KR101438839B1 - 글루카곤 유사 펩타이드 1 (glp-1) 약제학적 제제 - Google Patents
글루카곤 유사 펩타이드 1 (glp-1) 약제학적 제제 Download PDFInfo
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- KR101438839B1 KR101438839B1 KR1020087027774A KR20087027774A KR101438839B1 KR 101438839 B1 KR101438839 B1 KR 101438839B1 KR 1020087027774 A KR1020087027774 A KR 1020087027774A KR 20087027774 A KR20087027774 A KR 20087027774A KR 101438839 B1 KR101438839 B1 KR 101438839B1
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- South Korea
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- glp
- fdkp
- diketopiperazine
- molecule
- solution
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/19—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
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- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/26—Glucagons
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- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
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Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US74488206P | 2006-04-14 | 2006-04-14 | |
US60/744,882 | 2006-04-14 | ||
PCT/US2007/066728 WO2007121411A2 (en) | 2006-04-14 | 2007-04-16 | Glucagon-like peptide 1(glp-1) pharmaceutical formulations |
Related Child Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
KR1020147011316A Division KR101558829B1 (ko) | 2006-04-14 | 2007-04-16 | 글루카곤 유사 펩타이드 1 (glp-1) 약제학적 제제 |
Publications (2)
Publication Number | Publication Date |
---|---|
KR20080111533A KR20080111533A (ko) | 2008-12-23 |
KR101438839B1 true KR101438839B1 (ko) | 2014-10-02 |
Family
ID=38567214
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
KR1020087027774A KR101438839B1 (ko) | 2006-04-14 | 2007-04-16 | 글루카곤 유사 펩타이드 1 (glp-1) 약제학적 제제 |
KR1020157008571A KR20150042304A (ko) | 2006-04-14 | 2007-04-16 | 글루카곤 유사 펩타이드 1 (glp-1) 약제학적 제제 |
KR1020147011316A KR101558829B1 (ko) | 2006-04-14 | 2007-04-16 | 글루카곤 유사 펩타이드 1 (glp-1) 약제학적 제제 |
Family Applications After (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
KR1020157008571A KR20150042304A (ko) | 2006-04-14 | 2007-04-16 | 글루카곤 유사 펩타이드 1 (glp-1) 약제학적 제제 |
KR1020147011316A KR101558829B1 (ko) | 2006-04-14 | 2007-04-16 | 글루카곤 유사 펩타이드 1 (glp-1) 약제학적 제제 |
Country Status (11)
Country | Link |
---|---|
EP (1) | EP2010155A2 (ru) |
JP (3) | JP5415938B2 (ru) |
KR (3) | KR101438839B1 (ru) |
CN (2) | CN101453988A (ru) |
AU (1) | AU2007238000B2 (ru) |
BR (1) | BRPI0709964A2 (ru) |
CA (1) | CA2646400A1 (ru) |
HK (1) | HK1206241A1 (ru) |
MX (1) | MX2008013216A (ru) |
RU (3) | RU2542500C2 (ru) |
WO (1) | WO2007121411A2 (ru) |
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BRPI0709964A2 (pt) * | 2006-04-14 | 2011-08-02 | Mannkind Corp | formulações farmacêuticas contendo peptìdeo glucagon do tipo 1 (glp-1) |
US8785396B2 (en) | 2007-10-24 | 2014-07-22 | Mannkind Corporation | Method and composition for treating migraines |
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US8217047B2 (en) | 2008-05-27 | 2012-07-10 | Dmi Acquisition Corp. | Therapeutic methods and compounds |
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AR105284A1 (es) | 2015-07-10 | 2017-09-20 | Sanofi Sa | Derivados de exendina-4 como agonistas peptídicos duales específicos de los receptores de glp-1 / glucagón |
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WO2007121411A2 (en) | 2007-10-25 |
RU2409349C2 (ru) | 2011-01-20 |
WO2007121411A3 (en) | 2007-12-13 |
JP5415938B2 (ja) | 2014-02-12 |
HK1206241A1 (en) | 2016-01-08 |
AU2007238000A1 (en) | 2007-10-25 |
KR20150042304A (ko) | 2015-04-20 |
EP2010155A2 (en) | 2009-01-07 |
MX2008013216A (es) | 2008-10-27 |
CN104288756A (zh) | 2015-01-21 |
KR20140072138A (ko) | 2014-06-12 |
JP2016104736A (ja) | 2016-06-09 |
JP5898156B2 (ja) | 2016-04-06 |
JP2009533476A (ja) | 2009-09-17 |
RU2542500C2 (ru) | 2015-02-20 |
RU2014152320A (ru) | 2016-07-20 |
AU2007238000B2 (en) | 2013-01-17 |
KR20080111533A (ko) | 2008-12-23 |
BRPI0709964A2 (pt) | 2011-08-02 |
JP2014043445A (ja) | 2014-03-13 |
CA2646400A1 (en) | 2007-10-25 |
CN101453988A (zh) | 2009-06-10 |
RU2010137392A (ru) | 2012-03-20 |
RU2008144965A (ru) | 2010-05-20 |
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