MA28045A1 - Solvat acetonique du dimethoxy docetaxel et son procede de preparation - Google Patents

Solvat acetonique du dimethoxy docetaxel et son procede de preparation

Info

Publication number
MA28045A1
MA28045A1 MA28881A MA28881A MA28045A1 MA 28045 A1 MA28045 A1 MA 28045A1 MA 28881 A MA28881 A MA 28881A MA 28881 A MA28881 A MA 28881A MA 28045 A1 MA28045 A1 MA 28045A1
Authority
MA
Morocco
Prior art keywords
acetonic
solvat
preparing
same
dimethoxy
Prior art date
Application number
MA28881A
Other languages
English (en)
French (fr)
Inventor
Eric Didier
Marc-Antoine Perrin
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34224354&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA28045(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of MA28045A1 publication Critical patent/MA28045A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Epoxy Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
MA28881A 2003-09-19 2006-03-17 Solvat acetonique du dimethoxy docetaxel et son procede de preparation MA28045A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0311016A FR2859996B1 (fr) 2003-09-19 2003-09-19 Solvat acetonique du dimethoxy docetaxel et son procede de preparation

Publications (1)

Publication Number Publication Date
MA28045A1 true MA28045A1 (fr) 2006-07-03

Family

ID=34224354

Family Applications (1)

Application Number Title Priority Date Filing Date
MA28881A MA28045A1 (fr) 2003-09-19 2006-03-17 Solvat acetonique du dimethoxy docetaxel et son procede de preparation

Country Status (37)

Country Link
US (1) US7241907B2 (OSRAM)
EP (1) EP1667986B1 (OSRAM)
JP (1) JP5010279B2 (OSRAM)
KR (1) KR101123588B1 (OSRAM)
CN (1) CN100429207C (OSRAM)
AR (1) AR045667A1 (OSRAM)
AU (1) AU2004274212B2 (OSRAM)
BE (1) BE2013C036I2 (OSRAM)
BR (1) BRPI0414492A8 (OSRAM)
CA (1) CA2539309A1 (OSRAM)
CR (1) CR8292A (OSRAM)
CY (2) CY1114575T1 (OSRAM)
DK (1) DK1667986T3 (OSRAM)
ES (1) ES2403149T4 (OSRAM)
FR (2) FR2859996B1 (OSRAM)
HR (1) HRP20130322T1 (OSRAM)
HU (1) HUS1300025I1 (OSRAM)
IL (1) IL174240A (OSRAM)
LU (1) LU92172I2 (OSRAM)
MA (1) MA28045A1 (OSRAM)
ME (2) MEP11708A (OSRAM)
MX (1) MXPA06002639A (OSRAM)
MY (1) MY136668A (OSRAM)
NO (2) NO335997B1 (OSRAM)
NZ (1) NZ545835A (OSRAM)
PA (1) PA8612401A1 (OSRAM)
PE (1) PE20050870A1 (OSRAM)
PL (1) PL1667986T3 (OSRAM)
PT (1) PT1667986E (OSRAM)
RS (2) RS54614B1 (OSRAM)
RU (1) RU2342373C2 (OSRAM)
SI (1) SI1667986T1 (OSRAM)
TN (1) TNSN06086A1 (OSRAM)
TW (1) TWI382022B (OSRAM)
UA (1) UA87115C2 (OSRAM)
WO (1) WO2005028462A1 (OSRAM)
ZA (1) ZA200602255B (OSRAM)

