MEP24508A - Derivati 1-fenilsulfonil-1,3-dihidro-2x-indol-2-ona, njihovo dobijanje i primjena u terapiji - Google Patents

Derivati 1-fenilsulfonil-1,3-dihidro-2x-indol-2-ona, njihovo dobijanje i primjena u terapiji

Info

Publication number
MEP24508A
MEP24508A MEP-245/08A MEP24508A MEP24508A ME P24508 A MEP24508 A ME P24508A ME P24508 A MEP24508 A ME P24508A ME P24508 A MEP24508 A ME P24508A
Authority
ME
Montenegro
Prior art keywords
preparation
phenylsulfonyl
indole
dihydro
derivatives
Prior art date
Application number
MEP-245/08A
Other languages
English (en)
Inventor
Malta Alain Di
Georges Garcia
Richard Roux
Bruno Schoentjes
Gal Claudine Serradeil-Le
Bernard Tonnerre
Jean Wagnon
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of MEP24508A publication Critical patent/MEP24508A/bs

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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Abstract

Ovaj pronalazak se odnosi na jedinjenja formule (I) kao i na njihove adicione soli sa kisjelinama ili organski m kisjelinama, njihove solvate i-ili njihove hidrate, koji pokazuju afi nitet i selekti vnost prema receptorima arginin-vazopresina V1b i/ili receptorima ocitocina, a pored toga, i na neka jedinjenja sa afi nitetom prema receptorima V1a. Ovaj pronalazak se takođe odnosi na postupak za njihovo dobijanje, intermedijama jedinjenja formule (IV), koja su korisna za njihovo dobijanje, na farmaceutske preparate koji ih sadrže i na njihovu upotrebu za dobijanje medikamenata.
MEP-245/08A 2001-07-17 2002-07-15 Derivati 1-fenilsulfonil-1,3-dihidro-2x-indol-2-ona, njihovo dobijanje i primjena u terapiji MEP24508A (bs)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0110359A FR2827604B1 (fr) 2001-07-17 2001-07-17 Nouveaux derives de 1-phenylsulfonyl-1,3-dihydro-2h-indol-2- one, un procede pour leur preparation et les compositions pharmaceutiques en contenant
PCT/FR2002/002500 WO2003008407A2 (fr) 2001-07-17 2002-07-15 Derives de 1-phenylsulfonyl-1,3-dihydro-2h-indol-2-one, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
MEP24508A true MEP24508A (bs) 2010-10-10

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MEP-245/08A MEP24508A (bs) 2001-07-17 2002-07-15 Derivati 1-fenilsulfonil-1,3-dihidro-2x-indol-2-ona, njihovo dobijanje i primjena u terapiji

Country Status (32)

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US (1) US7119086B2 (bs)
EP (1) EP1419150B1 (bs)
JP (1) JP4262088B2 (bs)
KR (1) KR20040017325A (bs)
CN (1) CN1224623C (bs)
AR (1) AR034792A1 (bs)
AT (1) ATE294171T1 (bs)
AU (1) AU2002340999B2 (bs)
BR (1) BR0211284A (bs)
CA (1) CA2450437A1 (bs)
CO (1) CO5550440A2 (bs)
DE (1) DE60203917T2 (bs)
DK (1) DK1419150T3 (bs)
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MA27049A1 (fr) 2004-12-20
WO2003008407A3 (fr) 2003-10-16
CA2450437A1 (en) 2003-01-30
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