KR101050872B1 - 술포닐 클로라이드 및 피리딘의 존재하에 오르토-아미노방향족 카르복실산 및 카르복실산으로부터 융합된옥사지논의 제조 방법 - Google Patents
술포닐 클로라이드 및 피리딘의 존재하에 오르토-아미노방향족 카르복실산 및 카르복실산으로부터 융합된옥사지논의 제조 방법 Download PDFInfo
- Publication number
- KR101050872B1 KR101050872B1 KR1020057001577A KR20057001577A KR101050872B1 KR 101050872 B1 KR101050872 B1 KR 101050872B1 KR 1020057001577 A KR1020057001577 A KR 1020057001577A KR 20057001577 A KR20057001577 A KR 20057001577A KR 101050872 B1 KR101050872 B1 KR 101050872B1
- Authority
- KR
- South Korea
- Prior art keywords
- formula
- compound
- carboxylic acid
- optionally substituted
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- 0 O=C1OC(I)=*C2C1CCCC*CCCC2 Chemical compound O=C1OC(I)=*C2C1CCCC*CCCC2 0.000 description 10
- KHYCMZWBPIHDPX-UHFFFAOYSA-N CC(c1cccc(C(c2ccc[s]2)=O)c1)C(O1)=Nc([s]cc2C)c2C1=O Chemical compound CC(c1cccc(C(c2ccc[s]2)=O)c1)C(O1)=Nc([s]cc2C)c2C1=O KHYCMZWBPIHDPX-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US40035202P | 2002-07-31 | 2002-07-31 | |
| US60/400,352 | 2002-07-31 | ||
| US44643803P | 2003-02-11 | 2003-02-11 | |
| US60/446,438 | 2003-02-11 | ||
| PCT/US2003/023821 WO2004011447A2 (en) | 2002-07-31 | 2003-07-29 | Method for preparing fused oxazinones from ortho-amino aromatic carboxylic acid and a carboxylic acid in the presence of a sulfonyl chloride and pyridine |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| KR20050026534A KR20050026534A (ko) | 2005-03-15 |
| KR101050872B1 true KR101050872B1 (ko) | 2011-07-20 |
Family
ID=31191366
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020057001577A Expired - Fee Related KR101050872B1 (ko) | 2002-07-31 | 2003-07-29 | 술포닐 클로라이드 및 피리딘의 존재하에 오르토-아미노방향족 카르복실산 및 카르복실산으로부터 융합된옥사지논의 제조 방법 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US7339057B2 (https=) |
| EP (1) | EP1549643B1 (https=) |
| JP (1) | JP2006501203A (https=) |
| KR (1) | KR101050872B1 (https=) |
| CN (1) | CN100422177C (https=) |
| AT (1) | ATE371657T1 (https=) |
| AU (1) | AU2003257028B2 (https=) |
| BR (1) | BR0313341A (https=) |
| DE (1) | DE60316006T2 (https=) |
| ES (1) | ES2293040T3 (https=) |
| IL (1) | IL165503A (https=) |
| TW (1) | TWI326283B (https=) |
| WO (1) | WO2004011447A2 (https=) |
Families Citing this family (43)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY142967A (en) | 2001-08-13 | 2011-01-31 | Du Pont | Method for controlling particular insect pests by applying anthranilamide compounds |
| AR036872A1 (es) | 2001-08-13 | 2004-10-13 | Du Pont | Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados |
| EP1423379B1 (en) | 2001-08-15 | 2008-05-28 | E.I. du Pont de Nemours and Company | Ortho-substituted aryl amides for controlling invertebrate pests |
