KR20210015937A - 방광암을 치료하기 위한 방법 - Google Patents

방광암을 치료하기 위한 방법 Download PDF

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Publication number
KR20210015937A
KR20210015937A KR1020207037794A KR20207037794A KR20210015937A KR 20210015937 A KR20210015937 A KR 20210015937A KR 1020207037794 A KR1020207037794 A KR 1020207037794A KR 20207037794 A KR20207037794 A KR 20207037794A KR 20210015937 A KR20210015937 A KR 20210015937A
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KR
South Korea
Prior art keywords
compound
pharmaceutically acceptable
vol
sting
acceptable salt
Prior art date
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Pending
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KR1020207037794A
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English (en)
Korean (ko)
Inventor
대식 김
프랭크 팡
아츠시 엔도
형욱 최
밍홍 하오
싱펭 바오
콴춘 황
Original Assignee
에자이 알앤드디 매니지먼트 가부시키가이샤
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Application filed by 에자이 알앤드디 매니지먼트 가부시키가이샤 filed Critical 에자이 알앤드디 매니지먼트 가부시키가이샤
Publication of KR20210015937A publication Critical patent/KR20210015937A/ko
Pending legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7084—Compounds having two nucleosides or nucleotides, e.g. nicotinamide-adenine dinucleotide, flavine-adenine dinucleotide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
KR1020207037794A 2018-06-01 2019-05-31 방광암을 치료하기 위한 방법 Pending KR20210015937A (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201862679495P 2018-06-01 2018-06-01
US62/679,495 2018-06-01
US201962826347P 2019-03-29 2019-03-29
US62/826,347 2019-03-29
PCT/US2019/034933 WO2019232392A1 (en) 2018-06-01 2019-05-31 Methods for the treatment of bladder cancer

Publications (1)

Publication Number Publication Date
KR20210015937A true KR20210015937A (ko) 2021-02-10

Family

ID=67138025

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020207037794A Pending KR20210015937A (ko) 2018-06-01 2019-05-31 방광암을 치료하기 위한 방법

Country Status (11)

Country Link
US (1) US12251394B2 (https=)
EP (1) EP3801561B1 (https=)
JP (1) JP7335277B2 (https=)
KR (1) KR20210015937A (https=)
CN (1) CN112512531B (https=)
AU (1) AU2019277679B2 (https=)
BR (1) BR112020024605A2 (https=)
CA (1) CA3101623A1 (https=)
MX (1) MX2020012964A (https=)
SG (1) SG11202011434SA (https=)
WO (1) WO2019232392A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202200136A (zh) 2020-04-10 2022-01-01 日商小野藥品工業股份有限公司 癌治療方法
JP2024533394A (ja) 2021-09-09 2024-09-12 エーザイ・アール・アンド・ディー・マネジメント株式会社 Ｓｔｉｎｇアゴニストのバイオマーカー及びその使用方法

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WO2014179760A1 (en) 2013-05-03 2014-11-06 The Regents Of The University Of California Cyclic di-nucleotide induction of type i interferon
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US20180344758A1 (en) 2014-12-17 2018-12-06 Lipogen Llc Method of Treating Cancer with cGAMP or cGAsMP
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KR102222186B1 (ko) 2015-08-13 2021-03-03 머크 샤프 앤드 돔 코포레이션 Sting 효능제로서 시클릭 디-뉴클레오티드 화합물
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CN107849084B (zh) 2015-12-03 2021-09-14 葛兰素史密斯克莱知识产权发展有限公司 作为sting调节剂的环状嘌呤二核苷酸
US10723756B2 (en) 2016-01-11 2020-07-28 Innate Tumor Immunity Inc. Cyclic dinucleotides for treating conditions associated with STING activity such as cancer
JP2019510802A (ja) 2016-04-07 2019-04-18 グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッドＧｌａｘｏｓｍｉｔｈｋｌｉｎｅ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ Ｄｅｖｅｌｏｐｍｅｎｔ Ｌｉｍｉｔｅｄ タンパク質調節物質として有用な複素環アミド
JOP20170188A1 (ar) 2016-11-25 2019-01-30 Janssen Biotech Inc ثنائي النوكليوتيدات الحلقية كمنبهات ستينغ (sting)
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JP7208225B2 (ja) 2017-08-31 2023-01-18 ブリストル－マイヤーズ スクイブ カンパニー 抗癌剤としての環状ジヌクレオチド

Also Published As

Publication number Publication date
WO2019232392A1 (en) 2019-12-05
JP7335277B2 (ja) 2023-08-29
CN112512531A (zh) 2021-03-16
US12251394B2 (en) 2025-03-18
CA3101623A1 (en) 2019-12-05
US20210205348A1 (en) 2021-07-08
MX2020012964A (es) 2021-02-16
CN112512531B (zh) 2024-04-09
AU2019277679B2 (en) 2024-11-28
SG11202011434SA (en) 2020-12-30
EP3801561A1 (en) 2021-04-14
JP2021525758A (ja) 2021-09-27
BR112020024605A2 (pt) 2021-04-06
EP3801561B1 (en) 2025-03-19
AU2019277679A1 (en) 2020-12-24

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