KR20090082452A - 3-벤질-2-메틸-2,3,3ａ,4,5,6,7,7ａ-옥타히드로벤조[ｄ]이속사졸-4-온의 염 - Google Patents

3-벤질-2-메틸-2,3,3ａ,4,5,6,7,7ａ-옥타히드로벤조[ｄ]이속사졸-4-온의 염 Download PDF

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Publication number
KR20090082452A
KR20090082452A KR1020097011322A KR20097011322A KR20090082452A KR 20090082452 A KR20090082452 A KR 20090082452A KR 1020097011322 A KR1020097011322 A KR 1020097011322A KR 20097011322 A KR20097011322 A KR 20097011322A KR 20090082452 A KR20090082452 A KR 20090082452A
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KR
South Korea
Prior art keywords
fumarate
fumarate salt
formula
medicament
btg
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
KR1020097011322A
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English (en)
Korean (ko)
Inventor
파비오 네기아니
라우라 디니
Original Assignee
아비오젠 파르마 에스피에이
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Application filed by 아비오젠 파르마 에스피에이 filed Critical 아비오젠 파르마 에스피에이
Publication of KR20090082452A publication Critical patent/KR20090082452A/ko
Withdrawn legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/423—Oxazoles condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Addiction (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
KR1020097011322A 2006-11-02 2007-10-31 3-벤질-2-메틸-2,3,3ａ,4,5,6,7,7ａ-옥타히드로벤조[ｄ]이속사졸-4-온의 염 Withdrawn KR20090082452A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT002102A ITMI20062102A1 (it) 2006-11-02 2006-11-02 Nuovui sali di 3-benzil-2-metil-2,3,3a,4,5,6,7,7a-ottaidrobenzo-d-isossazol-4-one
ITMI2006A002102 2006-11-02

Publications (1)

Publication Number Publication Date
KR20090082452A true KR20090082452A (ko) 2009-07-30

Family

ID=39145485

Family Applications (2)

Application Number Title Priority Date Filing Date
KR1020097011322A Withdrawn KR20090082452A (ko) 2006-11-02 2007-10-31 3-벤질-2-메틸-2,3,3ａ,4,5,6,7,7ａ-옥타히드로벤조[ｄ]이속사졸-4-온의 염
KR1020097011287A Withdrawn KR20090077014A (ko) 2006-11-02 2007-10-31 3-벤질-2-메틸-2,3,3ａ,4,5,6,7,7ａ-옥타히드로벤조[ｄ]이속사졸-4-온의 염

Family Applications After (1)

Application Number Title Priority Date Filing Date
KR1020097011287A Withdrawn KR20090077014A (ko) 2006-11-02 2007-10-31 3-벤질-2-메틸-2,3,3ａ,4,5,6,7,7ａ-옥타히드로벤조[ｄ]이속사졸-4-온의 염

Country Status (20)

Country Link
US (2) US20100069451A1 (OSRAM)
EP (2) EP2094674B1 (OSRAM)
JP (2) JP2010509309A (OSRAM)
KR (2) KR20090082452A (OSRAM)
CN (2) CN101535282A (OSRAM)
AT (2) ATE504578T1 (OSRAM)
AU (2) AU2007315833A1 (OSRAM)
BR (2) BRPI0718392A2 (OSRAM)
CA (2) CA2667513A1 (OSRAM)
DE (2) DE602007013801D1 (OSRAM)
HR (2) HRP20090477A2 (OSRAM)
IL (2) IL198444A0 (OSRAM)
IT (1) ITMI20062102A1 (OSRAM)
MX (2) MX2009004293A (OSRAM)
NO (2) NO20092115L (OSRAM)
NZ (2) NZ577311A (OSRAM)
RS (2) RS20090388A (OSRAM)
RU (2) RU2009120724A (OSRAM)
WO (2) WO2008053325A1 (OSRAM)
ZA (2) ZA200903618B (OSRAM)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ITMI20080768A1 (it) * 2008-04-24 2009-10-25 Abiogen Pharma Spa Procedimento per la preparazione di un composto in forma cristallina di 3-benzil-2-metil-2,3,3a,4,5,6,7,7a-ottaidro-benzo[d]isossazol-4-one
EP2112142A1 (en) * 2008-04-24 2009-10-28 Abiogen Pharma S.p.A. Process for preparing a crystalline form compound of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one
EP2218721A1 (en) * 2009-02-11 2010-08-18 LEK Pharmaceuticals d.d. Novel salts of sitagliptin
WO2011010332A1 (en) * 2009-07-23 2011-01-27 Abiogen Pharma S.P.A. Process for preparing rel-(3r*,3as*,7as*)-3-benzyl-2-methyl-2,3, 3a,4,5,6,7,7a- octahydrobenzo[d]isoxazoi-4-one or a salt thereof
WO2016123275A1 (en) * 2015-01-30 2016-08-04 Boehringer Ingelheim International Gmbh Aldosterone synthase inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4161595A (en) * 1978-10-02 1979-07-17 Bristol-Myers Company Levulinic acid salt
US4419358A (en) * 1981-11-12 1983-12-06 Mead Johnson & Company Isethionic acid salt of 9-cyclohexyl-2-propoxy-9H-purine-6-amine and compositions containing an effective bronchodilating concentration of it
GB2264299B (en) * 1992-02-19 1995-07-26 British Tech Group Iso-oxazolidine derivatives

Also Published As

Publication number Publication date
NO20092114L (no) 2009-05-29
CN101535282A (zh) 2009-09-16
US20100069451A1 (en) 2010-03-18
HRP20090477A2 (hr) 2009-11-30
DE602007013801D1 (de) 2011-05-19
MX2009004293A (es) 2009-05-08
CN101535281A (zh) 2009-09-16
EP2094674B1 (en) 2011-03-16
WO2008053326A1 (en) 2008-05-08
NO20092115L (no) 2009-05-29
WO2008053325A1 (en) 2008-05-08
RS20090388A (sr) 2010-12-31
ITMI20062102A1 (it) 2008-05-03
JP2010509310A (ja) 2010-03-25
IL198443A0 (en) 2010-02-17
ZA200903618B (en) 2010-07-28
BRPI0718391A2 (pt) 2013-11-26
AU2007315832A1 (en) 2008-05-08
ATE504578T1 (de) 2011-04-15
NZ577311A (en) 2010-10-29
RS20090389A (sr) 2010-12-31
RU2009120667A (ru) 2010-12-10
US20100069450A1 (en) 2010-03-18
DE602007013278D1 (de) 2011-04-28
CA2667513A1 (en) 2008-05-08
MX2009004294A (es) 2009-05-08
CA2667515A1 (en) 2008-05-08
ZA200903810B (en) 2010-07-28
EP2094675A1 (en) 2009-09-02
ATE502021T1 (de) 2011-04-15
HRP20090470A2 (hr) 2009-11-30
RU2009120724A (ru) 2010-12-10
BRPI0718392A2 (pt) 2013-11-26
NZ577978A (en) 2010-10-29
EP2094674A1 (en) 2009-09-02
JP2010509309A (ja) 2010-03-25
KR20090077014A (ko) 2009-07-13
AU2007315833A1 (en) 2008-05-08
EP2094675B1 (en) 2011-04-06
IL198444A0 (en) 2010-02-17

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