RS204A - Phenylsulfonyl-1,3-dihydro-2h-indole-2- one derivatives,their preparation and their therapeutic use - Google Patents

Phenylsulfonyl-1,3-dihydro-2h-indole-2- one derivatives,their preparation and their therapeutic use

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Publication number
RS204A
RS204A YU204A YUP204A RS204A RS 204 A RS204 A RS 204A YU 204 A YU204 A YU 204A YU P204 A YUP204 A YU P204A RS 204 A RS204 A RS 204A
Authority
RS
Serbia
Prior art keywords
preparation
phenylsulfonyl
indole
dihydro
derivatives
Prior art date
Application number
YU204A
Other languages
Serbian (sr)
Inventor
Alain Di Malta
Georges Garcia
Richard Roux
Bruno Schoentjes
Gal Claudine Serradeil-Le
Bernard Tonnerre
Jean Wagnon
Original Assignee
Sanofi-Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi-Aventis filed Critical Sanofi-Aventis
Publication of RS204A publication Critical patent/RS204A/en

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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Abstract

The invention concerns compounds of formula (I), as well as their addition salts with acids or organic salts, their solvates and/or hydrate(s), exhibiting affinity and selectivity for arginine-vasopressin V1b receptors and/or for ocytocin receptors, and further, for certain compounds an affinity for V1a receptors. The invention also concerns the method for preparing them, intermediate compounds of formula (IV) useful for their preparation, pharmaceutical compositions containing them and their use for preparing medicines.
YU204A 2001-07-17 2002-07-15 Phenylsulfonyl-1,3-dihydro-2h-indole-2- one derivatives,their preparation and their therapeutic use RS204A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0110359A FR2827604B1 (en) 2001-07-17 2001-07-17 NOVEL 1-PHENYLSULFONYL-1,3-DIHYDRO-2H-INDOL-2- ONE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
PCT/FR2002/002500 WO2003008407A2 (en) 2001-07-17 2002-07-15 Phenylsulfonyl-1,3-dihydro-2h-indole-2-one derivatives, their preparation and their therapeutic use

Publications (1)

Publication Number Publication Date
RS204A true RS204A (en) 2006-12-15

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Family Applications (1)

Application Number Title Priority Date Filing Date
YU204A RS204A (en) 2001-07-17 2002-07-15 Phenylsulfonyl-1,3-dihydro-2h-indole-2- one derivatives,their preparation and their therapeutic use

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US (1) US7119086B2 (en)
EP (1) EP1419150B1 (en)
JP (1) JP4262088B2 (en)
KR (1) KR20040017325A (en)
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AR (1) AR034792A1 (en)
AT (1) ATE294171T1 (en)
AU (1) AU2002340999B2 (en)
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CO (1) CO5550440A2 (en)
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DK (1) DK1419150T3 (en)
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HR (1) HRP20040027A2 (en)
HU (1) HUP0401461A3 (en)
IL (1) IL159275A0 (en)
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MA (1) MA27049A1 (en)
ME (1) MEP24508A (en)
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NO (1) NO20040219L (en)
NZ (1) NZ530144A (en)
PL (1) PL366829A1 (en)
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