MA44225A - Sulfonylurées et composés apparentés et leur utilisation - Google Patents
Sulfonylurées et composés apparentés et leur utilisationInfo
- Publication number
- MA44225A MA44225A MA044225A MA44225A MA44225A MA 44225 A MA44225 A MA 44225A MA 044225 A MA044225 A MA 044225A MA 44225 A MA44225 A MA 44225A MA 44225 A MA44225 A MA 44225A
- Authority
- MA
- Morocco
- Prior art keywords
- sulphonylurides
- related compounds
- compounds
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07—ORGANIC CHEMISTRY
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- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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- A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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US10538487B2 (en) | 2015-02-16 | 2020-01-21 | The University Of Queensland | Sulfonylureas and related compounds and use of same |
BR112018016671A2 (pt) | 2016-02-16 | 2018-12-26 | The University Of Queensland | sulfonilureias e compostos relacionados e uso do mesmo |
EP4364794A3 (fr) | 2016-09-06 | 2024-07-24 | Axsome Malta Ltd. | Forme solvatee de (r)-2-amino-3-phenylpropyl carbamate |
CR20190356A (es) | 2017-01-23 | 2019-11-20 | Genentech Inc | Compuestos químicos como inhibidores de la actividad de la interleuquina-1 |
US11840543B2 (en) | 2017-05-24 | 2023-12-12 | The University Of Queensland | Compounds and uses |
US11370776B2 (en) | 2017-07-07 | 2022-06-28 | Inflazome Limited | Sulfonylureas and sulfonylthioureas as NLRP3 inhibitors |
HRP20220195T1 (hr) | 2017-07-07 | 2022-04-15 | Inflazome Limited | Novi spojevi sulfonamid karboksamida |
US11926600B2 (en) | 2017-08-15 | 2024-03-12 | Inflazome Limited | Sulfonylureas and sulfonylthioureas as NLRP3 inhibitors |
WO2019034692A1 (fr) * | 2017-08-15 | 2019-02-21 | Inflazome Limited | Sulfonylurées et sulfonylthiourées en tant qu'inhibiteurs de nlrp3 |
JP2020531453A (ja) | 2017-08-15 | 2020-11-05 | インフレイゾーム リミテッド | Nlrp3阻害剤としてのスルホニルウレアおよびスルホニルチオウレア |
US11518739B2 (en) | 2017-08-15 | 2022-12-06 | Inflazome Limited | Sulfonamide carboxamide compounds |
JP2020531448A (ja) | 2017-08-15 | 2020-11-05 | インフレイゾーム リミテッド | 新規なスルホンアミドカルボキサミド化合物 |
JP6984818B2 (ja) * | 2017-09-01 | 2021-12-22 | 学校法人近畿大学 | ゼルンボン誘導化合物と癌細胞増殖抑制剤およびそれらの製造方法 |
US11623922B2 (en) | 2017-10-03 | 2023-04-11 | Inflazome Limited | Compounds |
EP3707134A1 (fr) * | 2017-11-09 | 2020-09-16 | Inflazome Limited | Nouveaux composés de sulfonamide carboxamide |
GB201721185D0 (en) * | 2017-12-18 | 2018-01-31 | Nodthera Ltd | Sulphonyl urea derivatives |
WO2019166633A1 (fr) | 2018-03-02 | 2019-09-06 | Inflazome Limited | Dérivés de sulfonamide utilisés en tant qu'inhibiteurs de nlrp3 |
WO2019166632A1 (fr) | 2018-03-02 | 2019-09-06 | Inflazome Limited | Nouveaux composés |
WO2019166619A1 (fr) * | 2018-03-02 | 2019-09-06 | Inflazome Limited | Nouveaux composés |
US11884645B2 (en) | 2018-03-02 | 2024-01-30 | Inflazome Limited | Sulfonyl acetamides as NLRP3 inhibitors |
WO2019166629A1 (fr) | 2018-03-02 | 2019-09-06 | Inflazome Limited | Nouveaux composés |
GB201803393D0 (en) | 2018-03-02 | 2018-04-18 | Inflazome Ltd | Novel compounds |
WO2019166627A1 (fr) | 2018-03-02 | 2019-09-06 | Inflazome Limited | Nouveaux composés |
GB201803394D0 (en) | 2018-03-02 | 2018-04-18 | Inflazome Ltd | Novel compounds |
GB201806578D0 (en) | 2018-04-23 | 2018-06-06 | Inflazome Ltd | Novel compound |
