ITMI20062102A1 - Nuovui sali di 3-benzil-2-metil-2,3,3a,4,5,6,7,7a-ottaidrobenzo-d-isossazol-4-one - Google Patents
Nuovui sali di 3-benzil-2-metil-2,3,3a,4,5,6,7,7a-ottaidrobenzo-d-isossazol-4-oneInfo
- Publication number
- ITMI20062102A1 ITMI20062102A1 IT002102A ITMI20062102A ITMI20062102A1 IT MI20062102 A1 ITMI20062102 A1 IT MI20062102A1 IT 002102 A IT002102 A IT 002102A IT MI20062102 A ITMI20062102 A IT MI20062102A IT MI20062102 A1 ITMI20062102 A1 IT MI20062102A1
- Authority
- IT
- Italy
- Prior art keywords
- benzyl
- methyl
- octoidrobenzo
- isossazol
- new salts
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/423—Oxazoles condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Biomedical Technology (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Addiction (AREA)
- Hospice & Palliative Care (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Priority Applications (39)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT002102A ITMI20062102A1 (it) | 2006-11-02 | 2006-11-02 | Nuovui sali di 3-benzil-2-metil-2,3,3a,4,5,6,7,7a-ottaidrobenzo-d-isossazol-4-one |
AT07825549T ATE502021T1 (de) | 2006-11-02 | 2007-10-31 | Salz von 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a- octahydrobenzoädüisoxazol-4-on |
AU2007315832A AU2007315832A1 (en) | 2006-11-02 | 2007-10-31 | A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
PCT/IB2007/003292 WO2008053326A1 (en) | 2006-11-02 | 2007-10-31 | A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
RSP-2009/0389A RS20090389A (en) | 2006-11-02 | 2007-10-31 | A salt of -benzyl -2- metil - 2,3,3a,4,5,6,7,7a-oktahydrobenzo (d)isoxazol -4- one |
CA002667513A CA2667513A1 (en) | 2006-11-02 | 2007-10-31 | A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
EP07825550A EP2094675B1 (en) | 2006-11-02 | 2007-10-31 | A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
MX2009004294A MX2009004294A (es) | 2006-11-02 | 2007-10-31 | Una sal de 3-bencil-2-metil-2,3,3a,4,5,6,7,7a-octahidrobenzo[d]iso xasol-4-ona. |
CNA2007800406691A CN101535282A (zh) | 2006-11-02 | 2007-10-31 | 3-苄基-2-甲基-2,3,3a,4,5,6,7,7a-八氢苯并[d]异噁唑-4-酮的盐 |
RU2009120724/04A RU2009120724A (ru) | 2006-11-02 | 2007-10-31 | Соль 3-бензил-2-метил-2,3,3а,4,5,6,7,7а-октагидробензо[d]изоксазол-4-она |
AT07825550T ATE504578T1 (de) | 2006-11-02 | 2007-10-31 | Salz von 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a- octahydrobenzoädüisoxazol-4-on |
DE602007013278T DE602007013278D1 (de) | 2006-11-02 | 2007-10-31 | Salz von 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzoädüisoxazol-4-on |
MX2009004293A MX2009004293A (es) | 2006-11-02 | 2007-10-31 | Una sal de 3-bencil-2-metil-2,3,3a,4,5,6,7,7a-octahidrobenzo[d]iso xasol-4-ona. |
JP2009535825A JP2010509310A (ja) | 2006-11-02 | 2007-10-31 | 3−ベンジル−2−メチル−2,3,3a,4,5,6,7,7a−オクタヒドロベンゾ[d]イソオキサゾール−4−オンの塩 |
KR1020097011322A KR20090082452A (ko) | 2006-11-02 | 2007-10-31 | 3-벤질-2-메틸-2,3,3a,4,5,6,7,7a-옥타히드로벤조[d]이속사졸-4-온의 염 |
NZ577978A NZ577978A (en) | 2006-11-02 | 2007-10-31 | The fumarate salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
EP07825549A EP2094674B1 (en) | 2006-11-02 | 2007-10-31 | A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
DE602007013801T DE602007013801D1 (de) | 2006-11-02 | 2007-10-31 | Salz von 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzoädüisoxazol-4-on |
PCT/IB2007/003291 WO2008053325A1 (en) | 2006-11-02 | 2007-10-31 | A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
BRPI0718391-7A BRPI0718391A2 (pt) | 2006-11-02 | 2007-10-31 | SAL DO COMPOSTO DE 3-BENZIL-2-METIL-2,3,3a,4,5,6,7,7a-OCTAIDROBENZO [D] ISOXAZOL-4-ONA |
CNA2007800406598A CN101535281A (zh) | 2006-11-02 | 2007-10-31 | 3-苄基-2-甲基-2,3,3a,4,5,6,7,7a-八氢苯并[d]异噁唑-4-酮的盐 |
KR1020097011287A KR20090077014A (ko) | 2006-11-02 | 2007-10-31 | 3-벤질-2-메틸-2,3,3a,4,5,6,7,7a-옥타히드로벤조[d]이속사졸-4-온의 염 |