| ES2319743T3 (es) | 2001-08-16 | 2009-05-12 | E.I. Du Pont De Nemours And Company | Antranilamidas sustituidas para controlar plagas de invertebrados. |
| TWI283164B (en) | 2001-09-21 | 2007-07-01 | Du Pont | Anthranilamide arthropodicide treatment |
| TWI343376B (en) | 2002-07-31 | 2011-06-11 | Du Pont | Method for preparing 3-halo-4, 5-dihydro-1h-pyrazoles |
| WO2004046129A2 (en) * | 2002-11-15 | 2004-06-03 | E.I. Du Pont De Nemours And Company | Novel anthranilamide insecticides |
| SI1599463T1 (sl) | 2003-01-28 | 2013-10-30 | E.I. Du Pont De Nemours And Company | Ciano antranilamidni insekticidi |
| KR20060008336A (ko) * | 2003-06-12 | 2006-01-26 | 이 아이 듀폰 디 네모아 앤드 캄파니 | 융합된 옥사지논 제조 방법 |
| US7126026B2 (en) * | 2003-11-13 | 2006-10-24 | Sanofi-Aventis Deutschland Gmbh | Process for preparing 4-pentafluorosulfanylbenzoylguanidines |
| US20050124666A1 (en) * | 2003-11-13 | 2005-06-09 | Aventis Pharma Deutschland Gmbh | Pentafluorosulfanylbenzoylguanidines, process for their preparation, use as a medicament or diagnostic aid, and medicament comprising same |
| US7317124B2 (en) | 2003-11-13 | 2008-01-08 | Sanofi-Aventis Deutschland Gmbh | Ortho-substituted pentafluorosulfanylbenzenes, process for their preparation and their use as valuable synthetic intermediates |
| RU2006139953A (ru) * | 2004-04-13 | 2008-05-20 | Е.И. Дюпон Де Немур Энд Компани (Us) | Антраниламидные инсектициды |
| ES2413442T3 (es) * | 2004-11-18 | 2013-07-16 | E. I. Du Pont De Nemours And Company | Insecticidas de antranilamida |
| TWI363756B (en) | 2004-12-07 | 2012-05-11 | Du Pont | Method for preparing n-phenylpyrazole-1-carboxamides |
| EP1871760B1 (en) * | 2005-04-20 | 2010-08-11 | Syngenta Participations AG | Cyano anthranilamide insecticides |
| US8143292B2 (en) | 2005-07-07 | 2012-03-27 | Basf Se | N-Thio-anthranilamid compounds and their use as pesticides |
| AU2006283181A1 (en) * | 2005-08-24 | 2007-03-01 | E. I. Du Pont De Nemours And Company | Anthranilamides for controlling invertebrate pests |
| PL2066662T3 (pl) | 2006-09-21 | 2013-05-31 | Kyorin Seiyaku Kk | Inhibitory hydrolaz serynowych |
| CN102134238A (zh) * | 2010-01-25 | 2011-07-27 | 中化蓝天集团有限公司 | 一种含一氟甲氧基吡唑的4h-苯并[1,3]噁嗪-4-酮类化合物、其制备方法及应用 |
| CN102285971B (zh) * | 2010-06-21 | 2013-12-18 | 中国中化股份有限公司 | 吡唑基喹唑啉酮类化合物及其应用 |
| CN102260245A (zh) * | 2011-06-02 | 2011-11-30 | 南开大学 | 2,3-二氢喹唑啉酮类衍生物及其制备方法和应用 |
| JP2014522872A (ja) | 2011-08-12 | 2014-09-08 | ビーエーエスエフ ソシエタス・ヨーロピア | N−チオ−アントラニルアミド化合物、及び殺有害生物剤としてのそれらの使用 |
| AU2012297002A1 (en) * | 2011-08-12 | 2014-03-06 | Basf Se | Process for preparing N-substituted 1H-pyrazole-5-carbonylchloride compounds |
| CA2843084A1 (en) | 2011-08-12 | 2013-02-21 | Basf Se | Anthranilamide compounds and their use as pesticides |
