MX2012007868A - Metodo para preparar sales de acido tetrazol-mentasulfonico, y un nuevo compuesto utilizado en las mismas. - Google Patents

Metodo para preparar sales de acido tetrazol-mentasulfonico, y un nuevo compuesto utilizado en las mismas.

Info

Publication number
MX2012007868A
MX2012007868A MX2012007868A MX2012007868A MX2012007868A MX 2012007868 A MX2012007868 A MX 2012007868A MX 2012007868 A MX2012007868 A MX 2012007868A MX 2012007868 A MX2012007868 A MX 2012007868A MX 2012007868 A MX2012007868 A MX 2012007868A
Authority
MX
Mexico
Prior art keywords
methanesulfonic acid
acid salts
same
compound used
novel compound
Prior art date
Application number
MX2012007868A
Other languages
English (en)
Inventor
Keuk Chan Bang
Young Gil Ahn
Maeng Sup Kim
Jae Chul Lee
Bum Woo Park
Jong Won Choi
Yong Hoon An
Original Assignee
Hanmi Science Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hanmi Science Co Ltd filed Critical Hanmi Science Co Ltd
Publication of MX2012007868A publication Critical patent/MX2012007868A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

De acuerdo a la presente invención, un método para preparar sales de ácido tetrazol-metansulfónico que comprende una reacción de acilación que utiliza un nuevo S-benzotiazol 2-il-éster del ácido 4-iodin-4H-cromen-2-carbotiónico. El comparación con los métodos convencionales, y puede preparar sales de ácido tetrazol-metansulfónico de alta pureza a una elevada relación de rendimiento sin utilizar un método de cromatografía de columna.
MX2012007868A 2010-01-15 2011-01-14 Metodo para preparar sales de acido tetrazol-mentasulfonico, y un nuevo compuesto utilizado en las mismas. MX2012007868A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR1020100003835A KR101466245B1 (ko) 2010-01-15 2010-01-15 테트라졸 메탄설폰산 염의 제조방법 및 이에 사용되는 신규 화합물
PCT/KR2011/000291 WO2011087316A2 (ko) 2010-01-15 2011-01-14 테트라졸 메탄설폰산 염의 제조방법 및 이에 사용되는 신규 화합물

Publications (1)

Publication Number Publication Date
MX2012007868A true MX2012007868A (es) 2012-08-03

Family

ID=44304835

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2012007868A MX2012007868A (es) 2010-01-15 2011-01-14 Metodo para preparar sales de acido tetrazol-mentasulfonico, y un nuevo compuesto utilizado en las mismas.

Country Status (20)

Country Link
US (2) US8680277B2 (es)
EP (1) EP2524916B1 (es)
JP (1) JP5575921B2 (es)
KR (1) KR101466245B1 (es)
CN (1) CN102812020B (es)
AU (1) AU2011205891B2 (es)
BR (1) BR112012017448B1 (es)
CA (1) CA2786434C (es)
DK (1) DK2524916T3 (es)
ES (1) ES2514340T3 (es)
HK (1) HK1177211A1 (es)
IL (1) IL220851A (es)
MX (1) MX2012007868A (es)
NO (1) NO342589B1 (es)
NZ (1) NZ601805A (es)
PL (1) PL2524916T3 (es)
RU (1) RU2509769C1 (es)
SG (1) SG182430A1 (es)
WO (1) WO2011087316A2 (es)
ZA (1) ZA201206084B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101986683B1 (ko) * 2012-12-13 2019-06-10 한미약품 주식회사 테트라졸 유도체를 활성 성분으로 포함하는 용해도가 개선된 고체 분산체
CN103804352B (zh) * 2014-01-23 2017-06-13 中国药科大学 三氮唑苯乙基四氢异喹啉类化合物及其制备方法和应用
JO3737B1 (ar) * 2015-07-21 2021-01-31 Athenex Therapeutics Ltd تركيبات علاجية من باكليتاكسيل تعطى عن طريق الفم ومثبط P-gp لعلاج السرطان
US11165722B2 (en) 2016-06-29 2021-11-02 International Business Machines Corporation Cognitive messaging with dynamically changing inputs
WO2020168144A1 (en) 2019-02-14 2020-08-20 Teva Pharmaceuticals International Gmbh Solid state forms of n-[2-(2-{4-[2-(6,7-dimethoxy-3,4-dihydro-2(lh)- isoquinolinyl)ethyl] phenyl }-2h-tetrazol-5-yl)-4,5-dimethoxyphenyl] -4- oxo-4h-chromene-2-carboxamide and of its mesylate salt
WO2020194175A1 (en) * 2019-03-25 2020-10-01 Dr. Reddy's Laboratories Limited Solid forms of encequidar mesylate and processes thereof
WO2020230037A1 (en) * 2019-05-13 2020-11-19 Dr. Reddy's Laboratories Limited Alternate process for the preparation of encequidar
WO2021044350A1 (en) * 2019-09-04 2021-03-11 Dr. Reddy’S Laboratories Limited Solid forms of encequidar mesylate and processes thereof
US20230278990A1 (en) 2020-07-10 2023-09-07 Teva Czech Industries S.R.O Solid state forms of n-[2-(2-{4-[2-(6,7-dimethoxy-3,4-dihydro-2(1h)-isoquinolinyl)ethyl]phenyl}-2h-tetrazol-5-yl)-4,5-dimethoxyphenyl]-4-oxo-4h-chromene-2-carboxamide mesylate salt
CA3194694A1 (en) 2020-10-07 2022-04-14 Sameer Urgaonkar Acetamido-phenyltetrazole derivatives and methods of using the same

