KR101956399B1 - C4­모노메틸 트리터페노이드 유도체 및 그의 이용 방법 - Google Patents

C4­모노메틸 트리터페노이드 유도체 및 그의 이용 방법 Download PDF

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KR101956399B1
KR101956399B1 KR1020137026782A KR20137026782A KR101956399B1 KR 101956399 B1 KR101956399 B1 KR 101956399B1 KR 1020137026782 A KR1020137026782 A KR 1020137026782A KR 20137026782 A KR20137026782 A KR 20137026782A KR 101956399 B1 KR101956399 B1 KR 101956399B1
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KR20140025383A (ko
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에릭 앤더슨
신 지앙
멜리언 비스닉
크리스토퍼 에프. 벤더
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리아타 파마슈티컬즈, 아이엔씨.
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J63/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C07J63/008Expansion of ring D by one atom, e.g. D homo steroids
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    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J63/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • AHUMAN NECESSITIES
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    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
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    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
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    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
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    • A61P39/00General protective or antinoxious agents
    • A61P39/06Free radical scavengers or antioxidants
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring

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  • Health & Medical Sciences (AREA)
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  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Neurology (AREA)
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  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Psychology (AREA)
  • Pulmonology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Toxicology (AREA)
  • Biochemistry (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Emergency Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Transplantation (AREA)
KR1020137026782A 2011-03-11 2012-03-09 C4­모노메틸 트리터페노이드 유도체 및 그의 이용 방법 Active KR101956399B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161452017P 2011-03-11 2011-03-11
US61/452,017 2011-03-11
PCT/US2012/028569 WO2012125488A1 (en) 2011-03-11 2012-03-09 C4-monomethyl triterpenoid derivatives and methods of use thereof

Publications (2)

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KR20140025383A KR20140025383A (ko) 2014-03-04
KR101956399B1 true KR101956399B1 (ko) 2019-03-08

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US (1) US9290536B2 (enExample)
EP (1) EP2683731B1 (enExample)
JP (1) JP6129084B2 (enExample)
KR (1) KR101956399B1 (enExample)
CN (1) CN103619866B (enExample)
AR (1) AR085666A1 (enExample)
AU (1) AU2012229244B2 (enExample)
BR (1) BR112013023174B1 (enExample)
CA (1) CA2829618C (enExample)
CL (1) CL2013002612A1 (enExample)
CO (1) CO6801741A2 (enExample)
CY (1) CY1121744T1 (enExample)
DK (1) DK2683731T3 (enExample)
EA (1) EA026847B1 (enExample)
ES (1) ES2729405T3 (enExample)
HR (1) HRP20191164T1 (enExample)
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ME (1) ME03469B (enExample)
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