KR840000678B1 - 당유도체의 제조방법 - Google Patents

당유도체의 제조방법 Download PDF

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Publication number
KR840000678B1
KR840000678B1 KR1019800002441A KR800002441A KR840000678B1 KR 840000678 B1 KR840000678 B1 KR 840000678B1 KR 1019800002441 A KR1019800002441 A KR 1019800002441A KR 800002441 A KR800002441 A KR 800002441A KR 840000678 B1 KR840000678 B1 KR 840000678B1
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KR
South Korea
Prior art keywords
formula
group
acetyl
methyl
propenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
KR1019800002441A
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English (en)
Korean (ko)
Other versions
KR830002800A (ko
Inventor
볼라크 베르너
삐에르-챨스위
Original Assignee
에프. 호프만-라 롯슈 앤드 캄파니 아크티엔게젤샤프트
쿠르트 네젤보쉬
한스 스튀클린
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by 에프. 호프만-라 롯슈 앤드 캄파니 아크티엔게젤샤프트, 쿠르트 네젤보쉬, 한스 스튀클린 filed Critical 에프. 호프만-라 롯슈 앤드 캄파니 아크티엔게젤샤프트
Publication of KR830002800A publication Critical patent/KR830002800A/ko
Priority to KR1019840001868A priority Critical patent/KR840000850B1/ko
Application granted granted Critical
Publication of KR840000678B1 publication Critical patent/KR840000678B1/ko
Expired legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H3/00—Compounds containing only hydrogen atoms and saccharide radicals having only carbon, hydrogen, and oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00—Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/38—Alcohols containing six-membered aromatic rings and other rings and having unsaturation outside the aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/45—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
    • C07C45/46—Friedel-Crafts reactions
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
    • C07C49/782—Ketones containing a keto group bound to a six-membered aromatic ring polycyclic
    • C07C49/792—Ketones containing a keto group bound to a six-membered aromatic ring polycyclic containing rings other than six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C63/00—Compounds having carboxyl groups bound to a carbon atoms of six-membered aromatic rings
    • C07C63/33—Polycyclic acids
    • C07C63/49—Polycyclic acids containing rings other than six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H13/00—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids
    • C07H13/02—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids
    • C07H13/08—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids having the esterifying carboxyl radicals directly attached to carbocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/04—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/18—Acyclic radicals, substituted by carbocyclic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
KR1019800002441A 1979-06-21 1980-06-20 당유도체의 제조방법 Expired KR840000678B1 (ko)

Priority Applications (1)

Application Number Priority Date Filing Date Title
KR1019840001868A KR840000850B1 (ko) 1979-06-21 1984-04-09 당 유도체의 제조방법

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH580879 1979-06-21
CH5808 1979-06-21

Publications (2)

Publication Number Publication Date
KR830002800A KR830002800A (ko) 1983-05-30
KR840000678B1 true KR840000678B1 (ko) 1984-05-18

Family

ID=4299652

Family Applications (2)

Application Number Title Priority Date Filing Date
KR1019800002441A Expired KR840000678B1 (ko) 1979-06-21 1980-06-20 당유도체의 제조방법
KR1019840001868A Expired KR840000850B1 (ko) 1979-06-21 1984-04-09 당 유도체의 제조방법

Family Applications After (1)

Application Number Title Priority Date Filing Date
KR1019840001868A Expired KR840000850B1 (ko) 1979-06-21 1984-04-09 당 유도체의 제조방법

Country Status (22)

