MX2014015794A - Procesos para la preparacion de 1,2,4-oxadiazoles 3,5-disustituidos. - Google Patents

Procesos para la preparacion de 1,2,4-oxadiazoles 3,5-disustituidos.

Info

Publication number
MX2014015794A
MX2014015794A MX2014015794A MX2014015794A MX2014015794A MX 2014015794 A MX2014015794 A MX 2014015794A MX 2014015794 A MX2014015794 A MX 2014015794A MX 2014015794 A MX2014015794 A MX 2014015794A MX 2014015794 A MX2014015794 A MX 2014015794A
Authority
MX
Mexico
Prior art keywords
disubstituted
processes
preparation
oxadiazo
les
Prior art date
Application number
MX2014015794A
Other languages
English (en)
Other versions
MX352351B (es
Inventor
David Louis Brown
William Harold Miller
Charles Richard Graham
Original Assignee
Monsanto Technology Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Monsanto Technology Llc filed Critical Monsanto Technology Llc
Publication of MX2014015794A publication Critical patent/MX2014015794A/es
Publication of MX352351B publication Critical patent/MX352351B/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

En la presente se proporcionan procesos para la preparación de 1,2,4-oxadiazoles 3,5-disustituidos y sales de los mismos que comprenden hacer reaccionar una N-hidroxiamidina con un cloruro de acilo en una mezcla de reacción que comprende un solvente orgánico inmiscible en agua y una base acuosa a temperaturas de reacción relativamente bajas.
MX2014015794A 2012-07-02 2013-07-02 Procesos para la preparacion de 1,2,4-oxadiazoles 3,5-disustituidos. MX352351B (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201261667361P 2012-07-02 2012-07-02
US201361777210P 2013-03-12 2013-03-12
US201361783466P 2013-03-14 2013-03-14
PCT/US2013/049060 WO2014008257A2 (en) 2012-07-02 2013-07-02 Processes for the preparation of 3,5-disubstituted-1,2,4-oxadiazoles

Publications (2)

Publication Number Publication Date
MX2014015794A true MX2014015794A (es) 2015-03-10
MX352351B MX352351B (es) 2017-11-21

Family

ID=49882590

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2014015794A MX352351B (es) 2012-07-02 2013-07-02 Procesos para la preparacion de 1,2,4-oxadiazoles 3,5-disustituidos.

Country Status (13)

Country Link
US (2) US9040711B2 (es)
EP (1) EP2867230B1 (es)
CN (1) CN104428296B (es)
AR (1) AR091655A1 (es)
AU (1) AU2013286860B2 (es)
BR (1) BR112014032956B1 (es)
CA (1) CA2876215A1 (es)
DK (1) DK2867230T3 (es)
ES (1) ES2782509T3 (es)
MX (1) MX352351B (es)
UA (1) UA114915C2 (es)
WO (1) WO2014008257A2 (es)
ZA (1) ZA201409000B (es)

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UA118254C2 (uk) 2012-12-04 2018-12-26 Монсанто Текнолоджи Ллс Нематоцидні водні композиції концентрату суспензії
AR095330A1 (es) 2013-03-15 2015-10-07 Monsanto Technology Llc Azoles n-,c-disustituidos y composiciones y métodos para controlar plagas de nematodos
JP6348568B2 (ja) 2013-03-15 2018-06-27 モンサント テクノロジー エルエルシー 線虫害虫防除のためのn−,c−二置換アゾール
CN103980265A (zh) * 2014-05-14 2014-08-13 武汉工程大学 3-苯基-5-(噻吩-2基)-1,2,4-噁二唑的合成工艺
US10982293B2 (en) 2014-05-20 2021-04-20 Monsanto Technology Llc Methods for improving plant resistance to soybean cyst nematode and compositions thereof
AU2015364465B2 (en) * 2014-12-19 2019-07-04 Monsanto Technology Llc Compositions and methods for improving agronomic characteristics of plants
WO2016143654A1 (ja) * 2015-03-06 2016-09-15 旭硝子株式会社 1,2,4-オキサジアゾール誘導体の製造方法
US10035793B2 (en) 2015-03-06 2018-07-31 Asahi Glass Company, Limited Method for producing 1,2,4-oxadiazole derivative
WO2016150937A1 (en) 2015-03-25 2016-09-29 Lonza Ltd Method for preparation of thiophenecarbonyl chlorides
CA2981066A1 (en) * 2015-03-31 2016-10-06 Monsanto Technology Llc Processes for the preparation of 2-thiophenecarbonyl chloride
TW201720807A (zh) * 2015-11-04 2017-06-16 隆薩有限公司 用草醯氯製備噻吩-2-羰醯氯的方法
CN109195961A (zh) * 2016-03-24 2019-01-11 孟山都技术公司 用于制备杂芳基羧酸的方法
CN111675672A (zh) * 2020-05-12 2020-09-18 石家庄市度智医药科技有限公司 一种制备阿塔鲁伦的方法

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Also Published As

Publication number Publication date
US20140039197A1 (en) 2014-02-06
EP2867230A2 (en) 2015-05-06
BR112014032956A2 (pt) 2017-06-27
WO2014008257A2 (en) 2014-01-09
US20150225382A1 (en) 2015-08-13
EP2867230B1 (en) 2020-02-12
MX352351B (es) 2017-11-21
CA2876215A1 (en) 2014-01-09
CN104428296A (zh) 2015-03-18
ZA201409000B (en) 2017-04-26
CN104428296B (zh) 2017-11-14
AU2013286860A1 (en) 2015-01-22
AR091655A1 (es) 2015-02-18
ES2782509T3 (es) 2020-09-15
BR112014032956B1 (pt) 2020-02-27
US9273037B2 (en) 2016-03-01
EP2867230A4 (en) 2016-04-13
AU2013286860B2 (en) 2017-10-26
US9040711B2 (en) 2015-05-26
UA114915C2 (uk) 2017-08-28
DK2867230T3 (da) 2020-04-14
WO2014008257A3 (en) 2014-02-27

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