| JP2014529587A (ja) | 2011-08-12 | 2014-11-13 | ビーエーエスエフ ソシエタス・ヨーロピアBasf Se | N−チオ−アントラニルアミド化合物、及び殺有害生物剤としてのそれらの使用 |
| MX2014001604A (es) | 2011-08-12 | 2014-04-14 | Basf Se | Compuestos de antranilamida y sus usos como plaguicidas. |
| CN103889956A (zh) | 2011-08-18 | 2014-06-25 | 巴斯夫欧洲公司 | 用于防治无脊椎动物害虫的氨基甲酰基甲氧基-和氨基甲酰基甲硫基-及氨基甲酰基甲基氨基苯甲酰胺 |
| US20140243197A1 (en) | 2011-08-18 | 2014-08-28 | Basf Se | Carbamoylmethoxy- and carbamoylmethylthio- and carbamoylmethylamino benzamides for combating invertebrate pests |
| US20140200135A1 (en) | 2011-08-18 | 2014-07-17 | Basf Se | Carbamoylmethoxy- and carbamoylmethylthio- and carbamoylmethylamino benzamides for combating invertebrate pests |
| CA2873266A1 (en) | 2012-05-24 | 2013-11-28 | Basf Se | N-thio-anthranilamide compounds and their use as pesticides |
| EP2928471B1 (en) | 2012-12-06 | 2020-10-14 | Celgene Quanticel Research, Inc. | Histone demethylase inhibitors |
| CN106366046B (zh) * | 2016-08-29 | 2019-12-31 | 鲁南制药集团股份有限公司 | 一种新利司他的制备方法 |
| CN106366047B (zh) * | 2016-08-31 | 2019-12-31 | 鲁南制药集团股份有限公司 | 一种一锅法制备新利司他的方法 |
| CN107033135B (zh) * | 2017-05-26 | 2020-09-11 | 浙江省诸暨合力化学对外贸易有限公司 | 一种制备异噁嗪酮化合物的方法及其应用 |
| CN108033944B (zh) * | 2017-12-28 | 2020-10-16 | 利尔化学股份有限公司 | 氯虫苯甲酰胺杂质制备工艺 |
| CN108689988A (zh) * | 2018-06-22 | 2018-10-23 | 南开大学 | 含n-芳基吡咯的邻甲酰氨基苯甲酰胺类化合物与制备方法和应用 |
| CN113692406B (zh) | 2019-02-18 | 2024-07-23 | Pi工业有限公司 | 制备邻甲酰胺基苯甲酰胺类化合物及其中间体的方法 |
| CN111825653A (zh) | 2019-04-19 | 2020-10-27 | 安道麦马克西姆有限公司 | 取代吡唑类化合物的制备及其作为邻氨基苯甲酰胺前体的用途 |
| CN111423431B (zh) * | 2020-04-01 | 2022-10-28 | 利尔化学股份有限公司 | 一种氯虫苯甲酰胺及其中间体的制备方法 |
| AR123593A1 (es) | 2020-09-26 | 2022-12-21 | Pi Industries Ltd | Un proceso para la síntesis de compuestos antranílicos de ácido / amida e intermedios de los mismos |
| AU2022331725A1 (en) | 2021-08-19 | 2024-03-07 | Syngenta Crop Protection Ag | Method for controlling diamide resistant pests & compounds therefor |
| WO2023110710A1 (en) * | 2021-12-13 | 2023-06-22 | Syngenta Crop Protection Ag | Method for controlling diamide resistant pests & compounds therefor |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH07309851A (ja) * | 1994-05-16 | 1995-11-28 | Fuji Chem Ind Co Ltd | ベンゾオキサジノン誘導体の製造方法 |
| US5932726A (en) * | 1996-12-16 | 1999-08-03 | Dupont Pharmaceuticals Company | Asymmetric synthesis of benzoxazinones |
| JP2001519810A (ja) * | 1997-04-07 | 2001-10-23 | デュポン ファーマシューティカルズ カンパニー | 新規中間体を経由するベンゾオキサジノン類の不斉合成 |
| MY138097A (en) | 2000-03-22 | 2009-04-30 | Du Pont | Insecticidal anthranilamides |
| AU2002227243A1 (en) * | 2000-12-11 | 2002-06-24 | E.I. Du Pont De Nemours And Company | Quinazolinones and pyridinopyrimidinones for controlling invertebrate pests |