NZ577311A NZ577311A (en) | 2006-11-02 | 2007-10-31 | The oxalate salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
US12/513,351 US20100069450A1 (en) | 2006-11-02 | 2007-10-31 | Salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7, 7a- octahydrobenzo[d]isoxazol-4-one |
AU2007315833A AU2007315833A1 (en) | 2006-11-02 | 2007-10-31 | A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
JP2009535824A JP2010509309A (ja) | 2006-11-02 | 2007-10-31 | 3−ベンジル−2−メチル−2,3,3a,4,5,6,7,7a−オクタヒドロベンゾ[d]イソオキサゾール−4−オンの塩 |
US12/513,352 US20100069451A1 (en) | 2006-11-02 | 2007-10-31 | Salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7, 7a- octahydrobenzo[d]isoxazol-4-one |
RU2009120667/04A RU2009120667A (ru) | 2006-11-02 | 2007-10-31 | Соль 3-бензил-2-метил-2,3,3а,4,5,6,7,7а-октагидробензо[d]изоксазол-4-она |
CA002667515A CA2667515A1 (en) | 2006-11-02 | 2007-10-31 | A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
BRPI0718392-5A BRPI0718392A2 (pt) | 2006-11-02 | 2007-10-31 | SAL COMPOSTO DE 3-BENZIL-2-METIL-2,3,3a,4,5,6,7,7a-OCTAIDROBENZO [d] ISOXAZOL-4-ONA |
RSP-2009/0388A RS20090388A (en) | 2006-11-02 | 2007-10-31 | A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
IL198443A IL198443A0 (en) | 2006-11-02 | 2009-04-28 | A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a- |
IL198444A IL198444A0 (en) | 2006-11-02 | 2009-04-28 | A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a- |
ZA200903618A ZA200903618B (en) | 2006-11-02 | 2009-05-25 | A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
NO20092114A NO20092114L (no) | 2006-11-02 | 2009-05-29 | Salt av 3-benzyl-2-metyl-2,3,3a,4,5,6,7,7a-oktahydrobenzo[d]isoksazol-4-on |
NO20092115A NO20092115L (no) | 2006-11-02 | 2009-05-29 | Salt av 3-benzyl-2-metyl-2,3,3a,4,5,6,7,7a-oktahydrobenzo[d]isoksazol-4-on |
ZA200903810A ZA200903810B (en) | 2006-11-02 | 2009-06-01 | A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
HR20090470A HRP20090470A2 (hr) | 2006-11-02 | 2009-09-03 | Sol 3-benzil-2-methil-2.3.3.a.4.5.6.7,7a-octahidrobenzo[d]isoksazol-4-ona |
HR20090477A HRP20090477A2 (hr) | 2006-11-02 | 2009-09-08 | SOL 3-BENZIL-2-METIL-2,3,3A,4,5,6,7,7A-OKTAHIDROBENZO[d]IZOKSAZOL-4-ONA |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT002102A ITMI20062102A1 (it) | 2006-11-02 | 2006-11-02 | Nuovui sali di 3-benzil-2-metil-2,3,3a,4,5,6,7,7a-ottaidrobenzo-d-isossazol-4-one |
Publications (1)
Publication Number | Publication Date |
---|---|
ITMI20062102A1 true ITMI20062102A1 (it) | 2008-05-03 |
Family
ID=39145485
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT002102A ITMI20062102A1 (it) | 2006-11-02 | 2006-11-02 | Nuovui sali di 3-benzil-2-metil-2,3,3a,4,5,6,7,7a-ottaidrobenzo-d-isossazol-4-one |
Country Status (20)
Country | Link |
---|---|
US (2) | US20100069450A1 (it) |
EP (2) | EP2094675B1 (it) |
JP (2) | JP2010509310A (it) |
KR (2) | KR20090082452A (it) |
CN (2) | CN101535281A (it) |
AT (2) | ATE502021T1 (it) |
AU (2) | AU2007315833A1 (it) |
BR (2) | BRPI0718392A2 (it) |
CA (2) | CA2667515A1 (it) |
DE (2) | DE602007013278D1 (it) |
HR (2) | HRP20090470A2 (it) |
IL (2) | IL198443A0 (it) |
IT (1) | ITMI20062102A1 (it) |
MX (2) | MX2009004293A (it) |
NO (2) | NO20092115L (it) |
NZ (2) | NZ577311A (it) |
RS (2) | RS20090388A (it) |
RU (2) | RU2009120724A (it) |
WO (2) | WO2008053325A1 (it) |
ZA (2) | ZA200903618B (it) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2112142A1 (en) * | 2008-04-24 | 2009-10-28 | Abiogen Pharma S.p.A. | Process for preparing a crystalline form compound of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
ITMI20080768A1 (it) * | 2008-04-24 | 2009-10-25 | Abiogen Pharma Spa | Procedimento per la preparazione di un composto in forma cristallina di 3-benzil-2-metil-2,3,3a,4,5,6,7,7a-ottaidro-benzo[d]isossazol-4-one |
EP2218721A1 (en) * | 2009-02-11 | 2010-08-18 | LEK Pharmaceuticals d.d. | Novel salts of sitagliptin |
