MX349985B - Procedimiento de preparación de ésteres de fenilacetil aminoácido espirocíclicos con sustitución cis-alcoxi y derivados de 1h-pirrolidin-2,4-diona espirocicíclicos con sustitución cis-alcoxi. - Google Patents

Procedimiento de preparación de ésteres de fenilacetil aminoácido espirocíclicos con sustitución cis-alcoxi y derivados de 1h-pirrolidin-2,4-diona espirocicíclicos con sustitución cis-alcoxi.

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Publication number
MX349985B
MX349985B MX2014011577A MX2014011577A MX349985B MX 349985 B MX349985 B MX 349985B MX 2014011577 A MX2014011577 A MX 2014011577A MX 2014011577 A MX2014011577 A MX 2014011577A MX 349985 B MX349985 B MX 349985B
Authority
MX
Mexico
Prior art keywords
alkoxy
cis
substituted spirocyclic
pyrrolidine
acid esters
Prior art date
Application number
MX2014011577A
Other languages
English (en)
Other versions
MX2014011577A (es
Inventor
Rafael Warsitz
Winfried Etzel
Taraneh Farida
Berndt Maiwald
Martin Littmann
Nicolas Henck
Michael Esser
Original Assignee
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Publication of MX2014011577A publication Critical patent/MX2014011577A/es
Publication of MX349985B publication Critical patent/MX349985B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/45—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/46—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/51—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/45—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/52—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/54—Spiro-condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)
  • Indole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

La presente invención se refiere a un nuevo procedimiento de preparación de ésteres de fenilacetil aminoácido espirocíclicos con sustitución de cis-alcoxi y derivados de 1H-pirrolidin-2,4-dio na espirocíclicos con sustitución de cis-alcoxi y también a nuevos intermedios y materiales de partida que se producen y/o se usan en el procedimiento de acuerdo con la invención.
MX2014011577A 2012-03-28 2013-03-25 Procedimiento de preparación de ésteres de fenilacetil aminoácido espirocíclicos con sustitución cis-alcoxi y derivados de 1h-pirrolidin-2,4-diona espirocicíclicos con sustitución cis-alcoxi. MX349985B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12161837 2012-03-28
PCT/EP2013/056318 WO2013144101A1 (de) 2012-03-28 2013-03-25 Verfahren zur herstellung von cis-alkoxysubstituierten spirocyclischen phenylacetylaminosäureestern und cis-alkoxysubstituierten spirocyclischen 1-h-pyrrolidin-2,4-dion-derivaten

Publications (2)

Publication Number Publication Date
MX2014011577A MX2014011577A (es) 2014-11-21
MX349985B true MX349985B (es) 2017-08-22

Family

ID=47997506

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2014011577A MX349985B (es) 2012-03-28 2013-03-25 Procedimiento de preparación de ésteres de fenilacetil aminoácido espirocíclicos con sustitución cis-alcoxi y derivados de 1h-pirrolidin-2,4-diona espirocicíclicos con sustitución cis-alcoxi.

Country Status (13)

Country Link
US (2) US9376374B2 (es)
EP (1) EP2831038B1 (es)
JP (1) JP6158293B2 (es)
KR (1) KR102057491B1 (es)
CN (2) CN104245664B (es)
BR (1) BR112014023999B8 (es)
DK (1) DK2831038T3 (es)
ES (1) ES2644126T3 (es)
IL (1) IL234626A (es)
IN (1) IN2014DN07407A (es)
MX (1) MX349985B (es)
TW (1) TWI579260B (es)
WO (1) WO2013144101A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK3452446T3 (da) * 2016-05-04 2023-09-18 Bayer Cropscience Ag Fremgamgsmåde til fremstilling af cis-alkoxysubstituerede spirocykliske 1-h-pyrrolidin-2,4-dion-derivater
EP3301092A3 (de) 2018-01-26 2018-09-12 Bayer CropScience Aktiengesellschaft Verfahren zur herstellung von spiroketal-substituierten phenylacetylaminosäureestern und spiroketal-substituierten cyclischen ketoenolen
CN115448869A (zh) * 2021-06-09 2022-12-09 顺毅南通化工有限公司 一种螺虫乙酯合成用中间体的制备方法

