KR100823805B1 - 5-ｈｔ6 수용체, 5-ｈｔ2ａ 수용체 또는 둘다를 조절하기에유용한 아릴설포닐 벤조다이옥산 - Google Patents

5-ｈｔ6 수용체, 5-ｈｔ2ａ 수용체 또는 둘다를 조절하기에유용한 아릴설포닐 벤조다이옥산 Download PDF

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KR100823805B1
KR100823805B1 KR1020067023073A KR20067023073A KR100823805B1 KR 100823805 B1 KR100823805 B1 KR 100823805B1 KR 1020067023073 A KR1020067023073 A KR 1020067023073A KR 20067023073 A KR20067023073 A KR 20067023073A KR 100823805 B1 KR100823805 B1 KR 100823805B1
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alkyl
formula
dihydro
benzo
benzenesulfonyl
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KR20070009664A (ko
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제이콥 버거
슈 하이 자오
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에프. 호프만-라 로슈 아게
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    • C07—ORGANIC CHEMISTRY
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    • C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes
    • C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
    • C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D319/20—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring with substituents attached to the hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
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    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
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  • Hospice & Palliative Care (AREA)
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  • Diabetes (AREA)
  • Hematology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
KR1020067023073A 2004-05-05 2005-04-27 5-ｈｔ6 수용체, 5-ｈｔ2ａ 수용체 또는 둘다를 조절하기에유용한 아릴설포닐 벤조다이옥산 KR100823805B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US56831404P 2004-05-05 2004-05-05
US60/568,314 2004-05-05

Publications (2)

Publication Number Publication Date
KR20070009664A KR20070009664A (ko) 2007-01-18
KR100823805B1 true KR100823805B1 (ko) 2008-04-21

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KR1020067023073A KR100823805B1 (ko) 2004-05-05 2005-04-27 5-ｈｔ6 수용체, 5-ｈｔ2ａ 수용체 또는 둘다를 조절하기에유용한 아릴설포닐 벤조다이옥산

Country Status (21)

Country Link
US (1) US7368567B2 (ru)
EP (1) EP1748995B1 (ru)
JP (1) JP2007536302A (ru)
KR (1) KR100823805B1 (ru)
CN (1) CN100540546C (ru)
AR (1) AR048936A1 (ru)
AT (1) ATE458727T1 (ru)
AU (1) AU2005238179B2 (ru)
BR (1) BRPI0510642A (ru)
CA (1) CA2566196A1 (ru)
DE (1) DE602005019562D1 (ru)
ES (1) ES2338668T3 (ru)
HK (1) HK1104533A1 (ru)
IL (1) IL178819A0 (ru)
MX (1) MXPA06012621A (ru)
NO (1) NO20065510L (ru)
NZ (1) NZ550441A (ru)
RU (1) RU2372344C2 (ru)
TW (1) TWI298636B (ru)
WO (1) WO2005105776A1 (ru)
ZA (1) ZA200608588B (ru)

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ES2359725T3 (es) * 2004-09-30 2011-05-26 F. Hoffmann-La Roche Ag Composiciones y métodos para el tratamiento de trastornos cognitivos.
CN101119989B (zh) * 2004-12-21 2010-06-09 弗·哈夫曼-拉罗切有限公司 色满衍生物及其在治疗cns疾病中的用途
JP2008538575A (ja) * 2005-04-22 2008-10-30 ワイス ベンゾジオキサンおよびベンゾジオキソラン誘導体ならびにそれらの使用
NZ567285A (en) 2005-11-03 2010-06-25 Hoffmann La Roche Arylsulfonylchromans as 5-HT6 inhibitors indolylmaleimide derivatives as protein kinase inhibitors
WO2007120596A1 (en) * 2006-04-12 2007-10-25 Wyeth DIHYDRO[1,4]DIOXINO[2,3-e]INDAZOLE DERIVATIVES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS
JP2009541249A (ja) * 2006-06-20 2009-11-26 エフ．ホフマン−ラ ロシュ アーゲー アリールスルホニルナフタレン誘導体およびその使用
FR2913886B1 (fr) 2007-03-22 2012-03-02 Guerbet Sa Utilisation de nanoparticules metalliques dans le diagnostique de la maladie d'alzheimer
KR20100135325A (ko) * 2008-04-29 2010-12-24 엔에스아베 필리알 아프 뉴로서치 스웨덴 아베 스베리게 도파민 신경전달의 조절제
US20110105462A1 (en) * 2008-04-29 2011-05-05 Nsab, Filial Af Neurosearch Sweden Ab, Sverige Modulators of dopamine neurotransmission
AU2009242095A1 (en) 2008-04-29 2009-11-05 Nsab, Filial Af Neurosearch Sweden Ab, Sverige Modulators of dopamine neurotransmission
CN114890978B (zh) * 2022-04-19 2023-07-25 宿迁医美科技有限公司 酚类化合物及其制备方法和应用

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Also Published As

Publication number Publication date
RU2372344C2 (ru) 2009-11-10
CN1960983A (zh) 2007-05-09
DE602005019562D1 (de) 2010-04-08
TW200605894A (en) 2006-02-16
AU2005238179B2 (en) 2010-08-26
EP1748995B1 (en) 2010-02-24
BRPI0510642A (pt) 2007-11-20
ES2338668T3 (es) 2010-05-11
RU2006138180A (ru) 2008-06-10
TWI298636B (en) 2008-07-11
CA2566196A1 (en) 2005-11-10
MXPA06012621A (es) 2006-12-15
ZA200608588B (en) 2008-06-25
EP1748995A1 (en) 2007-02-07
CN100540546C (zh) 2009-09-16
US7368567B2 (en) 2008-05-06
ATE458727T1 (de) 2010-03-15
KR20070009664A (ko) 2007-01-18
WO2005105776A1 (en) 2005-11-10
NZ550441A (en) 2009-07-31
WO2005105776A8 (en) 2007-01-11
JP2007536302A (ja) 2007-12-13
NO20065510L (no) 2007-01-12
AU2005238179A1 (en) 2005-11-10
AR048936A1 (es) 2006-06-14
US20050250943A1 (en) 2005-11-10
HK1104533A1 (en) 2008-01-18
IL178819A0 (en) 2007-03-08

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