| AR036872A1 (es) * | 2001-08-13 | 2004-10-13 | Du Pont | Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados |
| MY142967A (en) | 2001-08-13 | 2011-01-31 | Du Pont | Method for controlling particular insect pests by applying anthranilamide compounds |
| TWI327566B (en) * | 2001-08-13 | 2010-07-21 | Du Pont | Novel substituted ihydro 3-halo-1h-pyrazole-5-carboxylates,their preparation and use |
| DE60236600D1 (de) | 2001-08-13 | 2010-07-15 | Du Pont | Substituierte 1h-dihydropyrazole, ihre herstellung und verwendung |
| TWI283164B (en) | 2001-09-21 | 2007-07-01 | Du Pont | Anthranilamide arthropodicide treatment |
| TWI343376B (en) | 2002-07-31 | 2011-06-11 | Du Pont | Method for preparing 3-halo-4, 5-dihydro-1h-pyrazoles |
-
2003
- 2003-07-02 TW TW092118080A patent/TWI326283B/zh not_active IP Right Cessation
- 2003-07-29 US US10/518,324 patent/US7339057B2/en not_active Expired - Lifetime
- 2003-07-29 AU AU2003257028A patent/AU2003257028B2/en not_active Ceased
- 2003-07-29 JP JP2004524204A patent/JP2006501203A/ja active Pending
- 2003-07-29 DE DE60316006T patent/DE60316006T2/de not_active Expired - Lifetime
- 2003-07-29 WO PCT/US2003/023821 patent/WO2004011447A2/en not_active Ceased
- 2003-07-29 CN CNB038182025A patent/CN100422177C/zh not_active Expired - Lifetime
- 2003-07-29 ES ES03772097T patent/ES2293040T3/es not_active Expired - Lifetime
- 2003-07-29 BR BR0313341-9A patent/BR0313341A/pt not_active IP Right Cessation
- 2003-07-29 AT AT03772097T patent/ATE371657T1/de not_active IP Right Cessation
- 2003-07-29 KR KR1020057001577A patent/KR101050872B1/ko not_active Expired - Fee Related
- 2003-07-29 EP EP03772097A patent/EP1549643B1/en not_active Expired - Lifetime
-
2004
- 2004-12-01 IL IL165503A patent/IL165503A/en not_active IP Right Cessation
Non-Patent Citations (1)
| Title |
|---|
| Organic Preparations and Procedures International 25(5): 588-590(1993)* |
Also Published As
| Publication number | Publication date |
|---|---|
| EP1549643B1 (en) | 2007-08-29 |
| EP1549643A2 (en) | 2005-07-06 |
| TW200410962A (en) | 2004-07-01 |
| TWI326283B (en) | 2010-06-21 |
| WO2004011447A2 (en) | 2004-02-05 |
| WO2004011447A3 (en) | 2004-03-18 |
| DE60316006T2 (de) | 2008-05-15 |
| ES2293040T3 (es) | 2008-03-16 |
| AU2003257028A1 (en) | 2004-02-16 |
| IL165503A0 (en) | 2006-01-15 |
| KR20050026534A (ko) | 2005-03-15 |
| BR0313341A (pt) | 2005-07-12 |
| CN100422177C (zh) | 2008-10-01 |
| ATE371657T1 (de) | 2007-09-15 |
| US7339057B2 (en) | 2008-03-04 |
| IL165503A (en) | 2010-11-30 |
| DE60316006D1 (de) | 2007-10-11 |
| CN1671703A (zh) | 2005-09-21 |
| US20050215785A1 (en) | 2005-09-29 |
| AU2003257028B2 (en) | 2010-12-09 |
| JP2006501203A (ja) | 2006-01-12 |
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