LT2436B - (3H) -IMIDAZO- (5,1-A) -1,2,3,5-TETRAZIN-4-ONO BACKGROUND OF THE INVENTION - Google Patents

(3H) -IMIDAZO- (5,1-A) -1,2,3,5-TETRAZIN-4-ONO BACKGROUND OF THE INVENTION

Info

Publication number
LT2436B
LT2436B LTRP1286A LTRP1286A LT2436B LT 2436 B LT2436 B LT 2436B LT RP1286 A LTRP1286 A LT RP1286A LT RP1286 A LTRP1286 A LT RP1286A LT 2436 B LT2436 B LT 2436B
Authority
LT
Lithuania
Prior art keywords
tetrazin
ono
imidazo
background
ono background
Prior art date
Application number
LTRP1286A
Other languages
Lithuanian (lt)
Inventor
Edward Lunt
Malcolm Francis Graham Stevens
Robert Stone
Kenneth Robert Harr Wooldridge
Original Assignee
May & Baker Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by May & Baker Ltd filed Critical May & Baker Ltd
Publication of LT2436B publication Critical patent/LT2436B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D407/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/04Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
LTRP1286A 1981-08-24 1993-09-29 (3H) -IMIDAZO- (5,1-A) -1,2,3,5-TETRAZIN-4-ONO BACKGROUND OF THE INVENTION LT2436B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8125791 1981-08-24

Publications (1)

Publication Number Publication Date
LT2436B true LT2436B (en) 1994-02-15

Family

ID=10524141

Family Applications (1)

Application Number Title Priority Date Filing Date
LTRP1286A LT2436B (en) 1981-08-24 1993-09-29 (3H) -IMIDAZO- (5,1-A) -1,2,3,5-TETRAZIN-4-ONO BACKGROUND OF THE INVENTION

Country Status (29)

Country Link
JP (1) JPS5843975A (en)
KR (1) KR890000094B1 (en)
AT (1) AT380256B (en)
AU (1) AU571430B2 (en)
BE (1) BE894175A (en)
CA (1) CA1197247A (en)
CH (1) CH655114A5 (en)
DE (2) DE3231255A1 (en)
DK (1) DK161147C (en)
ES (1) ES8400438A1 (en)
FI (1) FI73434C (en)
FR (1) FR2511679A1 (en)
GB (1) GB2104522B (en)
GE (1) GEP19960641B (en)
GR (1) GR76863B (en)
HU (1) HU186107B (en)
IE (1) IE53408B1 (en)
IL (1) IL66606A (en)
IT (1) IT1152505B (en)
LT (1) LT2436B (en)
LU (1) LU84347A1 (en)
LV (2) LV5511A3 (en)
NL (2) NL192739C (en)
NZ (1) NZ201668A (en)
OA (1) OA07174A (en)
SE (1) SE448543B (en)
SU (1) SU1447284A3 (en)
UA (1) UA5971A1 (en)
ZA (1) ZA826120B (en)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5260291A (en) * 1981-08-24 1993-11-09 Cancer Research Campaign Technology Limited Tetrazine derivatives
GB2125402B (en) * 1982-08-17 1985-11-13 May & Baker Ltd New tetrazine derivatives
FR2531958B1 (en) * 1982-08-17 1986-10-31 May & Baker Ltd NEW DERIVATIVES
US4517182A (en) * 1983-05-24 1985-05-14 Warner-Lambert Company 3-(Haloethyl)-4-oxopyrazolo-[5,1-d]-1,2,3,5-tetrazine-8-carboxamide composition
GB8616125D0 (en) * 1986-07-02 1986-08-06 May & Baker Ltd Compositions of matter
AU622330B2 (en) * 1989-06-23 1992-04-02 Takeda Chemical Industries Ltd. Condensed heterocyclic compounds having a nitrogen atom in the bridgehead for use as fungicides
BRPI0417117A (en) * 2003-12-30 2007-03-06 Chemagis Ltd crystallized temozolomide, crystallized temozolomide preparation process, pharmaceutical composition, method of producing medicament containing temozolomide and method of treating a medical condition for which thermozolomide is beneficial
US20090036435A1 (en) 2005-01-21 2009-02-05 Astex Therapeutics Limited Pharmaceutical Compounds
AR060635A1 (en) 2006-04-27 2008-07-02 Banyu Pharma Co Ltd DERIVATIVES OF 1,2-DIHIDRO-3H-PIRAZOLO [3,4-D] PIRIMIDIN-3-ONA, PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THEM AND THEIR USE IN THE TREATMENT OF CANCER
JP2008081492A (en) 2006-08-31 2008-04-10 Banyu Pharmaceut Co Ltd New aminopyridine derivative having aurora a selective inhibitory action
US8916552B2 (en) 2006-10-12 2014-12-23 Astex Therapeutics Limited Pharmaceutical combinations
EP2073807A1 (en) 2006-10-12 2009-07-01 Astex Therapeutics Limited Pharmaceutical combinations
CA2703489A1 (en) 2007-10-23 2009-04-30 Banyu Pharmaceutical Co., Ltd. Pyridone-substituted-dihydropyrazolopyrimidinone derivative
PE20091101A1 (en) * 2007-12-18 2009-07-26 Pharminox Ltd 3-SUBSTITUTED-4-OXO-3,4-DIHYDRO-IMIDAZO [5,1-d] [1,2,3,5-TETRACINE-8-CARBOXYL ACID AMIDES AND ITS USE
CA2744560A1 (en) * 2008-11-24 2010-05-27 Reliance Life Sciences Pvt. Ltd. Process for the preparation of tetrazine derivatives
EP2403339B1 (en) 2009-03-06 2017-01-18 Merck Sharp & Dohme Corp. Combination cancer therapy with an akt inhibitor and other anticancer agents
EP2445915B1 (en) 2009-06-23 2016-04-20 Pharminox Limited 3-substituted-8-substituted-3h imidazo[5,1-d][1,2,3,5-tetrazin-4-one compounds and their use
RU2462466C1 (en) * 2011-06-24 2012-09-27 Автономная Некоммерческая Организация "Научно-Исследовательский Центр Биотехнологии Антибиотиков И Других Биологически Активных Веществ "Биоан" Substituted azolo[1,2,4,5]tetrazines - inhibitors of antibacterial serine-threonine protein kinases
US20140271657A1 (en) 2011-10-12 2014-09-18 Children's Medical Center Corporation Combinatorial compositions and methods of treating hemoglobinopathies
CN109195593A (en) 2016-03-15 2019-01-11 奥莱松基因组股份有限公司 For treating the combination of the LSD1 inhibitor of solid tumor
KR101847342B1 (en) * 2017-05-08 2018-04-11 (주)센텍코리아 Wearable body fat burning measurement device

