KR20080077010A - 1-벤조일-4-[2-[4-메톡시-7-(3-메틸-1Ｈ-1,2,4-트리아졸-1-일)-1-[(포스포노옥시)메틸]-1Ｈ-피롤로[2,3-ｃ]피리딘-3-일]-1,2-디옥소에틸]-피페라진의 결정질 형태 - Google Patents

1-벤조일-4-[2-[4-메톡시-7-(3-메틸-1Ｈ-1,2,4-트리아졸-1-일)-1-[(포스포노옥시)메틸]-1Ｈ-피롤로[2,3-ｃ]피리딘-3-일]-1,2-디옥소에틸]-피페라진의 결정질 형태 Download PDF

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KR20080077010A
KR20080077010A KR1020087016884A KR20087016884A KR20080077010A KR 20080077010 A KR20080077010 A KR 20080077010A KR 1020087016884 A KR1020087016884 A KR 1020087016884A KR 20087016884 A KR20087016884 A KR 20087016884A KR 20080077010 A KR20080077010 A KR 20080077010A
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crystalline form
temperature
powder
group
crystalline
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Korean (ko)
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청-핀 에이치 첸
던 디기우그노
치 가오
총-후이 구
자쿠안 칼라니 르봉
빙-시오우 양
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브리스톨-마이어스 스큅 컴퍼니
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Publication of KR20080077010A publication Critical patent/KR20080077010A/ko
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/06—Phosphorus compounds without P—C bonds
    • C07F9/08—Esters of oxyacids of phosphorus
    • C07F9/09—Esters of phosphoric acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1020087016884A 2005-12-14 2006-12-13 1-벤조일-4-[2-[4-메톡시-7-(3-메틸-1Ｈ-1,2,4-트리아졸-1-일)-1-[(포스포노옥시)메틸]-1Ｈ-피롤로[2,3-ｃ]피리딘-3-일]-1,2-디옥소에틸]-피페라진의 결정질 형태 Ceased KR20080077010A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US75024705P 2005-12-14 2005-12-14
US60/750,247 2005-12-14

Publications (1)

Publication Number Publication Date
KR20080077010A true KR20080077010A (ko) 2008-08-20

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KR1020087016884A Ceased KR20080077010A (ko) 2005-12-14 2006-12-13 1-벤조일-4-[2-[4-메톡시-7-(3-메틸-1Ｈ-1,2,4-트리아졸-1-일)-1-[(포스포노옥시)메틸]-1Ｈ-피롤로[2,3-ｃ]피리딘-3-일]-1,2-디옥소에틸]-피페라진의 결정질 형태

Country Status (17)

Country Link
US (1) US7851476B2 (enExample)
EP (1) EP1963342A2 (enExample)
JP (1) JP5400387B2 (enExample)
KR (1) KR20080077010A (enExample)
CN (1) CN101365708B (enExample)
AU (1) AU2006326432B2 (enExample)
BR (1) BRPI0619851A2 (enExample)
CA (1) CA2635717A1 (enExample)
EA (1) EA014706B1 (enExample)
GE (1) GEP20125413B (enExample)
IL (1) IL191769A (enExample)
MY (1) MY144293A (enExample)
NO (1) NO20082477L (enExample)
NZ (2) NZ568776A (enExample)
UA (1) UA94928C2 (enExample)
WO (1) WO2007070589A2 (enExample)
ZA (1) ZA200805063B (enExample)

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Also Published As

Publication number Publication date
EP1963342A2 (en) 2008-09-03
IL191769A0 (en) 2008-12-29
WO2007070589A2 (en) 2007-06-21
MY144293A (en) 2011-08-29
GEP20125413B (en) 2012-03-12
JP2009521414A (ja) 2009-06-04
EA014706B1 (ru) 2011-02-28
CA2635717A1 (en) 2007-06-21
US20070155702A1 (en) 2007-07-05
US7851476B2 (en) 2010-12-14
JP5400387B2 (ja) 2014-01-29
CN101365708B (zh) 2012-12-12
AU2006326432A1 (en) 2007-06-21
BRPI0619851A2 (pt) 2011-10-25
CN101365708A (zh) 2009-02-11
NO20082477L (no) 2008-09-05
EA200801529A1 (ru) 2009-02-27
ZA200805063B (en) 2009-10-28
NZ568776A (en) 2011-06-30
WO2007070589A3 (en) 2007-09-27
IL191769A (en) 2011-08-31
NZ592684A (en) 2012-07-27
AU2006326432B2 (en) 2012-07-12
UA94928C2 (en) 2011-06-25

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