KR101155365B1 - 인간 단백질 타이로신 포스파타아제 억제제 및 사용 방법 - Google Patents

인간 단백질 타이로신 포스파타아제 억제제 및 사용 방법 Download PDF

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KR101155365B1
KR101155365B1 KR1020097001678A KR20097001678A KR101155365B1 KR 101155365 B1 KR101155365 B1 KR 101155365B1 KR 1020097001678 A KR1020097001678 A KR 1020097001678A KR 20097001678 A KR20097001678 A KR 20097001678A KR 101155365 B1 KR101155365 B1 KR 101155365B1
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ethyl
thiazol
phenylsulfamic acid
substituted
tert
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KR20090024819A (ko
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제프리 라일 그레이
칸데 아마라싱헤
신시아 모네사 클락
매튜 브라이언 마이어
라이언 니콜스
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에르피오 세러퓨틱스 인코포레이티드
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
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  • Immunology (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
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  • Dermatology (AREA)
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  • Molecular Biology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hematology (AREA)
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  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Hospice & Palliative Care (AREA)
  • Neurology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
KR1020097001678A 2006-06-27 2007-06-27 인간 단백질 타이로신 포스파타아제 억제제 및 사용 방법 Expired - Fee Related KR101155365B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US81673006P 2006-06-27 2006-06-27
US60/816,730 2006-06-27
PCT/US2007/014822 WO2008002569A2 (en) 2006-06-27 2007-06-27 Human protein tyrosine phosphatase inhibitors and methods of use

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KR20090024819A KR20090024819A (ko) 2009-03-09
KR101155365B1 true KR101155365B1 (ko) 2012-06-20

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US (13) US7622593B2 (enExample)
EP (3) EP2592072B1 (enExample)
JP (2) JP5232778B2 (enExample)
KR (1) KR101155365B1 (enExample)
CN (1) CN101506183B (enExample)
AU (1) AU2007265453B2 (enExample)
BR (1) BRPI0713570A2 (enExample)
CA (1) CA2657096C (enExample)
CO (1) CO6150144A2 (enExample)
DK (3) DK2041102T3 (enExample)
ES (3) ES2650598T3 (enExample)
IL (1) IL196128A (enExample)
MX (1) MX2009000288A (enExample)
NZ (1) NZ574407A (enExample)
PL (3) PL3323815T3 (enExample)
PT (3) PT2041102E (enExample)
RU (1) RU2447065C2 (enExample)
SI (1) SI2041102T1 (enExample)
WO (1) WO2008002569A2 (enExample)
ZA (1) ZA200900559B (enExample)

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AU2007237096C1 (en) 2006-04-07 2012-12-13 EyePoint Pharmaceuticals, Inc. Antibodies that bind human protein tyrosine phosphatase beta (HPTPbeta) and uses thereof
US7795444B2 (en) * 2006-06-27 2010-09-14 Warner Chilcott Company Human protein tyrosine phosphatase inhibitors and methods of use
US7622593B2 (en) * 2006-06-27 2009-11-24 The Procter & Gamble Company Human protein tyrosine phosphatase inhibitors and methods of use
US7589212B2 (en) 2006-06-27 2009-09-15 Procter & Gamble Company Human protein tyrosine phosphatase inhibitors and methods of use
US8846685B2 (en) 2006-06-27 2014-09-30 Aerpio Therapeutics Inc. Human protein tyrosine phosphatase inhibitors and methods of use
CN108635350A (zh) * 2009-01-12 2018-10-12 爱尔皮奥治疗有限公司 治疗血管渗漏综合征的方法
US9096555B2 (en) 2009-01-12 2015-08-04 Aerpio Therapeutics, Inc. Methods for treating vascular leak syndrome
AU2016203254B2 (en) * 2009-01-12 2018-09-13 EyePoint Pharmaceuticals, Inc. Methods for treating vascular leak syndrome
AU2014202211B2 (en) * 2009-01-12 2016-06-02 EyePoint Pharmaceuticals, Inc. Methods for treating vascular leak syndrome
CA2748765C (en) * 2009-07-06 2014-07-22 Akebia Therapeutics Inc. Compounds, compositions, and methods for preventing metastasis of cancer cells
US8883832B2 (en) 2009-07-06 2014-11-11 Aerpio Therapeutics Inc. Compounds, compositions, and methods for preventing metastasis of cancer cells
ES2644998T3 (es) 2009-11-06 2017-12-01 Aerpio Therapeutics Inc. Métodos para aumentar la estabilización del factor-1 alfa inducible por hipoxia
JP2013525290A (ja) * 2010-04-15 2013-06-20 ノバルティス アーゲー Ｋｓｐ阻害剤としてのオキサゾールおよびチアゾール化合物
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