MX2011009901A - Sistemas de administracion intraocular de farmacos de liberacion sostenida y metodos para tratar afecciones oculares. - Google Patents
Sistemas de administracion intraocular de farmacos de liberacion sostenida y metodos para tratar afecciones oculares.Info
- Publication number
- MX2011009901A MX2011009901A MX2011009901A MX2011009901A MX2011009901A MX 2011009901 A MX2011009901 A MX 2011009901A MX 2011009901 A MX2011009901 A MX 2011009901A MX 2011009901 A MX2011009901 A MX 2011009901A MX 2011009901 A MX2011009901 A MX 2011009901A
- Authority
- MX
- Mexico
- Prior art keywords
- microspheres
- compound
- implant
- days
- latanoprost
- Prior art date
Links
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- AKHNMLFCWUSKQB-UHFFFAOYSA-L sodium thiosulfate Chemical compound [Na+].[Na+].[O-]S([O-])(=O)=S AKHNMLFCWUSKQB-UHFFFAOYSA-L 0.000 description 1
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- 208000009056 telangiectasis Diseases 0.000 description 1
- 229940126585 therapeutic drug Drugs 0.000 description 1
- RTKIYNMVFMVABJ-UHFFFAOYSA-L thimerosal Chemical compound [Na+].CC[Hg]SC1=CC=CC=C1C([O-])=O RTKIYNMVFMVABJ-UHFFFAOYSA-L 0.000 description 1
- 229940033663 thimerosal Drugs 0.000 description 1
- 229960000454 timolol hemihydrate Drugs 0.000 description 1
- 229960005221 timolol maleate Drugs 0.000 description 1
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
- A61K9/0051—Ocular inserts, ocular implants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/557—Eicosanoids, e.g. leukotrienes or prostaglandins
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/557—Eicosanoids, e.g. leukotrienes or prostaglandins
- A61K31/5575—Eicosanoids, e.g. leukotrienes or prostaglandins having a cyclopentane, e.g. prostaglandin E2, prostaglandin F2-alpha
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
- A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2121/00—Preparations for use in therapy
Landscapes
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- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
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- Life Sciences & Earth Sciences (AREA)
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- Animal Behavior & Ethology (AREA)
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- Epidemiology (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Ophthalmology & Optometry (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| US12/411,250 US20100247606A1 (en) | 2009-03-25 | 2009-03-25 | Intraocular sustained release drug delivery systems and methods for treating ocular conditions |
| PCT/US2010/028584 WO2010111449A1 (en) | 2009-03-25 | 2010-03-25 | Intraocular sustained release drug delivery systems and methods for treating ocular conditions |
Publications (1)
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| MX2011009901A true MX2011009901A (es) | 2011-11-18 |
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| JP (2) | JP2012521997A (enExample) |
| KR (4) | KR20120006998A (enExample) |
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| BR (1) | BRPI1012324A2 (enExample) |
| CA (1) | CA2756065A1 (enExample) |
| IL (1) | IL215205A0 (enExample) |
| MX (1) | MX2011009901A (enExample) |
| NZ (1) | NZ595294A (enExample) |
| RU (2) | RU2532333C2 (enExample) |
| WO (1) | WO2010111449A1 (enExample) |
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| US9498457B2 (en) | 2004-04-30 | 2016-11-22 | Allergan, Inc. | Hypotensive prostamide-containing biodegradable intraocular implants and related implants |
| US8673341B2 (en) * | 2004-04-30 | 2014-03-18 | Allergan, Inc. | Intraocular pressure reduction with intracameral bimatoprost implants |
| US8722097B2 (en) | 2004-04-30 | 2014-05-13 | Allergan, Inc. | Oil-in-water method for making polymeric implants containing a hypotensive lipid |
| US7799336B2 (en) | 2004-04-30 | 2010-09-21 | Allergan, Inc. | Hypotensive lipid-containing biodegradable intraocular implants and related methods |