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2733233A (en) * 1956-01-31 Vinyl esters of n-carbacyl-alpha-mono-
DE4431730A1 (de) * 1994-02-09 1995-08-10 Bayer Ag Substituierte 1H-3-Aryl-pyrrolidin-2,4-dion-Derivate
CA2187015A1 (en) * 1994-04-05 1995-10-12 Reiner Fischer Alkoxy-alkyl-substituted 1-h-3-aryl-pyrrolidine-2,4-diones used as herbicides and pesticides
CN1154634C (zh) * 1995-02-13 2004-06-23 拜尔公司 作为除草剂和杀虫剂的2-苯基取代杂环1,3-酮烯醇
JP4153033B2 (ja) * 1995-05-09 2008-09-17 バイエル アクチェンゲゼルシャフト 有害生物防除剤及び除草剤として有用なアルキルジハロゲン化フェニル置換ケトエノール
MX9710373A (es) * 1995-06-28 1998-07-31 Bayer Ag Fenilcetoenoles 2,4,5-trisubstituidos para el empleo como pesticidas y herbicidas.
CN100339352C (zh) * 1996-08-05 2007-09-26 拜尔公司 2－和2,5－取代的苯基酮烯醇
DE10016544A1 (de) * 2000-04-03 2001-10-11 Bayer Ag C2-phenylsubstituierte Ketoenole
DE10032587A1 (de) * 2000-07-05 2002-01-17 Bayer Ag 4-Alkoxy-cyclohexan-1-amino-carbonsäureester und Verfahren zu ihrer Herstellung
DE10231333A1 (de) * 2002-07-11 2004-01-22 Bayer Cropscience Ag Cis-Alkoxysubstituierte spirocyclische 1-H-Pyrrolidin-2,4-dion-Derivate
DE10239479A1 (de) * 2002-08-28 2004-03-04 Bayer Cropscience Ag Substituierte spirocyclische Ketoenole
DE102004030753A1 (de) * 2004-06-25 2006-01-19 Bayer Cropscience Ag 3'-Alkoxy spirocyclische Tetram- und Tretronsäuren
DE102004044827A1 (de) * 2004-09-16 2006-03-23 Bayer Cropscience Ag Jod-phenylsubstituierte cyclische Ketoenole
JP4012239B2 (ja) * 2006-01-11 2007-11-21 生化学工業株式会社 オキサゾロン誘導体
JP3975226B2 (ja) * 2006-01-11 2007-09-12 生化学工業株式会社 シクロアルキルカルボニルアミノ酸誘導体及びその製造方法
CN102241590B (zh) * 2011-05-17 2013-06-19 永农生物科学有限公司 一种螺环季酮酸类化合物关键中间体的合成方法
DE102011080406A1 (de) * 2011-08-04 2013-02-07 Bayer Pharma AG Substituierte 3-(Biphenyl-3-yl)-4-hydroxy-8-methoxy-1-azaspiro8[4.5]dec-3-en-2-one

Also Published As

Publication number Publication date
IL234626A (en) 2017-07-31
BR112014023999B8 (pt) 2020-05-12
CN106748861A (zh) 2017-05-31
TWI579260B (zh) 2017-04-21
EP2831038A1 (de) 2015-02-04
KR20140140045A (ko) 2014-12-08
US9376374B2 (en) 2016-06-28
DK2831038T3 (en) 2017-10-30
MX2014011577A (es) 2014-11-21
CN106748861B (zh) 2018-10-19
US20150051407A1 (en) 2015-02-19
CN104245664A (zh) 2014-12-24
KR102057491B1 (ko) 2019-12-19
TW201400440A (zh) 2014-01-01
JP6158293B2 (ja) 2017-07-05
JP2015516380A (ja) 2015-06-11
US9840459B2 (en) 2017-12-12
IN2014DN07407A (es) 2015-04-24
WO2013144101A1 (de) 2013-10-03
EP2831038B1 (de) 2017-07-19
US20160264516A1 (en) 2016-09-15
ES2644126T3 (es) 2017-11-27
CN104245664B (zh) 2016-12-07

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