, gastroenteritis, hepatitis, miocarditis; en la prevención y tratamiento de rinorrea, rinitis infecciosa y aguda, faringitis, nasofaringitis, tonsilitis, laringitis, laringotraqueitis, laringotraqueobronquitis, bronquitis, bronquiolitis, neumonía o síndrome obstructivo de la vía aérea.
MX2016011771A 2014-03-12 2015-02-27 Compuestos de amida, metodos de preparacion y uso de los mismos como agentes para el tratamiento y prevención de enfermedades ocasionadas por virus que contienen arn y/o adn y enfermedades concomitantes. MX2016011771A (es)

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RU2014109441A RU2628800C2 (ru) 2014-03-12 2014-03-12 Амидные соединения, способы получения, применение в качестве средств для лечения и профилактики заболеваний, вызываемых рнк-содержащими вирусами
PCT/RU2015/000121 WO2015137846A1 (ru) 2014-03-12 2015-02-27 Амидные соединения, способы их получения и применение

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MX2018009360A MX2018009360A (es) 2014-03-12 2016-09-09 Compuesto de amida y uso del mismo como agente para el tratamiento y prevencion de enfermedades ocasionadas por virus que contienen arn y/o adn, y enfermedades concomitantes.

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EA202090465A1 (ru) 2020-05-21
ES2938085T3 (es) 2023-04-04
EA201691694A1 (ru) 2017-01-30
EA201891417A1 (ru) 2018-11-30
SG10201806681YA (en) 2018-09-27
JP2017511374A (ja) 2017-04-20
JP6915911B2 (ja) 2021-08-04
UA123951C2 (uk) 2021-06-30
US20170183318A1 (en) 2017-06-29
EP3118211B1 (en) 2022-10-12
AU2015230061B2 (en) 2019-09-05

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