MA31289B1 - Derives de thiazolidine - Google Patents

Derives de thiazolidine

Info

Publication number
MA31289B1
MA31289B1 MA32243A MA32243A MA31289B1 MA 31289 B1 MA31289 B1 MA 31289B1 MA 32243 A MA32243 A MA 32243A MA 32243 A MA32243 A MA 32243A MA 31289 B1 MA31289 B1 MA 31289B1
Authority
MA
Morocco
Prior art keywords
thiazolidine derivatives
derivatives
thiazolidine
medicaments
antagonists
Prior art date
Application number
MA32243A
Other languages
Arabic (ar)
English (en)
Inventor
Hamed Aissaoui
Christoph Boss
Markus Gude
Ralf Koberstein
Thierry Sifferlen
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of MA31289B1 publication Critical patent/MA31289B1/fr

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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
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  • Anesthesiology (AREA)
  • Psychology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Toxicology (AREA)
  • Emergency Medicine (AREA)

Abstract

L'invention porte sur de nouveaux dérivés de thiazolidine de la formule (i), dans laquelle a et r1 sont tels que décrits dans la description, et sur leur utilisation comme médicaments, notamment comme antagonistes du récepteur de l'orexine.
MA32243A 2007-03-26 2009-10-02 Derives de thiazolidine MA31289B1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IB2007051048 2007-03-26
IB2008050620 2008-02-21
PCT/IB2008/051110 WO2008117241A2 (fr) 2007-03-26 2008-03-25 Dérivés de thiazolidine

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MA31289B1 true MA31289B1 (fr) 2010-04-01

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US (1) US8236964B2 (fr)
EP (1) EP2125760A2 (fr)
JP (1) JP2010522737A (fr)
KR (1) KR20090125195A (fr)
CN (1) CN101641342B (fr)
AR (1) AR065822A1 (fr)
AU (1) AU2008231441A1 (fr)
BR (1) BRPI0808504A2 (fr)
CA (1) CA2677991A1 (fr)
CL (1) CL2008000836A1 (fr)
IL (1) IL201112A0 (fr)
MA (1) MA31289B1 (fr)
MX (1) MX2009009690A (fr)
NO (1) NO20093200L (fr)
RU (1) RU2009139285A (fr)
TW (1) TW200901988A (fr)
WO (1) WO2008117241A2 (fr)

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Publication number Publication date
CA2677991A1 (fr) 2008-10-02
WO2008117241A3 (fr) 2008-12-31
US20100113531A1 (en) 2010-05-06
CN101641342A (zh) 2010-02-03
MX2009009690A (es) 2009-12-14
IL201112A0 (en) 2010-05-17
AR065822A1 (es) 2009-07-01
EP2125760A2 (fr) 2009-12-02
AU2008231441A1 (en) 2008-10-02
BRPI0808504A2 (pt) 2014-08-19
US8236964B2 (en) 2012-08-07
CN101641342B (zh) 2012-10-03
JP2010522737A (ja) 2010-07-08
NO20093200L (no) 2009-10-23
TW200901988A (en) 2009-01-16
RU2009139285A (ru) 2011-05-10
WO2008117241A2 (fr) 2008-10-02
KR20090125195A (ko) 2009-12-03
CL2008000836A1 (es) 2008-11-07

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