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL129871A (en) * 1994-05-06 2003-11-23 Pharmacia & Upjohn Inc Process for preparing 4-phenyl-substituted octanoyl-oxazolidin-2-one intermediates that are useful for preparing pyran-2-ones useful for treating retroviral infections
KR100508019B1 (ko) * 2003-07-19 2005-08-17 한미약품 주식회사 고순도 1-안드로스텐 유도체의 제조 방법
KR100557093B1 (ko) * 2003-10-07 2006-03-03 한미약품 주식회사 다약제 내성 저해 활성을 갖는 테트라졸 유도체 및 그의제조방법
US7279471B2 (en) * 2004-04-15 2007-10-09 Boehringer Ingelheim International Gmbh Selected CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions
KR100686695B1 (ko) * 2005-06-11 2007-02-26 주식회사 에스텍파마 프란루카스트 또는 그의 수화물의 제조방법 및 그의 합성중간체
US20070161791A1 (en) * 2006-01-09 2007-07-12 Narsimha Reddy Penthala Process for the preparation of terazosin hydrocloride dihydrate

Also Published As

Publication number Publication date
EP2524916B1 (en) 2014-07-23
US8680277B2 (en) 2014-03-25
NO20120841A1 (no) 2012-07-20
CA2786434C (en) 2014-05-13
CN102812020A (zh) 2012-12-05
US20140148602A1 (en) 2014-05-29
CA2786434A1 (en) 2011-07-21
US8940908B2 (en) 2015-01-27
JP2013517267A (ja) 2013-05-16
KR20110083870A (ko) 2011-07-21
ES2514340T3 (es) 2014-10-28
ZA201206084B (en) 2013-10-30
EP2524916A2 (en) 2012-11-21
DK2524916T3 (da) 2014-09-08
SG182430A1 (en) 2012-08-30
IL220851A0 (en) 2012-09-24
RU2509769C1 (ru) 2014-03-20
NO342589B1 (no) 2018-06-18
NZ601805A (en) 2014-07-25
JP5575921B2 (ja) 2014-08-20
KR101466245B1 (ko) 2014-12-01
WO2011087316A2 (ko) 2011-07-21
HK1177211A1 (en) 2013-08-16
WO2011087316A3 (ko) 2011-11-10
BR112012017448A2 (pt) 2016-08-09
EP2524916A4 (en) 2013-07-17
US20120330020A1 (en) 2012-12-27
AU2011205891A1 (en) 2012-09-06
CN102812020B (zh) 2015-03-18
PL2524916T3 (pl) 2015-01-30
BR112012017448B1 (pt) 2021-05-25
IL220851A (en) 2015-10-29
RU2012134783A (ru) 2014-02-20
AU2011205891B2 (en) 2013-09-05

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