LT4329B - Išorinio vartojimo priešuždegiminis agentas - Google Patents
Išorinio vartojimo priešuždegiminis agentas Download PDFInfo
- Publication number
- LT4329B LT4329B LT97-100A LT97100A LT4329B LT 4329 B LT4329 B LT 4329B LT 97100 A LT97100 A LT 97100A LT 4329 B LT4329 B LT 4329B
- Authority
- LT
- Lithuania
- Prior art keywords
- nimesulide
- weight
- inflammatory agent
- component
- oil
- Prior art date
Links
- HYWYRSMBCFDLJT-UHFFFAOYSA-N nimesulide Chemical compound CS(=O)(=O)NC1=CC=C([N+]([O-])=O)C=C1OC1=CC=CC=C1 HYWYRSMBCFDLJT-UHFFFAOYSA-N 0.000 claims abstract description 67
- 229960000965 nimesulide Drugs 0.000 claims abstract description 66
- 229940121363 anti-inflammatory agent Drugs 0.000 claims abstract description 21
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- 239000004480 active ingredient Substances 0.000 claims abstract description 10
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- 238000002360 preparation method Methods 0.000 claims description 37
- -1 fatty acid ester Chemical class 0.000 claims description 17
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- 239000000194 fatty acid Substances 0.000 claims description 16
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- 239000000126 substance Substances 0.000 claims description 15
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- 238000010438 heat treatment Methods 0.000 claims description 11
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- LVTYICIALWPMFW-UHFFFAOYSA-N diisopropanolamine Chemical group CC(O)CNCC(C)O LVTYICIALWPMFW-UHFFFAOYSA-N 0.000 claims description 9
- 229940043276 diisopropanolamine Drugs 0.000 claims description 9
- XBRDBODLCHKXHI-UHFFFAOYSA-N epolamine Chemical compound OCCN1CCCC1 XBRDBODLCHKXHI-UHFFFAOYSA-N 0.000 claims description 9
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- 238000000926 separation method Methods 0.000 description 1
- 235000010234 sodium benzoate Nutrition 0.000 description 1
- 239000004299 sodium benzoate Substances 0.000 description 1
- 239000011780 sodium chloride Substances 0.000 description 1
- LUPNKHXLFSSUGS-UHFFFAOYSA-M sodium;2,2-dichloroacetate Chemical compound [Na+].[O-]C(=O)C(Cl)Cl LUPNKHXLFSSUGS-UHFFFAOYSA-M 0.000 description 1
- 230000003381 solubilizing effect Effects 0.000 description 1
- 229940032094 squalane Drugs 0.000 description 1
- 229940012831 stearyl alcohol Drugs 0.000 description 1
- 230000001629 suppression Effects 0.000 description 1
- TUNFSRHWOTWDNC-HKGQFRNVSA-N tetradecanoic acid Chemical compound CCCCCCCCCCCCC[14C](O)=O TUNFSRHWOTWDNC-HKGQFRNVSA-N 0.000 description 1
- OULAJFUGPPVRBK-UHFFFAOYSA-N tetratriacontyl alcohol Natural products CCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCO OULAJFUGPPVRBK-UHFFFAOYSA-N 0.000 description 1
- 239000012049 topical pharmaceutical composition Substances 0.000 description 1
- 235000015112 vegetable and seed oil Nutrition 0.000 description 1
- 235000019871 vegetable fat Nutrition 0.000 description 1
