KR20130087002A - 글리신 수송체-1 저해제, 그의 제조 방법 및 그의 용도 - Google Patents

글리신 수송체-1 저해제, 그의 제조 방법 및 그의 용도 Download PDF

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Publication number
KR20130087002A
KR20130087002A KR1020137000117A KR20137000117A KR20130087002A KR 20130087002 A KR20130087002 A KR 20130087002A KR 1020137000117 A KR1020137000117 A KR 1020137000117A KR 20137000117 A KR20137000117 A KR 20137000117A KR 20130087002 A KR20130087002 A KR 20130087002A
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South Korea
Prior art keywords
methyl
piperazin
benzamide
cyclohexyl
difluoro
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Abandoned
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KR1020137000117A
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English (en)
Korean (ko)
Inventor
크로시토퍼 엘 시오피
마크 에이 울프
피터 알 구조
슈앙 리우
카시나쓰 사달라푸르
비스웨스와렌 파르타사라티
준호 맹
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알바니 몰레큘라 리써치, 인크.
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Publication of KR20130087002A publication Critical patent/KR20130087002A/ko
Abandoned legal-status Critical Current

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KR1020137000117A 2010-06-04 2011-06-02 글리신 수송체-1 저해제, 그의 제조 방법 및 그의 용도 Abandoned KR20130087002A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US35166210P 2010-06-04 2010-06-04
US61/351,662 2010-06-04
PCT/US2011/038939 WO2011153359A1 (en) 2010-06-04 2011-06-02 Glycine transporter-1 inhibitors, methods of making them, and uses thereof

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KR20130087002A true KR20130087002A (ko) 2013-08-05

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KR1020137000117A Abandoned KR20130087002A (ko) 2010-06-04 2011-06-02 글리신 수송체-1 저해제, 그의 제조 방법 및 그의 용도

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US (1) US9045445B2 (https=)
EP (1) EP2575815A4 (https=)
JP (1) JP5813101B2 (https=)
KR (1) KR20130087002A (https=)
CN (1) CN103096893B (https=)
AU (1) AU2011261375B2 (https=)
CA (1) CA2801074A1 (https=)
NZ (1) NZ604035A (https=)
SG (1) SG186885A1 (https=)
WO (1) WO2011153359A1 (https=)

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AU2009303335B2 (en) * 2008-10-09 2016-05-19 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Activators of human pyruvate kinase
WO2010118063A2 (en) 2009-04-06 2010-10-14 Agios Pharmaceuticals, Inc. Therapeutic compositions and related methods of use
WO2010129596A1 (en) 2009-05-04 2010-11-11 Agios Pharmaceuticals, Inc. Pmk2 modulators for use in the treatment of cancer
RU2561132C2 (ru) 2009-06-29 2015-08-20 Аджиос Фармасьютикалз, Инк. Производные хинолинсульфонамидов и их применение для модулирования пкм2 активности
ES2618630T3 (es) 2009-06-29 2017-06-21 Agios Pharmaceuticals, Inc. Composiciones terapéuticas y métodos de uso relacionados
US20130109672A1 (en) 2010-04-29 2013-05-02 The United States Of America,As Represented By The Secretary, Department Of Health And Human Service Activators of human pyruvate kinase
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EP2575815A4 (en) 2013-12-25
JP5813101B2 (ja) 2015-11-17
SG186885A1 (en) 2013-02-28
CA2801074A1 (en) 2011-12-08
CN103096893A (zh) 2013-05-08
US9045445B2 (en) 2015-06-02
AU2011261375B2 (en) 2016-09-22
JP2013530957A (ja) 2013-08-01
WO2011153359A1 (en) 2011-12-08
NZ604035A (en) 2015-02-27
AU2011261375A1 (en) 2012-12-20
EP2575815A1 (en) 2013-04-10
CN103096893B (zh) 2016-05-04

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