| US7993634B2 (en) | 2004-04-30 | 2011-08-09 | Allergan, Inc. | Oil-in-oil emulsified polymeric implants containing a hypotensive lipid and related methods |
| US7947732B2 (en) * | 2007-07-13 | 2011-05-24 | Allergan, Inc. | Therapeutic substituted chlorocyclopentanols |
| US9095404B2 (en) | 2008-05-12 | 2015-08-04 | University Of Utah Research Foundation | Intraocular drug delivery device and associated methods |
| US9877973B2 (en) | 2008-05-12 | 2018-01-30 | University Of Utah Research Foundation | Intraocular drug delivery device and associated methods |
| EP2276439A4 (en) | 2008-05-12 | 2013-11-27 | Univ Utah Res Found | DEVICE AND CORRESPONDING METHODS FOR INTRAOCULAR MEDICAMENT ADMINISTRATION |
| US10064819B2 (en) | 2008-05-12 | 2018-09-04 | University Of Utah Research Foundation | Intraocular drug delivery device and associated methods |
| US20100104654A1 (en) | 2008-10-27 | 2010-04-29 | Allergan, Inc. | Prostaglandin and prostamide drug delivery systems and intraocular therapeutic uses thereof |
| US10206813B2 (en) | 2009-05-18 | 2019-02-19 | Dose Medical Corporation | Implants with controlled drug delivery features and methods of using same |
| JP5937004B2 (ja) | 2009-05-18 | 2016-06-22 | ドーズ メディカル コーポレーションＤｏｓｅ Ｍｅｄｉｃａｌ Ｃｏｒｐｏｒａｔｉｏｎ | 薬剤溶出眼内インプラント |
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| WO2012071476A2 (en) | 2010-11-24 | 2012-05-31 | David Haffner | Drug eluting ocular implant |
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2009
- 2009-03-25 US US12/411,250 patent/US20100247606A1/en not_active Abandoned
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2010
- 2010-03-25 AU AU2010229891A patent/AU2010229891A1/en not_active Abandoned
- 2010-03-25 RU RU2011140433/15A patent/RU2532333C2/ru active
- 2010-03-25 KR KR1020117023983A patent/KR20120006998A/ko not_active Withdrawn
- 2010-03-25 KR KR1020187027407A patent/KR20180108883A/ko not_active Ceased
- 2010-03-25 NZ NZ595294A patent/NZ595294A/xx not_active IP Right Cessation
- 2010-03-25 CA CA2756065A patent/CA2756065A1/en not_active Abandoned
- 2010-03-25 CN CN2010800229237A patent/CN102497865A/zh active Pending
- 2010-03-25 BR BRPI1012324A patent/BRPI1012324A2/pt not_active Application Discontinuation
- 2010-03-25 JP JP2012502224A patent/JP2012521997A/ja active Pending
- 2010-03-25 WO PCT/US2010/028584 patent/WO2010111449A1/en not_active Ceased
- 2010-03-25 KR KR1020167027799A patent/KR20160120800A/ko not_active Withdrawn
- 2010-03-25 MX MX2011009901A patent/MX2011009901A/es not_active Application Discontinuation
- 2010-03-25 EP EP10723400.7A patent/EP2411013B1/en active Active
- 2010-03-25 KR KR1020177014845A patent/KR20170064556A/ko not_active Ceased
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2011
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2014
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- 2014-09-09 JP JP2014183177A patent/JP2015007117A/ja active Pending
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2016
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2018
- 2018-08-03 AU AU2018211329A patent/AU2018211329A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| KR20120006998A (ko) | 2012-01-19 |
| US20100247606A1 (en) | 2010-09-30 |
| WO2010111449A1 (en) | 2010-09-30 |
| RU2011140433A (ru) | 2013-04-27 |
| NZ595294A (en) | 2013-11-29 |
| EP2411013B1 (en) | 2020-08-19 |
| JP2012521997A (ja) | 2012-09-20 |
| RU2014133501A (ru) | 2016-03-10 |
| BRPI1012324A2 (pt) | 2016-03-15 |
| KR20170064556A (ko) | 2017-06-09 |
| IL215205A0 (en) | 2011-12-29 |
| AU2016231616A1 (en) | 2016-10-20 |
| CN102497865A (zh) | 2012-06-13 |
| KR20160120800A (ko) | 2016-10-18 |
| EP2411013A1 (en) | 2012-02-01 |
| RU2664686C2 (ru) | 2018-08-21 |
| KR20180108883A (ko) | 2018-10-04 |
| CA2756065A1 (en) | 2010-09-30 |
| JP2015007117A (ja) | 2015-01-15 |
| AU2010229891A1 (en) | 2011-10-20 |
| AU2018211329A1 (en) | 2018-08-23 |
| RU2532333C2 (ru) | 2014-11-10 |
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| Date | Code | Title | Description |
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| FA | Abandonment or withdrawal |