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2932305A1 (en) * 1979-08-09 1981-02-26 Basf Ag Pyrrolo-, pyrazolo-, imidazo- and thiazolo-tetrazin-4-one derivs. - prepd. from amino-azole cpds. by diazotisation and reaction with isocyanate

Also Published As

Publication number Publication date
GR76863B (en) 1984-09-04
FR2511679B1 (en) 1985-02-01
SU1447284A3 (en) 1988-12-23
DE19975037I2 (en) 2001-06-13
FR2511679A1 (en) 1983-02-25
IL66606A (en) 1987-07-31
NZ201668A (en) 1985-08-16
JPS5843975A (en) 1983-03-14
CA1197247A (en) 1985-11-26
KR890000094B1 (en) 1989-03-07
DK377882A (en) 1983-02-25
BE894175A (en) 1983-02-23
DE3231255A1 (en) 1983-03-03
IE822026L (en) 1983-02-24
SE448543B (en) 1987-03-02
NL192739C (en) 1998-01-06
FI822921A0 (en) 1982-08-23
DK161147C (en) 1991-11-18
CH655114A5 (en) 1986-03-27
NL8203286A (en) 1983-03-16
ES515176A0 (en) 1983-11-01
ZA826120B (en) 1983-07-27
IT1152505B (en) 1987-01-07
NL192739B (en) 1997-09-01
OA07174A (en) 1984-04-30
AU8749382A (en) 1983-03-03
DK161147B (en) 1991-06-03
KR840001175A (en) 1984-03-28
SE8204817D0 (en) 1982-08-23
LV5511A3 (en) 1994-03-10
FI73434B (en) 1987-06-30
GB2104522A (en) 1983-03-09
FI73434C (en) 1987-10-09
ES8400438A1 (en) 1983-11-01
AT380256B (en) 1986-05-12
GEP19960641B (en) 1996-11-15
UA5971A1 (en) 1994-12-29
HU186107B (en) 1985-06-28
LU84347A1 (en) 1983-06-07
IL66606A0 (en) 1982-12-31
SE8204817L (en) 1983-02-25
DE3231255C2 (en) 1992-02-27
LV5621A3 (en) 1994-05-10
NL990010I1 (en) 1999-07-01
JPH045029B2 (en) 1992-01-30
IT8222938A0 (en) 1982-08-23
ATA319182A (en) 1985-09-15
IE53408B1 (en) 1988-11-09
FI822921L (en) 1983-02-25
GB2104522B (en) 1985-06-12
NL990010I2 (en) 1999-09-01
AU571430B2 (en) 1988-04-21

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Legal Events

Date Code Title Description
PC9A Transfer of patents

Free format text: CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED,6-10 CAMBRIDGE TERRACE, REGENT S PARK, LONDON NW1 4JL,GB,940722

MM9A Lapsed patents

Effective date: 19970823