KR20160111520A - 디히드로프테리디논 유도체 및 그의 용도 - Google Patents

디히드로프테리디논 유도체 및 그의 용도 Download PDF

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KR20160111520A
KR20160111520A KR1020167023459A KR20167023459A KR20160111520A KR 20160111520 A KR20160111520 A KR 20160111520A KR 1020167023459 A KR1020167023459 A KR 1020167023459A KR 20167023459 A KR20167023459 A KR 20167023459A KR 20160111520 A KR20160111520 A KR 20160111520A
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substituted
unsubstituted
compound
certain embodiments
alkyl
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제임스 이. 브래드너
너대니얼 그레이
준 퀴
마이클 알. 맥케온
데니스 버클리
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다나-파버 캔서 인스티튜트 인크.
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/58—1,2-Diazines; Hydrogenated 1,2-diazines
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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KR1020167023459A 2014-01-31 2015-02-02 디히드로프테리디논 유도체 및 그의 용도 Withdrawn KR20160111520A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201461934624P 2014-01-31 2014-01-31
US61/934,624 2014-01-31
PCT/US2015/014044 WO2015117055A1 (en) 2014-01-31 2015-02-02 Dihydropteridinone derivatives and uses thereof

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KR20160111520A true KR20160111520A (ko) 2016-09-26

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US (1) US20160347750A1 (enExample)
EP (1) EP3099171A4 (enExample)
JP (1) JP2017512186A (enExample)
KR (1) KR20160111520A (enExample)
CN (1) CN105939607A (enExample)
CA (1) CA2936871A1 (enExample)
MX (1) MX2016009975A (enExample)
RU (1) RU2673944C2 (enExample)
WO (1) WO2015117055A1 (enExample)

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EP3099171A4 (en) 2017-08-09

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