JPWO2021229152A5 - - Google Patents

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Publication number
JPWO2021229152A5
JPWO2021229152A5 JP2022568879A JP2022568879A JPWO2021229152A5 JP WO2021229152 A5 JPWO2021229152 A5 JP WO2021229152A5 JP 2022568879 A JP2022568879 A JP 2022568879A JP 2022568879 A JP2022568879 A JP 2022568879A JP WO2021229152 A5 JPWO2021229152 A5 JP WO2021229152A5
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JP
Japan
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compound
methylsulfonyl
methyl
alkyl
pyran
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JP2022568879A
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English (en)
Japanese (ja)
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JP7789697B2 (ja
JP2023525137A (ja
JP2023525137A5 (https=
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Priority claimed from PCT/FI2021/050353 external-priority patent/WO2021229152A1/en
Publication of JP2023525137A publication Critical patent/JP2023525137A/ja
Publication of JPWO2021229152A5 publication Critical patent/JPWO2021229152A5/ja
Publication of JP2023525137A5 publication Critical patent/JP2023525137A5/ja
Priority to JP2025244683A priority Critical patent/JP2026048803A/ja
Application granted granted Critical
Publication of JP7789697B2 publication Critical patent/JP7789697B2/ja
Active legal-status Critical Current
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JP2022568879A 2020-05-14 2021-05-12 Cyp11a1阻害剤 Active JP7789697B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025244683A JP2026048803A (ja) 2020-05-14 2025-12-10 Cyp11a1阻害剤

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FI20205486 2020-05-14
FI20205486 2020-05-14
PCT/FI2021/050353 WO2021229152A1 (en) 2020-05-14 2021-05-12 Cyp11a1 inhibitors

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025244683A Division JP2026048803A (ja) 2020-05-14 2025-12-10 Cyp11a1阻害剤

Publications (4)

Publication Number Publication Date
JP2023525137A JP2023525137A (ja) 2023-06-14
JPWO2021229152A5 true JPWO2021229152A5 (https=) 2024-05-22
JP2023525137A5 JP2023525137A5 (https=) 2024-05-22
JP7789697B2 JP7789697B2 (ja) 2025-12-22

Family

ID=76325569

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022568879A Active JP7789697B2 (ja) 2020-05-14 2021-05-12 Cyp11a1阻害剤
JP2025244683A Pending JP2026048803A (ja) 2020-05-14 2025-12-10 Cyp11a1阻害剤

Family Applications After (1)

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JP2025244683A Pending JP2026048803A (ja) 2020-05-14 2025-12-10 Cyp11a1阻害剤

Country Status (8)

Country Link
US (1) US20230192677A1 (https=)
EP (1) EP4149924A1 (https=)
JP (2) JP7789697B2 (https=)
KR (1) KR20230010723A (https=)
CN (1) CN115551831A (https=)
AU (1) AU2021269872A1 (https=)
CA (1) CA3178067A1 (https=)
WO (1) WO2021229152A1 (https=)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN117242056A (zh) * 2021-03-26 2023-12-15 北京加科思新药研发有限公司 用作sting激动剂的新型化合物及其用途
PE20241583A1 (es) * 2021-09-28 2024-08-01 Orion Corp Inhibidor de cyp11a1 para su uso en el tratamiento del cancer de prostata
WO2023084158A1 (en) * 2021-11-10 2023-05-19 Orion Corporation Cyp11a1 inhibitors
CN115304591B (zh) * 2022-07-08 2024-10-01 广州中医药大学(广州中医药研究院) 一种桥环甾体合成酶抑制剂及其制备方法和应用
CN118307519A (zh) * 2023-01-06 2024-07-09 上海闻耐医药科技有限公司 一类cyp11a1抑制剂化合物及其制备方法和用途
WO2024199262A1 (zh) * 2023-03-29 2024-10-03 西藏海思科制药有限公司 Cyp11a1抑制剂及其用途
WO2024199421A1 (zh) * 2023-03-30 2024-10-03 山东轩竹医药科技有限公司 Cyp11a1抑制剂
CN121039123A (zh) * 2023-04-21 2025-11-28 西藏海思科制药有限公司 Cyp11a1抑制剂及其用途
AU2024270498A1 (en) * 2023-05-11 2025-11-27 Foshan Ionova Biotherapeutics Co., Inc. Novel compounds as cyp11a1 inhibitors and methods of use thereof
CN121605106A (zh) * 2023-07-27 2026-03-03 优领医药科技(香港)有限公司 Cyp11a1抑制剂
CN121889383A (zh) * 2023-09-08 2026-04-17 深圳众格生物科技有限公司 一种cyp11a1抑制剂、其制备方法及其应用
WO2025168117A1 (zh) * 2024-02-08 2025-08-14 盛睿泽华医药科技(苏州)有限公司 一种多环化合物及其制备方法和应用
WO2025237211A1 (zh) * 2024-05-11 2025-11-20 辽宁海思科制药有限公司 一种cyp11a1抑制剂的晶型物及其制备方法和应用
WO2025247149A1 (zh) * 2024-05-27 2025-12-04 辽宁海思科制药有限公司 一种cyp11a1抑制剂的盐及其晶型、其制备方法和应用
WO2026002207A1 (en) * 2024-06-28 2026-01-02 Acerand Therapeutics (Hong Kong) Limited Heterocyclic compounds as cyp11a1 inhibitors
WO2026040949A1 (zh) * 2024-08-19 2026-02-26 辽宁海思科制药有限公司 一种cyp11a1抑制剂的药物组合物及其制备方法和用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1471063A1 (en) 2003-02-28 2004-10-27 Exonhit Therapeutics S.A. Compounds and methods of treating cell proliferative diseases, retinopathies and arthritis
AR088320A1 (es) 2011-10-14 2014-05-28 Incyte Corp Derivados de isoindolinona y pirrolopiridinona como inhibidores de akt
US10357484B2 (en) 2015-07-17 2019-07-23 Takeda Pharmaceutical Company Limited Heterocyclic compound
AR110412A1 (es) * 2016-12-22 2019-03-27 Orion Corp Inhibidores de la cyp11a1

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