MX2010001368A - Forma cristalina de la sal diclorhidrato de ((1s)-1-(((2s)-2-(5-(4 ´-(2-((2s)-1-((2s)-2-((metoxicarbonil) amino)-3-metilbutanoil)-2-p irrolidinil)-1h-imidazol-5-il)-4-bifenilil)-1h-imidazol-2-il)-1-p irrolidinil) carbonil)-2-metilpropil)carbamato de - Google Patents

Forma cristalina de la sal diclorhidrato de ((1s)-1-(((2s)-2-(5-(4 ´-(2-((2s)-1-((2s)-2-((metoxicarbonil) amino)-3-metilbutanoil)-2-p irrolidinil)-1h-imidazol-5-il)-4-bifenilil)-1h-imidazol-2-il)-1-p irrolidinil) carbonil)-2-metilpropil)carbamato de

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Publication number
MX2010001368A
MX2010001368A MX2010001368A MX2010001368A MX2010001368A MX 2010001368 A MX2010001368 A MX 2010001368A MX 2010001368 A MX2010001368 A MX 2010001368A MX 2010001368 A MX2010001368 A MX 2010001368A MX 2010001368 A MX2010001368 A MX 2010001368A
Authority
MX
Mexico
Prior art keywords
imidazol
pyrrolidinyl
crystalline form
methylbutanoyl
biphenylyl
Prior art date
Application number
MX2010001368A
Other languages
English (en)
Spanish (es)
Inventor
Soojin Kim
Qi Gao
Fukang Yang
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39739413&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2010001368(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of MX2010001368A publication Critical patent/MX2010001368A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
MX2010001368A 2007-08-08 2008-07-31 Forma cristalina de la sal diclorhidrato de ((1s)-1-(((2s)-2-(5-(4 ´-(2-((2s)-1-((2s)-2-((metoxicarbonil) amino)-3-metilbutanoil)-2-p irrolidinil)-1h-imidazol-5-il)-4-bifenilil)-1h-imidazol-2-il)-1-p irrolidinil) carbonil)-2-metilpropil)carbamato de MX2010001368A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US95459207P 2007-08-08 2007-08-08
PCT/US2008/071734 WO2009020828A1 (en) 2007-08-08 2008-07-31 Crystalline form of methyl ((1s)-1-(((2s)-2-(5-(4'-(2-((2s)-1-((2s)-2-((methoxycarbonyl)amino)-3-methylbutanoyl)-2-pyrrolidinyl)-1h-imidazol-5-yl)-4-biphenylyl)-1h-imidazol-2-yl)-1-pyrrolidinyl)carbonyl)-2-methylpropyl)carbamate dihydrochloride salt

Publications (1)

Publication Number Publication Date
MX2010001368A true MX2010001368A (es) 2010-03-01

Family

ID=39739413

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2010001368A MX2010001368A (es) 2007-08-08 2008-07-31 Forma cristalina de la sal diclorhidrato de ((1s)-1-(((2s)-2-(5-(4 ´-(2-((2s)-1-((2s)-2-((metoxicarbonil) amino)-3-metilbutanoil)-2-p irrolidinil)-1h-imidazol-5-il)-4-bifenilil)-1h-imidazol-2-il)-1-p irrolidinil) carbonil)-2-metilpropil)carbamato de

Country Status (20)

Country Link
US (1) US8629171B2 (OSRAM)
EP (1) EP2183244B1 (OSRAM)
JP (1) JP5244179B2 (OSRAM)
KR (1) KR101508022B1 (OSRAM)
CN (1) CN101778840B (OSRAM)
AR (2) AR070016A1 (OSRAM)
AU (1) AU2008284100B2 (OSRAM)
BR (1) BRPI0815142B8 (OSRAM)
CA (1) CA2695729C (OSRAM)
CL (1) CL2008002354A1 (OSRAM)
CO (1) CO6160327A2 (OSRAM)
EA (1) EA018152B1 (OSRAM)
ES (1) ES2402791T3 (OSRAM)
IL (1) IL203684A (OSRAM)
MX (1) MX2010001368A (OSRAM)
NZ (1) NZ583148A (OSRAM)
PE (1) PE20090940A1 (OSRAM)
TW (1) TWI359813B (OSRAM)
WO (1) WO2009020828A1 (OSRAM)
ZA (1) ZA201000843B (OSRAM)

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JP2010535785A (ja) 2010-11-25
JP5244179B2 (ja) 2013-07-24
PE20090940A1 (es) 2009-07-13
EA201000196A1 (ru) 2010-06-30
ZA201000843B (en) 2011-04-28
AR104566A2 (es) 2017-08-02
TW200911790A (en) 2009-03-16
CN101778840A (zh) 2010-07-14
CO6160327A2 (es) 2010-05-20
US20090041716A1 (en) 2009-02-12
US8629171B2 (en) 2014-01-14
BRPI0815142A2 (pt) 2015-02-03
CL2008002354A1 (es) 2009-01-02
IL203684A (en) 2014-12-31
HK1144089A1 (en) 2011-01-28
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CA2695729A1 (en) 2009-02-12
BRPI0815142B8 (pt) 2021-05-25
CN101778840B (zh) 2013-11-13
AU2008284100B2 (en) 2014-01-16
CA2695729C (en) 2015-03-31
KR101508022B1 (ko) 2015-04-08
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EA018152B1 (ru) 2013-05-30
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AR070016A1 (es) 2010-03-10
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