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TWI526437B (zh) * 2011-09-09 2016-03-21 台灣神隆股份有限公司 卡巴他賽之結晶型
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DE112012004569T5 (de) 2011-11-01 2014-08-14 Fresenius Kabi Oncology Ltd. Amorphe Form von Cabazitaxel und Verfahren zum Herstellen davon
ES2716799T3 (es) * 2011-11-28 2019-06-17 Fresenius Kabi Oncology Ltd Forma cristalina de cabazitaxel y proceso para la preparación de la misma
EP2791122B1 (en) 2011-12-13 2019-01-23 Aventis Pharma S.A. Crystalline form of cabazitaxel and process for preparing the same
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CN102675257B (zh) * 2012-05-10 2014-07-02 上海金和生物技术有限公司 一种卡巴他赛晶体及其制备方法
CN102746258B (zh) 2012-07-25 2015-02-04 重庆泰濠制药有限公司 卡巴他赛的结晶形式及其制备方法
US9012665B2 (en) 2012-07-31 2015-04-21 Yung Shin Pharm. Ind. Co., Ltd. Amorphous cabazitaxel
US9198969B2 (en) 2012-08-15 2015-12-01 Yung Shin Pharm. Ind. Co., Ltd. Stable pharmaceutical formulation of cabazitaxel
CN103664836B (zh) * 2012-09-20 2016-04-20 齐鲁制药有限公司 7β,10β-二甲氧基多西紫杉醇氘代丙酮合物的晶型A及其制备方法
WO2014055493A1 (en) 2012-10-02 2014-04-10 Cerulean Pharma Inc. Methods and systems for polymer precipitation and generation of particles
CN103804323A (zh) * 2012-11-14 2014-05-21 上海希迈医药科技有限公司 一种卡巴他赛溶剂化物及其制备方法和应用
CN103058960B (zh) * 2012-12-12 2014-12-10 江苏奥赛康药业股份有限公司 卡巴他赛多晶型形式及其制备方法
EP2743264A1 (en) 2012-12-13 2014-06-18 INDENA S.p.A. New crystalline form of cabazitaxel, process for the preparation and pharmaceutical compositions thereof
CN103910698B (zh) * 2012-12-30 2016-01-20 上海医药工业研究院 卡巴他赛丙酮合物及其结晶
CN103910696B (zh) * 2012-12-30 2016-01-20 上海医药工业研究院 卡巴他赛异丙醚合物及其结晶
EP2777691A1 (en) 2013-03-14 2014-09-17 Pharmachemie B.V. Taxoid - Purification of Liquid Excipients
EP2815749A1 (en) 2013-06-20 2014-12-24 IP Gesellschaft für Management mbH Solid form of 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione having specified X-ray diffraction pattern
WO2015000165A1 (zh) * 2013-07-04 2015-01-08 北京新天宇科技开发有限公司 二甲氧基多西紫杉醇一丙酮化物的稳定转化物及其结晶形式、以及它们的制备方法
CN104277014A (zh) * 2013-07-04 2015-01-14 北京新天宇科技开发有限公司 二甲氧基多西紫杉醇一丙酮化物的稳定转化物及其结晶形式、以及它们的制备方法
EP2865674A1 (en) 2013-10-23 2015-04-29 INDENA S.p.A. Crystalline solvate forms of Cabazitaxel
EP2865675A1 (en) * 2013-10-23 2015-04-29 INDENA S.p.A. A crystalline anhydrous form of Cabazitaxel, process for the preparation and pharmaceutical compositions thereof
CN103601704B (zh) * 2013-11-22 2015-05-06 石家庄智恒医药科技有限公司 无定形卡巴他赛的制备
EP3247350B1 (en) 2015-01-12 2021-12-22 Emcure Pharmaceuticals Limited Liquid formulation of cabazitaxel
EP3258931B1 (en) 2015-02-17 2020-08-12 Erasmus University Medical Center Rotterdam Use of cabazitaxel in the treatment of prostate cancer
EP3093014A1 (en) * 2015-05-13 2016-11-16 Aventis Pharma S.A. Cabazitaxel and its use for treating cancer
US10188626B2 (en) 2015-11-03 2019-01-29 Cipla Limited Stabilized cabazitaxel formulations
EP3548487A4 (en) 2016-11-29 2020-04-29 Censa Pharmaceuticals Inc. POLYMORPHE SHAPE OF SEPIAPTERIN
JP7148533B2 (ja) 2016-11-29 2022-10-05 ピーティーシー セラピューティクス エムピー，インコーポレイテッド セピプテリン及びその塩の多形
BR112020003865A8 (pt) 2017-09-01 2022-08-16 Censa Pharmaceuticals Inc Composições farmacêuticas compreendendo sepiapterina e seus usos
CA3102105A1 (en) 2018-05-30 2019-12-05 Ptc Therapeutics Mp, Inc. Compositions and methods for increasing tetrahydrobiopterin plasma exposure
SI3801536T1 (sl) 2018-05-30 2024-12-31 Ptc Therapeutics Mp, Inc. Dajanje sepiapterina brez hrane za uporabo v postopku za zvišanje plazemske izpostavljenosti sepiapterinu
WO2020249507A1 (en) 2019-06-11 2020-12-17 Indena S.P.A. Anhydrous crystalline form of cabazitaxel, a process for its preparation and pharmaceutical compositions containing it
EP3797834A1 (en) 2019-09-25 2021-03-31 Sanofi Mature IP Cabazitaxel in mcrpc patients previously treated with docetaxel and who failed a prior androgen signaling targeted inhibitor agent
EP3808345A1 (en) 2019-10-15 2021-04-21 Sanofi Mature IP Cabazitaxel in mcrpc patients previously treated with docetaxel and who failed a prior androgen signaling targeted inhibitor agent

