KR880001843B1 - 카복시알킬 디펩타이드의 제조방법 - Google Patents

카복시알킬 디펩타이드의 제조방법 Download PDF

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Publication number
KR880001843B1
KR880001843B1 KR1019810004008A KR810004008A KR880001843B1 KR 880001843 B1 KR880001843 B1 KR 880001843B1 KR 1019810004008 A KR1019810004008 A KR 1019810004008A KR 810004008 A KR810004008 A KR 810004008A KR 880001843 B1 KR880001843 B1 KR 880001843B1
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KR
South Korea
Prior art keywords
compound
alanyl
carboxylic acid
phenylpropyl
carboethoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
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KR1019810004008A
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English (en)
Korean (ko)
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KR830007519A (ko
Inventor
알.노이 스태트 버나드
에이치.골드 엘리자
엠.스미스 엘라자베드
Original Assignee
쉐링 코포레이션
스타이나 캔스태드, 로즈마리 아이젠링
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26895254&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR880001843(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 쉐링 코포레이션, 스타이나 캔스태드, 로즈마리 아이젠링 filed Critical 쉐링 코포레이션
Publication of KR830007519A publication Critical patent/KR830007519A/ko
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Publication of KR880001843B1 publication Critical patent/KR880001843B1/ko
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Saccharide Compounds (AREA)
  • Apparatus For Disinfection Or Sterilisation (AREA)
  • Pyrrole Compounds (AREA)
KR1019810004008A 1980-10-23 1981-10-21 카복시알킬 디펩타이드의 제조방법 Expired KR880001843B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US19988680A 1980-10-23 1980-10-23
US199886 1980-10-23
US25848481A 1981-04-28 1981-04-28
US258484 1981-04-28

Publications (2)

Publication Number Publication Date
KR830007519A KR830007519A (ko) 1983-10-21
KR880001843B1 true KR880001843B1 (ko) 1988-09-21

Family

ID=26895254

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019810004008A Expired KR880001843B1 (ko) 1980-10-23 1981-10-21 카복시알킬 디펩타이드의 제조방법

Country Status (28)

Country Link
US (2) US4818749A (https=)
EP (1) EP0050800B2 (https=)
JP (1) JPH01163197A (https=)
KR (1) KR880001843B1 (https=)
AT (1) ATE20469T1 (https=)
AU (1) AU554362B2 (https=)
CA (1) CA1341206C (https=)
CY (1) CY1469A (https=)
DE (2) DE19575012I2 (https=)
DK (1) DK161523C (https=)
ES (1) ES506414A0 (https=)
FI (1) FI83222C (https=)
GR (1) GR75059B (https=)
HK (1) HK36189A (https=)
HU (1) HU193146B (https=)
IE (1) IE53802B1 (https=)
IL (1) IL64085A (https=)
KE (1) KE3845A (https=)
LU (1) LU88621I2 (https=)
MA (1) MA19309A1 (https=)
MY (1) MY8700683A (https=)
NL (1) NL940001I2 (https=)
NO (2) NO164983C (https=)
NZ (1) NZ198702A (https=)
OA (1) OA06929A (https=)
PH (1) PH21916A (https=)
PT (1) PT73861B (https=)
SG (1) SG78188G (https=)

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* Cited by examiner, † Cited by third party
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HU193146B (en) 1987-08-28
GR75059B (https=) 1984-07-13
MA19309A1 (fr) 1982-07-01
NO813546L (no) 1982-04-26
OA06929A (fr) 1983-05-31
NO164983C (no) 1990-12-05
PH21916A (en) 1988-04-08
DK161523C (da) 1991-12-23
IE812475L (en) 1982-04-23
ES8308838A1 (es) 1983-10-01
AU7661481A (en) 1982-04-29
NZ198702A (en) 1985-08-30
IL64085A (en) 1986-12-31
FI83222C (sv) 1991-06-10
FI83222B (fi) 1991-02-28
DK462581A (da) 1982-04-24
KR830007519A (ko) 1983-10-21
EP0050800A1 (en) 1982-05-05
MY8700683A (en) 1987-12-31
JPH01163197A (ja) 1989-06-27
NL940001I2 (nl) 1998-03-02
DE19575012I2 (de) 2002-01-24
AU554362B2 (en) 1986-08-21
IE53802B1 (en) 1989-03-01
DE3174844D1 (en) 1986-07-24
HK36189A (en) 1989-05-12
SG78188G (en) 1989-03-23
ATE20469T1 (de) 1986-07-15
CA1341206C (en) 2001-03-20
NL940001I1 (nl) 1994-03-01
NO1995008I1 (no) 1995-09-22
ES506414A0 (es) 1983-10-01
EP0050800B2 (en) 1995-06-07
PT73861B (en) 1985-11-12
EP0050800B1 (en) 1986-06-18
DK161523B (da) 1991-07-15
PT73861A (en) 1981-11-01
NO164983B (no) 1990-08-27
LU88621I2 (fr) 1995-09-01
US4818749A (en) 1989-04-04
US4831157A (en) 1989-05-16
KE3845A (en) 1989-04-07
CY1469A (en) 1989-07-21
FI813283L (fi) 1982-04-24

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