LU85191A1 - Nouveaux derives de la benzo(g)quinoleine,leur preparation et leur utilisation comme medicaments - Google Patents

Nouveaux derives de la benzo(g)quinoleine,leur preparation et leur utilisation comme medicaments Download PDF

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Publication number
LU85191A1
LU85191A1 LU85191A LU85191A LU85191A1 LU 85191 A1 LU85191 A1 LU 85191A1 LU 85191 A LU85191 A LU 85191A LU 85191 A LU85191 A LU 85191A LU 85191 A1 LU85191 A1 LU 85191A1
Authority
LU
Luxembourg
Prior art keywords
octahydro
trans
quinoline
benzo
hydroxy
Prior art date
Application number
LU85191A
Other languages
English (en)
French (fr)
Original Assignee
Sandoz Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Sa filed Critical Sandoz Sa
Publication of LU85191A1 publication Critical patent/LU85191A1/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • C07D221/06—Ring systems of three rings
    • C07D221/08—Aza-anthracenes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
LU85191A 1983-02-01 1984-01-31 Nouveaux derives de la benzo(g)quinoleine,leur preparation et leur utilisation comme medicaments LU85191A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH56083 1983-02-01
CH56083 1983-02-01

Publications (1)

Publication Number Publication Date
LU85191A1 true LU85191A1 (fr) 1984-10-24

Family

ID=4189841

Family Applications (1)

Application Number Title Priority Date Filing Date
LU85191A LU85191A1 (fr) 1983-02-01 1984-01-31 Nouveaux derives de la benzo(g)quinoleine,leur preparation et leur utilisation comme medicaments

Country Status (17)

Country Link
US (1) US4692453A (xx)
JP (1) JPS59144761A (xx)
AU (1) AU571482B2 (xx)
BE (1) BE898761A (xx)
DE (1) DE3402601A1 (xx)
DK (1) DK40984A (xx)
FR (1) FR2540112B1 (xx)
GB (1) GB2134515B (xx)
IE (1) IE56653B1 (xx)
IL (1) IL70845A (xx)
IT (1) IT1199056B (xx)
LU (1) LU85191A1 (xx)
NL (1) NL8400259A (xx)
NZ (1) NZ206981A (xx)
PH (1) PH22782A (xx)
SE (1) SE8400445L (xx)
ZA (1) ZA84757B (xx)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT393997B (de) * 1983-06-22 1992-01-10 Heidelberger Druckmasch Ag Vorrichtung zur entnahme von bedruckten bogen fuer deren begutachtung
DE69030665T2 (de) * 1989-07-13 1997-10-02 Pharmacia & Upjohn Co., Kalamazoo, Mich. (1,2n) und (3,2n)-karbozyklische-2-amino-tetralinderivate
US4939259A (en) * 1989-07-24 1990-07-03 Eli Lilly And Company 2-oxo-pyrido[2,3-g]quinoline derivatives
DE4114325A1 (de) * 1991-05-02 1992-11-05 Sandoz Ag Octahydrobenzo(g)chinolin, seine herstellung und verwendung
EP0586553A1 (en) * 1991-05-20 1994-03-16 The Upjohn Company Carboxamido-(3,2n)-carbocyclic-2-aminotetralin derivatives
US20090124651A1 (en) * 2007-08-31 2009-05-14 H. Lundbeck A/S Catecholamine derivatives and prodrugs thereof
JP2011525893A (ja) * 2008-06-27 2011-09-29 ハー・ルンドベック・アクチエゼルスカベット 新規のフェノールアミン類およびカテコールアミン類ならびにそのプロドラッグ
BR112019014981A2 (pt) 2017-11-24 2020-04-07 H Lundbeck As composto, sal farmaceuticamente aceitável, uso dos mesmos e composição farmacêutica
US11111263B2 (en) 2019-05-20 2021-09-07 H. Lundbeck A/S Process for the manufacture of (2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-(((4aR,10aR)-7-hydroxy-1-propyl-1,2,3,4,4a,5,10,10a-octahydrobenzo[g]quinolin-6-yl)oxy)tetrahydro-2H-pyran-2-carboxylic acid
US11104697B2 (en) 2019-05-20 2021-08-31 H. Lundbeck A/S Process for the manufacture of (2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-(((4AR,10AR)-7-hydroxy-1- propyl-1,2,3,4,4A,5,10,10A-octahydrobenzo[g]quinolin-6-yl)oxy)tetrahydro-2H-pyran-2-carboxylic acid
US11168056B2 (en) 2019-05-20 2021-11-09 H. Lundbeck A/S Process for the manufacturing of (6aR,10aR)-7-propyl-6,6a,7,8,9,10,10a,11-octahydro-[1,3]dioxolo[4′,5′:5,6]benzo[1,2-G]quinoline and (4aR,10aR)-1-propyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[G]quinoline-6,7-diol
US11130775B2 (en) 2019-05-20 2021-09-28 H. Lundbeck A/S Solid forms of (2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-(((4aR,10aR)-7-hydroxy-1-propyl-1,2,3,4,4A,5,10,10A-octahydrobenzo[g]quinolin-6-yl)oxy)tetrahydro-2H-pyran-2-carboxylic acid

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3839338A (en) * 1968-05-09 1974-10-01 W Michne 1,2,3,4,4A,5,10,10A-OCTAHYDROBENZO{8 g{9 QUINOLINES
US3639411A (en) * 1968-05-09 1972-02-01 Sterling Drug Inc 1-substituted-2-(phenyl or benzyl)-3- or 3 3 - piperidine(mono or dicarboxylic) acids and esters thereo fand octahydrobenzo(g) - quinolines and hexahydro-5h-inden (12-b)pyridines produced therefrom
US3898235A (en) * 1970-12-02 1975-08-05 Sterling Drug Inc Octahydrobenzo {8 g{9 {0 quinolines and hexahydroindeno {8 1,2,b{9 {0 pyridines
DE19575006I2 (de) * 1981-10-16 2003-01-09 Novartis Ag 1, 2, 3, 4a, 5, 10, 10a-Octahydrobenzo(g)chinolin-Derivate mit pharmazeutischer Wirkung

Also Published As

Publication number Publication date
NL8400259A (nl) 1984-09-03
SE8400445L (sv) 1984-08-02
GB2134515B (en) 1986-07-02
IE56653B1 (en) 1991-10-23
AU571482B2 (en) 1988-04-21
IL70845A (en) 1986-09-30
ZA84757B (en) 1985-09-25
PH22782A (en) 1988-12-12
IL70845A0 (en) 1984-05-31
GB2134515A (en) 1984-08-15
IT8447626A0 (it) 1984-02-01
IT1199056B (it) 1988-12-30
BE898761A (fr) 1984-07-26
DE3402601A1 (de) 1984-08-02
DK40984D0 (da) 1984-01-30
US4692453A (en) 1987-09-08
NZ206981A (en) 1987-03-31
SE8400445D0 (sv) 1984-01-30
GB8402358D0 (en) 1984-02-29
JPS59144761A (ja) 1984-08-18
DK40984A (da) 1984-08-02
FR2540112B1 (fr) 1986-08-29
AU2391184A (en) 1984-08-02
IE840209L (en) 1984-08-01
FR2540112A1 (fr) 1984-08-03

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