KR20100122914A - [페닐술파닐페닐]피페리딘의 제조 방법 - Google Patents

[페닐술파닐페닐]피페리딘의 제조 방법 Download PDF

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Publication number
KR20100122914A
KR20100122914A KR1020107019480A KR20107019480A KR20100122914A KR 20100122914 A KR20100122914 A KR 20100122914A KR 1020107019480 A KR1020107019480 A KR 1020107019480A KR 20107019480 A KR20107019480 A KR 20107019480A KR 20100122914 A KR20100122914 A KR 20100122914A
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KR
South Korea
Prior art keywords
compound
hydrogen
alkyl
acid
reaction
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
KR1020107019480A
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English (en)
Korean (ko)
Inventor
마이클 해롤드 록
세바스티안 브란데스
Original Assignee
하. 룬드벡 아크티에셀스카브
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by 하. 룬드벡 아크티에셀스카브 filed Critical 하. 룬드벡 아크티에셀스카브
Publication of KR20100122914A publication Critical patent/KR20100122914A/ko
Ceased legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/52—Oxygen atoms attached in position 4 having an aryl radical as the second substituent in position 4
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
KR1020107019480A 2008-03-03 2009-03-02 [페닐술파닐페닐]피페리딘의 제조 방법 Ceased KR20100122914A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA200800314 2008-03-03
DKPA200800314 2008-03-03

Publications (1)

Publication Number Publication Date
KR20100122914A true KR20100122914A (ko) 2010-11-23

Family

ID=40547924

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020107019480A Ceased KR20100122914A (ko) 2008-03-03 2009-03-02 [페닐술파닐페닐]피페리딘의 제조 방법

Country Status (28)

Country Link
US (1) US8362255B2 (https=)
EP (1) EP2260024B1 (https=)
JP (1) JP5564439B2 (https=)
KR (1) KR20100122914A (https=)
CN (1) CN101959859B (https=)
AR (1) AR070737A1 (https=)
AT (1) ATE539055T1 (https=)
AU (1) AU2009221170B2 (https=)
BR (1) BRPI0908166A2 (https=)
CA (1) CA2715579A1 (https=)
CL (1) CL2009000490A1 (https=)
CO (1) CO6290758A2 (https=)
CY (1) CY1113887T1 (https=)
DK (1) DK2260024T3 (https=)
EA (1) EA017855B1 (https=)
ES (1) ES2377862T3 (https=)
HR (1) HRP20120118T1 (https=)
IL (1) IL207471A (https=)
MX (1) MX2010008729A (https=)
NZ (1) NZ587593A (https=)
PL (1) PL2260024T3 (https=)
PT (1) PT2260024E (https=)
RS (1) RS52128B (https=)
SI (1) SI2260024T1 (https=)
TW (1) TW200940505A (https=)
UA (1) UA98698C2 (https=)
WO (1) WO2009109541A1 (https=)
ZA (1) ZA201006135B (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2007260356B2 (en) * 2006-06-16 2013-01-24 H. Lundbeck A/S Crystalline forms of 4- [2- (4-methylphenylsulfanyl) -phenyl] piperidine with combined serotonin and norepinephrine reuptake inhibition for the treatment of neuropathic pain
JP2012163850A (ja) * 2011-02-08 2012-08-30 Nippon Sheet Glass Co Ltd 正立等倍レンズアレイプレート、光走査ユニット、画像読取装置および画像書込装置
US9173883B2 (en) 2012-05-21 2015-11-03 Novartis Ag Ring-substituted N-pyridinyl amides as kinase inhibitors
CN104710345B (zh) * 2013-12-17 2017-09-05 江苏恩华药业股份有限公司 用于制备4‑（2‑（4‑甲基苯基硫基））苯基哌啶的化合物、其制备方法及应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2324087A (en) * 1997-04-10 1998-10-14 Merck & Co Inc Preparation of (S)-3-Carbethoxy-3-benzylpiperidine
EP1244623A1 (en) 1999-12-20 2002-10-02 Eli Lilly And Company A process for preparing 4-substituted piperidines
UA81749C2 (uk) * 2001-10-04 2008-02-11 Х. Луннбек А/С Фенілпіперазинові похідні як інгібітори зворотного захоплення серотоніну
UA81300C2 (en) * 2003-04-04 2007-12-25 Lundbeck & Co As H Derivates of 4-(2-fenilsulfanilfenil)-1,2,3,6-tetrahydropiridin as retarding agents of serotonin recapture
HRP20080478T3 (hr) 2003-04-04 2009-02-28 H. Lundbeck A/S Derivati 4-(2-fenilsulfanil-fenil)-piperidina kaoinhibitori ponovne pohrane serotonina
AU2007260356B2 (en) * 2006-06-16 2013-01-24 H. Lundbeck A/S Crystalline forms of 4- [2- (4-methylphenylsulfanyl) -phenyl] piperidine with combined serotonin and norepinephrine reuptake inhibition for the treatment of neuropathic pain

Also Published As

Publication number Publication date
IL207471A (en) 2014-06-30
CA2715579A1 (en) 2009-09-11
CN101959859A (zh) 2011-01-26
CY1113887T1 (el) 2016-07-27
EP2260024B1 (en) 2011-12-28
MX2010008729A (es) 2010-09-24
IL207471A0 (en) 2010-12-30
PT2260024E (pt) 2012-03-06
EA201071025A1 (ru) 2011-02-28
RS52128B (sr) 2012-08-31
BRPI0908166A2 (pt) 2015-08-11
CO6290758A2 (es) 2011-06-20
EP2260024A1 (en) 2010-12-15
HRP20120118T1 (hr) 2012-03-31
US8362255B2 (en) 2013-01-29
WO2009109541A1 (en) 2009-09-11
US20110054178A1 (en) 2011-03-03
SI2260024T1 (sl) 2012-04-30
AU2009221170B2 (en) 2013-08-22
DK2260024T3 (da) 2012-02-27
AR070737A1 (es) 2010-04-28
AU2009221170A1 (en) 2009-09-11
CL2009000490A1 (es) 2010-04-16
PL2260024T3 (pl) 2012-04-30
JP5564439B2 (ja) 2014-07-30
ZA201006135B (en) 2011-10-26
TW200940505A (en) 2009-10-01
ATE539055T1 (de) 2012-01-15
ES2377862T3 (es) 2012-04-02
CN101959859B (zh) 2013-08-14
EA017855B1 (ru) 2013-03-29
JP2011513358A (ja) 2011-04-28
HK1153458A1 (en) 2012-03-30
NZ587593A (en) 2012-03-30
UA98698C2 (en) 2012-06-11

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