- 239000008158 vegetable oil Substances 0.000 description 1
- 238000005303 weighing Methods 0.000 description 1
- 239000000080 wetting agent Substances 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/18—Sulfonamides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Dermatology (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/JP1995/002045 WO1996011002A1 (en) | 1994-10-05 | 1995-10-05 | Antiinflammatory agent for external use |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| LT97100A LT97100A (en) | 1997-12-29 |
| LT4329B true LT4329B (lt) | 1998-04-27 |
Family
ID=14126349
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| LT97-100A LT4329B (lt) | 1995-10-05 | 1997-06-03 | Išorinio vartojimo priešuždegiminis agentas |
Country Status (17)
| Country | Link |
|---|---|
| BG (1) | BG63328B1 (cs) |
| CZ (1) | CZ288398B6 (cs) |
| EE (1) | EE03419B1 (cs) |
| FI (1) | FI118953B (cs) |
| HU (1) | HU224686B1 (cs) |
| IS (1) | IS2271B (cs) |
| LT (1) | LT4329B (cs) |
| LV (1) | LV11966B (cs) |
| NO (1) | NO315732B1 (cs) |
| NZ (1) | NZ327092A (cs) |
| PL (1) | PL183588B1 (cs) |
| RO (1) | RO116040B1 (cs) |
| RU (1) | RU2157683C2 (cs) |
| SI (1) | SI9620016B (cs) |
| SK (1) | SK282637B6 (cs) |
| TR (1) | TR199700409T1 (cs) |
| WO (1) | WO1997012608A1 (cs) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1289973B1 (it) * | 1997-02-25 | 1998-10-19 | Helsinn Healthcare Sa | Sistemi gelificati di nimesulide per uso topico |
| IT1291997B1 (it) * | 1997-05-26 | 1999-01-25 | Schiena Michele Giuseppe Di | Preparati-farmaceutici-topici-contenenti nimesulide |
| IT1308187B1 (it) * | 1999-02-16 | 2001-12-07 | Formenti Farmaceutici Spa | Composizioni farmaceutiche topiche a base di antiinfiammatori nonsteroidei. |
| RU2424811C2 (ru) * | 2009-04-02 | 2011-07-27 | Евгений Петрович Гребенников | Лекарственное средство для лечения псориаза |
| RU2657803C1 (ru) * | 2017-03-21 | 2018-06-15 | федеральное государственное бюджетное образовательное учреждение высшего образования "Алтайский государственный университет" | Средство, обладающее противовоспалительным и анальгезирующим действием |
Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3480597A (en) | 1967-03-01 | 1969-11-25 | Vasily Vladimirovich Korshak | Method for the production of polyarylates |
| JPS5835989A (ja) | 1981-08-28 | 1983-03-02 | Sanyo Electric Co Ltd | 非晶質光半導体装置 |
| JPS5850984A (ja) | 1981-09-24 | 1983-03-25 | 松下電工株式会社 | 電気カミソリ |
| JPH06502842A (ja) | 1990-05-22 | 1994-03-31 | パットファルム ホウルディング ソシエテ アノニム | ニメスリドとシクロデキストリンの包接化合物 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR206496A1 (es) * | 1972-07-03 | 1976-07-30 | Riker Laboratories Inc | Procedimiento para la preparacion de 2-fenoxi-4-nitro-alquil o haloalquilsulfonanilidas |
| JPS60209515A (ja) * | 1984-04-03 | 1985-10-22 | Hokuriku Seiyaku Co Ltd | 消炎鎮痛クリ−ム剤 |
| JPH01224328A (ja) * | 1988-03-01 | 1989-09-07 | Kao Corp | 鎮痒剤組成物 |
| JPH05310508A (ja) * | 1992-05-13 | 1993-11-22 | Kanebo Ltd | 皮膚外用剤組成物 |