WO2011010332A1 (en) * | 2009-07-23 | 2011-01-27 | Abiogen Pharma S.P.A. | Process for preparing rel-(3r*,3as*,7as*)-3-benzyl-2-methyl-2,3, 3a,4,5,6,7,7a- octahydrobenzo[d]isoxazoi-4-one or a salt thereof |
JP6615896B2 (ja) * | 2015-01-30 | 2019-12-04 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | アルドステロン合成酵素阻害剤 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4161595A (en) * | 1978-10-02 | 1979-07-17 | Bristol-Myers Company | Levulinic acid salt |
US4419358A (en) * | 1981-11-12 | 1983-12-06 | Mead Johnson & Company | Isethionic acid salt of 9-cyclohexyl-2-propoxy-9H-purine-6-amine and compositions containing an effective bronchodilating concentration of it |
GB2264299B (en) * | 1992-02-19 | 1995-07-26 | British Tech Group | Iso-oxazolidine derivatives |
-
2006
- 2006-11-02 IT IT002102A patent/ITMI20062102A1/it unknown
-
2007
- 2007-10-31 NZ NZ577311A patent/NZ577311A/en unknown
- 2007-10-31 US US12/513,351 patent/US20100069450A1/en not_active Abandoned
- 2007-10-31 AT AT07825549T patent/ATE502021T1/de not_active IP Right Cessation
- 2007-10-31 MX MX2009004293A patent/MX2009004293A/es not_active Application Discontinuation
- 2007-10-31 RU RU2009120724/04A patent/RU2009120724A/ru not_active Application Discontinuation
- 2007-10-31 AU AU2007315833A patent/AU2007315833A1/en not_active Abandoned
- 2007-10-31 RU RU2009120667/04A patent/RU2009120667A/ru not_active Application Discontinuation
- 2007-10-31 CN CNA2007800406598A patent/CN101535281A/zh active Pending
- 2007-10-31 DE DE602007013278T patent/DE602007013278D1/de active Active
- 2007-10-31 AU AU2007315832A patent/AU2007315832A1/en not_active Abandoned
- 2007-10-31 KR KR1020097011322A patent/KR20090082452A/ko not_active Application Discontinuation
- 2007-10-31 RS RSP-2009/0388A patent/RS20090388A/sr unknown
- 2007-10-31 KR KR1020097011287A patent/KR20090077014A/ko not_active Application Discontinuation
- 2007-10-31 EP EP07825550A patent/EP2094675B1/en not_active Not-in-force
- 2007-10-31 WO PCT/IB2007/003291 patent/WO2008053325A1/en active Application Filing
- 2007-10-31 AT AT07825550T patent/ATE504578T1/de not_active IP Right Cessation
- 2007-10-31 JP JP2009535825A patent/JP2010509310A/ja active Pending
- 2007-10-31 DE DE602007013801T patent/DE602007013801D1/de active Active
- 2007-10-31 BR BRPI0718392-5A patent/BRPI0718392A2/pt not_active IP Right Cessation
- 2007-10-31 NZ NZ577978A patent/NZ577978A/en unknown
- 2007-10-31 RS RSP-2009/0389A patent/RS20090389A/sr unknown
- 2007-10-31 US US12/513,352 patent/US20100069451A1/en not_active Abandoned
- 2007-10-31 BR BRPI0718391-7A patent/BRPI0718391A2/pt not_active IP Right Cessation
- 2007-10-31 JP JP2009535824A patent/JP2010509309A/ja active Pending
- 2007-10-31 WO PCT/IB2007/003292 patent/WO2008053326A1/en active Application Filing
- 2007-10-31 CA CA002667515A patent/CA2667515A1/en not_active Abandoned
- 2007-10-31 EP EP07825549A patent/EP2094674B1/en not_active Not-in-force
- 2007-10-31 CN CNA2007800406691A patent/CN101535282A/zh active Pending
- 2007-10-31 MX MX2009004294A patent/MX2009004294A/es not_active Application Discontinuation
- 2007-10-31 CA CA002667513A patent/CA2667513A1/en not_active Abandoned
-
2009
- 2009-04-28 IL IL198443A patent/IL198443A0/en unknown
- 2009-04-28 IL IL198444A patent/IL198444A0/en unknown
- 2009-05-25 ZA ZA200903618A patent/ZA200903618B/xx unknown
- 2009-05-29 NO NO20092115A patent/NO20092115L/no not_active Application Discontinuation
- 2009-05-29 NO NO20092114A patent/NO20092114L/no not_active Application Discontinuation
- 2009-06-01 ZA ZA200903810A patent/ZA200903810B/xx unknown
- 2009-09-03 HR HR20090470A patent/HRP20090470A2/hr not_active Application Discontinuation
- 2009-09-08 HR HR20090477A patent/HRP20090477A2/hr not_active Application Discontinuation
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