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Also Published As

Publication number Publication date
HUS1300025I1 (hu) 2016-08-29
KR20060072147A (ko) 2006-06-27
NO2015013I2 (no) 2015-04-22
PA8612401A1 (es) 2005-08-04
PL1667986T3 (pl) 2013-06-28
TWI382022B (zh) 2013-01-11
RU2006113122A (ru) 2006-08-27
NO2015013I1 (no) 2015-05-04
FR13C0037I2 (fr) 2015-11-20
CN100429207C (zh) 2008-10-29
RS54614B1 (sr) 2016-08-31
NO20061714L (no) 2006-04-19
CR8292A (es) 2008-10-15
AR045667A1 (es) 2005-11-02
ES2403149T3 (es) 2013-05-14
SI1667986T1 (sl) 2013-05-31
IL174240A0 (en) 2006-08-01
EP1667986B1 (fr) 2013-01-16
CY1114575T1 (el) 2016-10-05
US20050065138A1 (en) 2005-03-24
MY136668A (en) 2008-11-28
CA2539309A1 (fr) 2005-03-31
PT1667986E (pt) 2013-04-24
FR2859996A1 (fr) 2005-03-25
AU2004274212A1 (en) 2005-03-31
FR2859996B1 (fr) 2006-02-03
UA87115C2 (ru) 2009-06-25
BRPI0414492A (pt) 2006-11-14
ME00054B (me) 2011-02-10
US7241907B2 (en) 2007-07-10
HRP20130322T1 (en) 2013-07-31
DK1667986T3 (da) 2013-05-06
EP1667986A1 (fr) 2006-06-14
WO2005028462A1 (fr) 2005-03-31
JP5010279B2 (ja) 2012-08-29
PE20050870A1 (es) 2005-11-21
BRPI0414492A8 (pt) 2019-01-15
CY2013016I1 (el) 2018-01-10
MEP11708A (en) 2010-06-10
AU2004274212B2 (en) 2010-03-04
CN1849311A (zh) 2006-10-18
NO335997B1 (no) 2015-04-20
IL174240A (en) 2010-12-30
ES2403149T4 (es) 2013-06-24
FR13C0037I1 (fr) 2013-09-08
RS20060189A (sr) 2008-06-05
LU92172I2 (fr) 2013-05-21
CY2013016I2 (el) 2018-01-10
KR101123588B1 (ko) 2012-03-22
RU2342373C2 (ru) 2008-12-27
TNSN06086A1 (en) 2007-10-03
HK1093340A1 (zh) 2007-03-02
TW200524891A (en) 2005-08-01
ZA200602255B (en) 2007-07-25
MXPA06002639A (es) 2006-06-05
NZ545835A (en) 2009-10-30
JP2007505866A (ja) 2007-03-15
BE2013C036I2 (OSRAM) 2023-12-14
LU92172I9 (OSRAM) 2019-01-03

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