MX352351B - Procesos para la preparacion de 1,2,4-oxadiazoles 3,5-disustituidos. - Google Patents

Procesos para la preparacion de 1,2,4-oxadiazoles 3,5-disustituidos.

Info

Publication number
MX352351B
MX352351B MX2014015794A MX2014015794A MX352351B MX 352351 B MX352351 B MX 352351B MX 2014015794 A MX2014015794 A MX 2014015794A MX 2014015794 A MX2014015794 A MX 2014015794A MX 352351 B MX352351 B MX 352351B
Authority
MX
Mexico
Prior art keywords
disubstituted
processes
preparation
oxadiazo
les
Prior art date
Application number
MX2014015794A
Other languages
English (en)
Other versions
MX2014015794A (es
Inventor
David Louis Brown
William Harold Miller
Charles Richard Graham
Original Assignee
Monsanto Technology Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Monsanto Technology Llc filed Critical Monsanto Technology Llc
Publication of MX2014015794A publication Critical patent/MX2014015794A/es
Publication of MX352351B publication Critical patent/MX352351B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles

Abstract

En la presente se proporcionan procesos para la preparación de 1,2,4-oxadiazoles 3,5-disustituidos y sales de los mismos que comprenden hacer reaccionar una N-hidroxiamidina con un cloruro de acilo en una mezcla de reacción que comprende un solvente orgánico inmiscible en agua y una base acuosa a temperaturas de reacción relativamente bajas.
MX2014015794A 2012-07-02 2013-07-02 Procesos para la preparacion de 1,2,4-oxadiazoles 3,5-disustituidos. MX352351B (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201261667361P 2012-07-02 2012-07-02
US201361777210P 2013-03-12 2013-03-12
US201361783466P 2013-03-14 2013-03-14
PCT/US2013/049060 WO2014008257A2 (en) 2012-07-02 2013-07-02 Processes for the preparation of 3,5-disubstituted-1,2,4-oxadiazoles

Publications (2)

Publication Number Publication Date
MX2014015794A MX2014015794A (es) 2015-03-10
MX352351B true MX352351B (es) 2017-11-21

Family

ID=49882590

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2014015794A MX352351B (es) 2012-07-02 2013-07-02 Procesos para la preparacion de 1,2,4-oxadiazoles 3,5-disustituidos.

Country Status (13)

Country Link
US (2) US9040711B2 (es)
EP (1) EP2867230B1 (es)
CN (1) CN104428296B (es)
AR (1) AR091655A1 (es)
AU (1) AU2013286860B2 (es)
BR (1) BR112014032956B1 (es)
CA (1) CA2876215A1 (es)
DK (1) DK2867230T3 (es)
ES (1) ES2782509T3 (es)
MX (1) MX352351B (es)
UA (1) UA114915C2 (es)
WO (1) WO2014008257A2 (es)
ZA (1) ZA201409000B (es)

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US9173401B2 (en) 2013-03-15 2015-11-03 Monsanto Technology Llc N-,C-disubstituted azoles and compositions and methods for controlling nematode pests
WO2014152132A1 (en) 2013-03-15 2014-09-25 Monsanto Technology Llc N-,c-disubstituted azoles for controlling nematode pests
CN103980265A (zh) * 2014-05-14 2014-08-13 武汉工程大学 3-苯基-5-(噻吩-2基)-1,2,4-噁二唑的合成工艺
CN106455509A (zh) 2014-05-20 2017-02-22 孟山都技术公司 用于改进植物对大豆孢囊线虫的抗性的方法及其组合物
CA2970944A1 (en) * 2014-12-19 2016-06-23 Monsanto Technology Llc Compositions and methods for improving agronomic characteristics of plants
WO2016143654A1 (ja) * 2015-03-06 2016-09-15 旭硝子株式会社 １，２，４－オキサジアゾール誘導体の製造方法
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CA2981066A1 (en) * 2015-03-31 2016-10-06 Monsanto Technology Llc Processes for the preparation of 2-thiophenecarbonyl chloride
WO2017076844A1 (en) * 2015-11-04 2017-05-11 Lonza Ltd Method for preparation of thiophene-2-carbonyl chlorides with oxalyl chloride
AU2017238056A1 (en) 2016-03-24 2018-10-04 Monsanto Technology Llc Processes for the preparation of heteroaryl carboxylic acids
CN111675672A (zh) * 2020-05-12 2020-09-18 石家庄市度智医药科技有限公司 一种制备阿塔鲁伦的方法

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Also Published As

Publication number Publication date
US9040711B2 (en) 2015-05-26
AU2013286860A1 (en) 2015-01-22
BR112014032956B1 (pt) 2020-02-27
DK2867230T3 (da) 2020-04-14
MX2014015794A (es) 2015-03-10
US20150225382A1 (en) 2015-08-13
EP2867230B1 (en) 2020-02-12
US9273037B2 (en) 2016-03-01
WO2014008257A2 (en) 2014-01-09
CN104428296B (zh) 2017-11-14
CA2876215A1 (en) 2014-01-09
BR112014032956A2 (pt) 2017-06-27
UA114915C2 (uk) 2017-08-28
EP2867230A2 (en) 2015-05-06
CN104428296A (zh) 2015-03-18
EP2867230A4 (en) 2016-04-13
AU2013286860B2 (en) 2017-10-26
AR091655A1 (es) 2015-02-18
US20140039197A1 (en) 2014-02-06
ZA201409000B (en) 2017-04-26
WO2014008257A3 (en) 2014-02-27
ES2782509T3 (es) 2020-09-15

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