KR20120063515A - Ｐｉ３ 키나제 억제제 및 이들의 용도 - Google Patents

Ｐｉ３ 키나제 억제제 및 이들의 용도 Download PDF

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KR20120063515A
KR20120063515A KR1020127009074A KR20127009074A KR20120063515A KR 20120063515 A KR20120063515 A KR 20120063515A KR 1020127009074 A KR1020127009074 A KR 1020127009074A KR 20127009074 A KR20127009074 A KR 20127009074A KR 20120063515 A KR20120063515 A KR 20120063515A
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South Korea
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ring
nitrogen
oxygen
sulfur
membered
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Korean (ko)
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더창 뉴
러셀 씨. 피터
저스윈더 싱
아서 에프. 클루지
호르모츠 마즈디야스니
정둥 주
리신 차오
케빈 쿤츠
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아빌라 테라퓨틱스, 인크.
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • C12N9/10—Transferases (2.)
    • C12N9/12—Transferases (2.) transferring phosphorus containing groups, e.g. kinases (2.7)
    • C12N9/1205—Phosphotransferases with an alcohol group as acceptor (2.7.1), e.g. protein kinases

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KR1020127009074A 2009-09-09 2010-09-09 Ｐｉ３ 키나제 억제제 및 이들의 용도 Ceased KR20120063515A (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US24094709P 2009-09-09 2009-09-09
US61/240,947 2009-09-09
US37139610P 2010-08-06 2010-08-06
US61/371,396 2010-08-06

Publications (1)

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KR20120063515A true KR20120063515A (ko) 2012-06-15

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KR1020127009074A Ceased KR20120063515A (ko) 2009-09-09 2010-09-09 Ｐｉ３ 키나제 억제제 및 이들의 용도

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Country Link
US (1) US20110230476A1 (enExample)
EP (1) EP2475375A4 (enExample)
JP (1) JP2013504325A (enExample)
KR (1) KR20120063515A (enExample)
CN (1) CN102625708A (enExample)
AU (1) AU2010292198A1 (enExample)
BR (1) BR112012008385A2 (enExample)
CA (1) CA2773848A1 (enExample)
IL (1) IL218555A0 (enExample)
MX (1) MX339584B (enExample)
NZ (2) NZ598808A (enExample)
PH (1) PH12012500491A1 (enExample)
RU (1) RU2595718C2 (enExample)
SG (2) SG10201405598QA (enExample)
TW (2) TW201609747A (enExample)
WO (1) WO2011031896A2 (enExample)

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