Country Link
US (1) US4316983A (enExample)
EP (1) EP0021339B1 (enExample)
JP (1) JPS567798A (enExample)
KR (2) KR840000678B1 (enExample)
AR (2) AR225312A1 (enExample)
AT (1) ATE2434T1 (enExample)
AU (1) AU530478B2 (enExample)
CA (1) CA1134819A (enExample)
DE (1) DE3061891D1 (enExample)
DK (1) DK154650C (enExample)
ES (2) ES8104322A1 (enExample)
FI (1) FI67386C (enExample)
GR (1) GR69283B (enExample)
HU (1) HU184915B (enExample)
IE (1) IE50463B1 (enExample)
IL (1) IL60324A (enExample)
MC (1) MC1338A1 (enExample)
NO (1) NO148644C (enExample)
NZ (1) NZ194061A (enExample)
PH (1) PH16243A (enExample)
PT (1) PT71435B (enExample)
ZA (1) ZA803538B (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4987223A (en) * 1981-12-23 1991-01-22 Choay S.A. Derivatives of the uronic acid
US4388457A (en) * 1982-02-11 1983-06-14 University Patents, Inc. Phyllanthostatin compounds
CH661516A5 (de) * 1983-12-08 1987-07-31 Hoffmann La Roche Phenylnonatetraenoylzuckerderivate.
AU582758B2 (en) * 1984-06-28 1989-04-13 Mect Corporation Sialic acid derivatives, galactose derivatives and method for producing the same
CH667868A5 (fr) * 1984-09-05 1988-11-15 Oreal Derives du benzonorbornene, leurs procedes de preparation et compositions medicamenteuse et cosmetique les contenant.
LU85726A1 (fr) * 1985-01-10 1986-08-04 Cird Nouveaux derives naphtaleniques du benzonorbornene,leur procede de preparation et compositions medicamenteuse et cosmetique les contenant
ES2058070T3 (es) * 1986-05-09 1994-11-01 Pulverer Gerhard Utilizacion de monosacaridos especificos para la preparacion de un medicamento para impedir metastasis de tumores malignos.
WO1989006654A1 (en) * 1988-01-19 1989-07-27 Board Of Regents, The University Of Texas System Glycosides, liposomal compositions thereof, and methods for their use
US4943563A (en) * 1988-10-03 1990-07-24 Cornell Research Foundation, Inc. 2,3,4-triacylhexose insect repellants
DE3929355A1 (de) * 1989-09-04 1991-03-07 Boehringer Mannheim Gmbh Verfahren zur spezifischen bestimmung von pankreas-(alpha)-amylase
JP2674843B2 (ja) * 1989-10-31 1997-11-12 新日本製鐵株式会社 鋳鉄用被覆アーク溶接棒
US5523398A (en) * 1994-08-31 1996-06-04 The Center For Innovative Technology Cellulose derivatives with a low degree of substitution

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3629238A (en) * 1968-09-20 1971-12-21 Sumitomo Chemical Co Novel glucuronides of 3-indolylaliphatic acid derivatives
FR2141532B1 (enExample) * 1971-06-14 1974-08-23 Anvar
FR2307820A1 (fr) * 1975-04-17 1976-11-12 Hayashibara Seibutsu Chem Inst Glycosides d'echinatine et leur preparation
JPS51125362A (en) * 1975-04-17 1976-11-01 Hayashibara Biochem Lab Inc Process for synthesizing echinatin glycosides
LU77254A1 (enExample) * 1977-05-04 1979-01-18
DK159967C (da) * 1977-12-22 1991-06-03 Hoffmann La Roche Analogifremgangsmaade til fremstilling af terapeutisk aktive stilbenderivater

Also Published As

Publication number Publication date
FI67386B (fi) 1984-11-30
JPH0131518B2 (enExample) 1989-06-26
NO148644C (no) 1983-11-16
CA1134819A (en) 1982-11-02
FI801472A7 (fi) 1980-12-22
DE3061891D1 (en) 1983-03-17
KR830002800A (ko) 1983-05-30
DK154650C (da) 1989-05-01
ES492616A0 (es) 1981-04-16
EP0021339B1 (de) 1983-02-09
DK154650B (da) 1988-12-05
ES8104322A1 (es) 1981-04-16
EP0021339A1 (de) 1981-01-07
NZ194061A (en) 1982-09-07
KR840000850B1 (ko) 1984-06-19
FI67386C (fi) 1985-03-11
NO148644B (no) 1983-08-08
ZA803538B (en) 1981-06-24
AR229247A1 (es) 1983-07-15
IE801280L (en) 1980-12-21
MC1338A1 (fr) 1981-04-21
ES498607A0 (es) 1981-12-01
IL60324A0 (en) 1980-09-16
PT71435B (en) 1981-10-22
US4316983A (en) 1982-02-23
HU184915B (en) 1984-11-28
DK262480A (da) 1980-12-22
IL60324A (en) 1984-01-31
PT71435A (en) 1980-07-01
AU530478B2 (en) 1983-07-14
PH16243A (en) 1983-08-11
NO801862L (no) 1980-12-22
ATE2434T1 (de) 1983-03-15
AR225312A1 (es) 1982-03-15
IE50463B1 (en) 1986-04-30
ES8201175A1 (es) 1981-12-01
AU5902980A (en) 1981-01-08
GR69283B (enExample) 1982-05-13
JPS567798A (en) 1981-01-27

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