| RU2007997C1 (ru) * | 1992-07-08 | 1994-02-28 | Леонидов Николай Борисович | Линимент метилурацила |
| BE1008307A3 (fr) * | 1994-06-16 | 1996-04-02 | Europharmaceuticals Sa | Sel de nimesulide hydrosoluble, solution aqueuse le contenant, sa preparation et son utilisation. |
-
1996
- 1996-04-01 HU HU9901126A patent/HU224686B1/hu not_active IP Right Cessation
- 1996-04-01 PL PL96320534A patent/PL183588B1/pl not_active IP Right Cessation
- 1996-04-01 RO RO97-01018A patent/RO116040B1/ro unknown
- 1996-04-01 CZ CZ19971703A patent/CZ288398B6/cs not_active IP Right Cessation
- 1996-04-01 NZ NZ327092A patent/NZ327092A/en unknown
- 1996-04-01 SI SI9620016A patent/SI9620016B/sl not_active IP Right Cessation
- 1996-04-01 SK SK704-97A patent/SK282637B6/sk not_active IP Right Cessation
- 1996-04-01 WO PCT/JP1996/000849 patent/WO1997012608A1/ja not_active Ceased
- 1996-04-01 EE EE9700123A patent/EE03419B1/xx not_active IP Right Cessation
- 1996-04-01 TR TR97/00409T patent/TR199700409T1/xx unknown
- 1996-04-01 RU RU97111164/14A patent/RU2157683C2/ru not_active IP Right Cessation
-
1997
- 1997-05-29 BG BG101526A patent/BG63328B1/bg unknown
- 1997-06-03 LT LT97-100A patent/LT4329B/lt not_active IP Right Cessation
- 1997-06-04 LV LVP-97-108A patent/LV11966B/en unknown
- 1997-06-04 IS IS4497A patent/IS2271B/is unknown
- 1997-06-04 FI FI972362A patent/FI118953B/fi active IP Right Grant
- 1997-06-04 NO NO19972537A patent/NO315732B1/no unknown
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3480597A (en) | 1967-03-01 | 1969-11-25 | Vasily Vladimirovich Korshak | Method for the production of polyarylates |
| JPS5835989A (ja) | 1981-08-28 | 1983-03-02 | Sanyo Electric Co Ltd | 非晶質光半導体装置 |
| JPS5850984A (ja) | 1981-09-24 | 1983-03-25 | 松下電工株式会社 | 電気カミソリ |
| JPH06502842A (ja) | 1990-05-22 | 1994-03-31 | パットファルム ホウルディング ソシエテ アノニム | ニメスリドとシクロデキストリンの包接化合物 |
Also Published As
| Publication number | Publication date |
|---|---|
| IS2271B (is) | 2007-07-15 |
| BG63328B1 (bg) | 2001-10-31 |
| LV11966A (lv) | 1998-02-20 |
| BG101526A (en) | 1998-01-30 |
| EE9700123A (et) | 1997-12-15 |
| NO972537L (no) | 1997-06-04 |
| RU2157683C2 (ru) | 2000-10-20 |
| FI972362L (fi) | 1997-07-25 |
| HU224686B1 (hu) | 2005-12-28 |
| LV11966B (en) | 1998-04-20 |
| PL183588B1 (pl) | 2002-06-28 |
| NO972537D0 (no) | 1997-06-04 |
| EE03419B1 (et) | 2001-06-15 |
| SI9620016B (sl) | 1999-06-30 |
| RO116040B1 (ro) | 2000-10-30 |
| WO1997012608A1 (fr) | 1997-04-10 |
| FI118953B (fi) | 2008-05-30 |
| CZ170397A3 (cs) | 1998-01-14 |
| CZ288398B6 (en) | 2001-06-13 |
| TR199700409T1 (xx) | 1999-08-23 |
| HUP9901126A3 (en) | 2000-08-28 |
| FI972362A0 (fi) | 1997-06-04 |
| IS4497A (is) | 1997-06-04 |
| HUP9901126A2 (hu) | 1999-08-30 |
| NZ327092A (en) | 1999-09-29 |
| SK282637B6 (sk) | 2002-10-08 |
| NO315732B1 (no) | 2003-10-20 |
| LT97100A (en) | 1997-12-29 |
| PL320534A1 (en) | 1997-10-13 |
| SI9620016A (en) | 1997-12-31 |
| SK70497A3 (en) | 1997-10-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM9A | Lapsed patents |
Effective date: 20090401 |