MX2016006337A - Compuestos heterociclicos novedosos. - Google Patents

Compuestos heterociclicos novedosos.

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Publication number
MX2016006337A
MX2016006337A MX2016006337A MX2016006337A MX2016006337A MX 2016006337 A MX2016006337 A MX 2016006337A MX 2016006337 A MX2016006337 A MX 2016006337A MX 2016006337 A MX2016006337 A MX 2016006337A MX 2016006337 A MX2016006337 A MX 2016006337A
Authority
MX
Mexico
Prior art keywords
heterocyclic compounds
novel heterocyclic
preparation
compounds
novel
Prior art date
Application number
MX2016006337A
Other languages
English (en)
Inventor
C Desai Ranjit
Srivastava Brijeshkumar
Original Assignee
Cadila Healthcare Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cadila Healthcare Ltd filed Critical Cadila Healthcare Ltd
Publication of MX2016006337A publication Critical patent/MX2016006337A/es

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/4162—1,2-Diazoles condensed with heterocyclic ring systems
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    • A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
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Abstract

La presente invención se refiere a agonistas de GPR 40 novedosos de la fórmula general (I), sus formas tautoméricas, sus estereoisómeros, sus sales farmacéuticamente aceptables, composiciones farmacéuticas que los contienen, métodos para su preparación, uso de estos compuestos en medicina y los intermedios implicados en su preparación. (ver Fórmula).
MX2016006337A 2013-11-14 2014-11-03 Compuestos heterociclicos novedosos. MX2016006337A (es)

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IN2013MU03577A (es) 2015-07-31
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US10246470B2 (en) 2019-04-02
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US20160257701A1 (en) 2016-09-08
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AU2014372114A1 (en) 2016-06-09
EP3068788A1 (en) 2016-09-21
AP2016009176A0 (en) 2016-04-30
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US20180346486A1 (en) 2018-12-06
JP2016537361A (ja) 2016-12-01
CA2928097A1 (en) 2015-07-02
CN105722841A (zh) 2016-06-29
MA38999A1 (fr) 2018-01-31
WO2015097713A1 (en) 2015-07-02
EA201690888A1 (ru) 2016-10-31

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