CA3099080A1 (fr) | 2018-05-04 | 2019-11-07 | Inflazome Limited | Nouveaux composes |
CN108404117B (zh) * | 2018-05-29 | 2020-06-30 | 广东龙帆生物科技有限公司 | 核苷酸结合寡聚化结构域样受体蛋白在治疗寨卡病毒感染药物中的应用 |
EP3823726A1 (fr) * | 2018-07-20 | 2021-05-26 | F. Hoffmann-La Roche SA | Composés de sulfonylurée en tant qu'inhibiteurs de l'activité de l'interleukine 1 |
GB201902327D0 (en) | 2019-02-20 | 2019-04-03 | Inflazome Ltd | Novel compounds |
CR20210139A (es) * | 2018-08-15 | 2021-06-24 | Inflazome Ltd | Compuestos de sulfonamidaurea novedosos |
GB201819083D0 (en) | 2018-11-23 | 2019-01-09 | Inflazome Ltd | Novel compounds |
JP7488267B2 (ja) | 2019-01-14 | 2024-05-21 | ザイダス・ライフサイエンシーズ・リミテッド | 新規な置換スルホニル尿素誘導体 |
BR112021014389A2 (pt) * | 2019-01-25 | 2021-09-28 | NodThera Limited | Derivados de carbamato e usos dos mesmos |
GB201905265D0 (en) | 2019-04-12 | 2019-05-29 | Inflazome Ltd | Inflammasome inhibition |
US12054461B2 (en) | 2019-06-12 | 2024-08-06 | NodThera Limited | Sulfonylurea derivatives and uses thereof |
WO2020249664A1 (fr) * | 2019-06-12 | 2020-12-17 | NodThera Limited | Dérivés de sulfonylurée et leurs utilisations |
US20220267300A1 (en) * | 2019-06-12 | 2022-08-25 | NodThera Limited | Sulfonamide derivatives and uses thereof |
WO2020254697A1 (fr) | 2019-06-21 | 2020-12-24 | Ac Immune Sa | 1,2-thiazoles et 1,2 thiazines fusionnés qui agissent en tant que modulateurs de nl3p3 |
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-
2017
- 2017-02-16 BR BR112018016671A patent/BR112018016671A2/pt not_active Application Discontinuation
- 2017-02-16 US US15/999,424 patent/US11858922B2/en active Active
- 2017-02-16 EP EP17705416.0A patent/EP3416948B1/fr active Active
- 2017-02-16 WO PCT/EP2017/053498 patent/WO2017140778A1/fr active Application Filing
- 2017-02-16 CA CA3014487A patent/CA3014487A1/fr not_active Abandoned
- 2017-02-16 KR KR1020187026790A patent/KR20180133244A/ko unknown
- 2017-02-16 SG SG11201806745RA patent/SG11201806745RA/en unknown
- 2017-02-16 CN CN201780022601.4A patent/CN109071454B/zh active Active
- 2017-02-16 AU AU2017219204A patent/AU2017219204A1/en not_active Abandoned
- 2017-02-16 JP JP2018543108A patent/JP2019512009A/ja active Pending
- 2017-02-16 MA MA044225A patent/MA44225A/fr unknown
- 2017-02-16 MX MX2018009840A patent/MX2018009840A/es unknown
- 2017-08-15 UY UY0001037362A patent/UY37362A/es not_active Application Discontinuation
- 2017-08-15 AR ARP170102277A patent/AR109348A1/es unknown
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2018
- 2018-08-07 IL IL261035A patent/IL261035A/en unknown
- 2018-12-27 HK HK18116654.3A patent/HK1257569A1/zh unknown
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CA3014487A1 (fr) | 2017-08-24 |
EP3416948A1 (fr) | 2018-12-26 |
AU2017219204A1 (en) | 2018-08-23 |
IL261035A (en) | 2018-10-31 |
UY37362A (es) | 2018-09-28 |
SG11201806745RA (en) | 2018-09-27 |
US11858922B2 (en) | 2024-01-02 |
CN109071454A (zh) | 2018-12-21 |
HK1257569A1 (zh) | 2019-10-25 |
MX2018009840A (es) | 2019-01-21 |
US20200299284A1 (en) | 2020-09-24 |
EP3416948B1 (fr) | 2024-07-24 |
JP2019512009A (ja) | 2019-05-09 |
AR109348A1 (es) | 2018-11-21 |
WO2017140778A1 (fr) | 2017-08-24 |
EP3416948C0 (fr) | 2024-07-24 |
KR20180133244A (ko) | 2018-12-13 |
CN109071454B (zh) | 2023-02-17 |
BR112018016671A2 (pt) | 2018-12-26 |
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