KR101424306B1 - 메타스틴 유도체 및 그의 용도 - Google Patents

메타스틴 유도체 및 그의 용도 Download PDF

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KR101424306B1
KR101424306B1 KR1020097010545A KR20097010545A KR101424306B1 KR 101424306 B1 KR101424306 B1 KR 101424306B1 KR 1020097010545 A KR1020097010545 A KR 1020097010545A KR 20097010545 A KR20097010545 A KR 20097010545A KR 101424306 B1 KR101424306 B1 KR 101424306B1
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KR20090090315A (ko
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다이지 아사미
나오키 니시자와
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다케다 야쿠힌 고교 가부시키가이샤
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • C07K14/4701—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals not used
    • C07K14/4702—Regulators; Modulating activity
    • C07K14/4703—Inhibitors; Suppressors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
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    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/1703—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • A61K38/1709—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Endocrinology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Hematology (AREA)
  • Reproductive Health (AREA)
  • Immunology (AREA)
  • Zoology (AREA)
  • Pulmonology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Molecular Biology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Toxicology (AREA)
  • Urology & Nephrology (AREA)
  • Obesity (AREA)
  • Pregnancy & Childbirth (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
KR1020097010545A 2006-10-25 2007-10-24 메타스틴 유도체 및 그의 용도 Active KR101424306B1 (ko)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
JP2006290536 2006-10-25
JPJP-P-2006-290536 2006-10-25
JP2007021387 2007-01-31
JPJP-P-2007-021387 2007-01-31
JPJP-P-2007-221911 2007-08-28
JP2007221911 2007-08-28
PCT/JP2007/071169 WO2008050897A1 (en) 2006-10-25 2007-10-24 Metastin derivatives and use thereof

Publications (2)

Publication Number Publication Date
KR20090090315A KR20090090315A (ko) 2009-08-25
KR101424306B1 true KR101424306B1 (ko) 2014-08-01

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KR1020097010545A Active KR101424306B1 (ko) 2006-10-25 2007-10-24 메타스틴 유도체 및 그의 용도

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US (2) US7786083B2 (enExample)
EP (1) EP2081955B1 (enExample)
JP (2) JP2010507565A (enExample)
KR (1) KR101424306B1 (enExample)
AR (1) AR063367A1 (enExample)
AU (1) AU2007309969B2 (enExample)
BR (1) BRPI0717441B8 (enExample)
CA (1) CA2667537C (enExample)
CL (1) CL2007003053A1 (enExample)
CR (1) CR10799A (enExample)
CY (1) CY1116627T1 (enExample)
DK (1) DK2081955T3 (enExample)
EC (1) ECSP099279A (enExample)
ES (1) ES2539430T3 (enExample)
GE (1) GEP20125568B (enExample)
HR (1) HRP20150819T1 (enExample)
HU (1) HUE025291T2 (enExample)
IL (1) IL198046A (enExample)
JO (1) JO3048B1 (enExample)
MA (1) MA30887B1 (enExample)
ME (1) ME00786B (enExample)
MX (1) MX2009004148A (enExample)
MY (1) MY145975A (enExample)
NO (1) NO341584B1 (enExample)
NZ (1) NZ576375A (enExample)
PE (1) PE20081469A1 (enExample)
PL (1) PL2081955T3 (enExample)
PT (1) PT2081955E (enExample)
RS (1) RS54083B1 (enExample)
SI (1) SI2081955T1 (enExample)
TN (1) TN2009000140A1 (enExample)
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WO (1) WO2008050897A1 (enExample)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2511858A1 (en) 2002-12-26 2004-07-29 Takeda Pharmaceutical Company Limited Metastin derivative and use thereof
US7625869B2 (en) * 2004-06-25 2009-12-01 Takeda Pharmaceutical Company Limited Metastin derivatives and use thereof
US20090093615A1 (en) * 2005-12-22 2009-04-09 Takeda Pharmaceutical Company Limited Metastin derivatives and use thereof
AR058584A1 (es) 2005-12-22 2008-02-13 Takeda Pharmaceutical Derivados de metastina y uso de los mismos
US8404643B2 (en) 2005-12-22 2013-03-26 Takeda Pharmaceutical Company Limited Metastin derivatives and use thereof
US20090099334A1 (en) * 2005-12-22 2009-04-16 Takeda Pharmaceutical Company Limited Metastin derivatives and use thereof
WO2007125619A1 (ja) * 2006-04-26 2007-11-08 Kyoto University Ｇｐｒ５４アゴニスト活性を有する新規化合物
JO3048B1 (ar) 2006-10-25 2016-09-05 Takeda Pharmaceuticals Co مشتقات متاستين واستخدامها
US8110639B2 (en) * 2006-11-17 2012-02-07 Solvay Advanced Polymers, L.L.C. Transparent and flame retardant polysulfone compositions
EP2277900A4 (en) * 2008-04-24 2011-08-03 Takeda Pharmaceutical METASTINE DERIVATIVE AND ITS USE
WO2009139298A1 (ja) * 2008-04-30 2009-11-19 国立大学法人京都大学 メタスチン誘導体およびその用途
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