JP2023525137A5 - - Google Patents
Info
- Publication number
- JP2023525137A5 JP2023525137A5 JP2022568879A JP2022568879A JP2023525137A5 JP 2023525137 A5 JP2023525137 A5 JP 2023525137A5 JP 2022568879 A JP2022568879 A JP 2022568879A JP 2022568879 A JP2022568879 A JP 2022568879A JP 2023525137 A5 JP2023525137 A5 JP 2023525137A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- methylsulfonyl
- methyl
- alkyl
- pyran
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2025244683A JP2026048803A (ja) | 2020-05-14 | 2025-12-10 | Cyp11a1阻害剤 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FI20205486 | 2020-05-14 | ||
| FI20205486 | 2020-05-14 | ||
| PCT/FI2021/050353 WO2021229152A1 (en) | 2020-05-14 | 2021-05-12 | Cyp11a1 inhibitors |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025244683A Division JP2026048803A (ja) | 2020-05-14 | 2025-12-10 | Cyp11a1阻害剤 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023525137A JP2023525137A (ja) | 2023-06-14 |
| JP2023525137A5 true JP2023525137A5 (https=) | 2024-05-22 |
| JP7789697B2 JP7789697B2 (ja) | 2025-12-22 |
Family
ID=76325569
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022568879A Active JP7789697B2 (ja) | 2020-05-14 | 2021-05-12 | Cyp11a1阻害剤 |
| JP2025244683A Pending JP2026048803A (ja) | 2020-05-14 | 2025-12-10 | Cyp11a1阻害剤 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025244683A Pending JP2026048803A (ja) | 2020-05-14 | 2025-12-10 | Cyp11a1阻害剤 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20230192677A1 (https=) |
| EP (1) | EP4149924A1 (https=) |
| JP (2) | JP7789697B2 (https=) |
| KR (1) | KR20230010723A (https=) |
| CN (1) | CN115551831A (https=) |
| AU (1) | AU2021269872A1 (https=) |
| CA (1) | CA3178067A1 (https=) |
| WO (1) | WO2021229152A1 (https=) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP4313946A4 (en) * | 2021-03-26 | 2025-03-12 | Jacobio Pharmaceuticals Co., Ltd. | NEW COMPOUNDS AS STING AGONISTS AND THEIR USES |
| US20250367184A1 (en) * | 2021-09-28 | 2025-12-04 | Orion Corporation | Cyp11a1 inhibitor for use in the treatment of prostate cancer |
| WO2023084158A1 (en) * | 2021-11-10 | 2023-05-19 | Orion Corporation | Cyp11a1 inhibitors |
| CN115304591B (zh) * | 2022-07-08 | 2024-10-01 | 广州中医药大学(广州中医药研究院) | 一种桥环甾体合成酶抑制剂及其制备方法和应用 |
| CN118307519A (zh) * | 2023-01-06 | 2024-07-09 | 上海闻耐医药科技有限公司 | 一类cyp11a1抑制剂化合物及其制备方法和用途 |
| CN121002012A (zh) * | 2023-03-29 | 2025-11-21 | 西藏海思科制药有限公司 | Cyp11a1抑制剂及其用途 |
| WO2024199421A1 (zh) * | 2023-03-30 | 2024-10-03 | 山东轩竹医药科技有限公司 | Cyp11a1抑制剂 |
| CN121039123A (zh) * | 2023-04-21 | 2025-11-28 | 西藏海思科制药有限公司 | Cyp11a1抑制剂及其用途 |
| KR20260040160A (ko) * | 2023-05-11 | 2026-03-24 | 셴젠 이오노바 라이프 사이언스 시오., 엘티디. | Cyp11a1 억제제로서의 신규 화합물 및 그 용도 |
| WO2025021182A1 (en) * | 2023-07-27 | 2025-01-30 | Acerand Therapeutics (Hong Kong) Limited | Cyp11a1 inhibitors |
| WO2025051216A1 (zh) * | 2023-09-08 | 2025-03-13 | 深圳众格生物科技有限公司 | 一种cyp11a1抑制剂、其制备方法及其应用 |
| WO2025168117A1 (zh) * | 2024-02-08 | 2025-08-14 | 盛睿泽华医药科技(苏州)有限公司 | 一种多环化合物及其制备方法和应用 |
| WO2025237211A1 (zh) * | 2024-05-11 | 2025-11-20 | 辽宁海思科制药有限公司 | 一种cyp11a1抑制剂的晶型物及其制备方法和应用 |
| WO2025247149A1 (zh) * | 2024-05-27 | 2025-12-04 | 辽宁海思科制药有限公司 | 一种cyp11a1抑制剂的盐及其晶型、其制备方法和应用 |
| WO2026002207A1 (en) * | 2024-06-28 | 2026-01-02 | Acerand Therapeutics (Hong Kong) Limited | Heterocyclic compounds as cyp11a1 inhibitors |
| WO2026040949A1 (zh) * | 2024-08-19 | 2026-02-26 | 辽宁海思科制药有限公司 | 一种cyp11a1抑制剂的药物组合物及其制备方法和用途 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1471063A1 (en) | 2003-02-28 | 2004-10-27 | Exonhit Therapeutics S.A. | Compounds and methods of treating cell proliferative diseases, retinopathies and arthritis |
| WO2013056015A1 (en) | 2011-10-14 | 2013-04-18 | Incyte Corporation | Isoindolinone and pyrrolopyridinone derivatives as akt inhibitors |
| JPWO2017014170A1 (ja) | 2015-07-17 | 2018-04-26 | 武田薬品工業株式会社 | 複素環化合物 |
| AR110412A1 (es) * | 2016-12-22 | 2019-03-27 | Orion Corp | Inhibidores de la cyp11a1 |
-
2021
- 2021-05-12 AU AU2021269872A patent/AU2021269872A1/en active Pending
- 2021-05-12 CA CA3178067A patent/CA3178067A1/en active Pending
- 2021-05-12 KR KR1020227043775A patent/KR20230010723A/ko active Pending
- 2021-05-12 WO PCT/FI2021/050353 patent/WO2021229152A1/en not_active Ceased
- 2021-05-12 CN CN202180034328.3A patent/CN115551831A/zh active Pending
- 2021-05-12 JP JP2022568879A patent/JP7789697B2/ja active Active
- 2021-05-12 US US17/924,857 patent/US20230192677A1/en active Pending
- 2021-05-12 EP EP21730972.3A patent/EP4149924A1/en active Pending
-
2025
- 2025-12-10 JP JP2025244683A patent/JP2026048803A/ja active Pending
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