KR20240115978A - Lpa 수용체 길항제 및 이의 용도 - Google Patents
Lpa 수용체 길항제 및 이의 용도 Download PDFInfo
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- KR20240115978A KR20240115978A KR1020247022743A KR20247022743A KR20240115978A KR 20240115978 A KR20240115978 A KR 20240115978A KR 1020247022743 A KR1020247022743 A KR 1020247022743A KR 20247022743 A KR20247022743 A KR 20247022743A KR 20240115978 A KR20240115978 A KR 20240115978A
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- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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| US202163287252P | 2021-12-08 | 2021-12-08 | |
| US63/287,252 | 2021-12-08 | ||
| PCT/US2022/081008 WO2023107938A1 (en) | 2021-12-08 | 2022-12-06 | Lpa receptor antagonists and uses thereof |
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| KR20240115978A true KR20240115978A (ko) | 2024-07-26 |
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| WO (1) | WO2023107938A1 (https=) |
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| EP4161936A1 (en) | 2020-06-03 | 2023-04-12 | Gilead Sciences, Inc. | Lpa receptor antagonists and uses thereof |
| CA3185111A1 (en) * | 2020-07-16 | 2022-01-20 | Elisabetta Armani | Amido cyclohexane acid derivatives as lpa receptor inhibitors |
| WO2022034568A1 (en) | 2020-08-11 | 2022-02-17 | Viva Star Biosciences Limited | Triazole-pyridinyl substituted azacyclohexyl acetic acid compounds as lpa receptor antagonists |
| CN114456147B (zh) | 2020-11-10 | 2025-07-15 | 武汉人福创新药物研发中心有限公司 | 氧取代氨基碳酸酯噻吩类化合物 |
| CN114456159A (zh) | 2020-11-10 | 2022-05-10 | 武汉人福创新药物研发中心有限公司 | 氮取代杂环噻吩类化合物及其用途 |
| CN114456157A (zh) | 2020-11-10 | 2022-05-10 | 武汉人福创新药物研发中心有限公司 | 氮取代氨基碳酸酯噻吩类化合物及其用途 |
| WO2022174882A1 (en) | 2021-02-16 | 2022-08-25 | Chiesi Farmaceutici S.P.A. | 5-membered heterocyclyl carbamate derivatives as dual lpa receptor 1 and lpa receptor 2 inhibitors |
| WO2022174883A1 (en) | 2021-02-16 | 2022-08-25 | Chiesi Farmaceutici S.P.A. | 5-membered heterocyclyl derivatives as dual lpa receptor 1 and lpa receptor 2 inhibitors |
| WO2022240879A1 (en) | 2021-05-11 | 2022-11-17 | Gilead Sciences, Inc. | Lpa receptor antagonists and uses thereof |
| KR20240007233A (ko) | 2021-05-13 | 2024-01-16 | 길리애드 사이언시즈, 인코포레이티드 | Lpa 수용체 길항제 및 이의 용도 |
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2022
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- 2022-12-06 AU AU2022405082A patent/AU2022405082B2/en active Active
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- 2022-12-06 JP JP2024531622A patent/JP7709612B2/ja active Active
- 2022-12-06 CA CA3238094A patent/CA3238094A1/en active Pending
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| AU2022405082A1 (en) | 2024-07-11 |
| AU2022405082B2 (en) | 2025-09-25 |
| US20230212150A1 (en) | 2023-07-06 |
| JP7709612B2 (ja) | 2025-07-16 |
| JP2024541569A (ja) | 2024-11-08 |
| EP4444707A1 (en) | 2024-10-16 |
| CN118541360A (zh) | 2024-08-23 |
| WO2023107938A1 (en) | 2023-06-15 |
| CA3238094A1 (en) | 2023-06-15 |
| US11939318B2 (en) | 2024-03-26 |
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