JPWO2020075080A5 - - Google Patents

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Publication number
JPWO2020075080A5
JPWO2020075080A5 JP2021519876A JP2021519876A JPWO2020075080A5 JP WO2020075080 A5 JPWO2020075080 A5 JP WO2020075080A5 JP 2021519876 A JP2021519876 A JP 2021519876A JP 2021519876 A JP2021519876 A JP 2021519876A JP WO2020075080 A5 JPWO2020075080 A5 JP WO2020075080A5
Authority
JP
Japan
Prior art keywords
alkyl
optionally substituted
independently selected
halo
substituents independently
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021519876A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022512676A5 (https=
JP2022512676A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2019/058591 external-priority patent/WO2020075080A1/en
Publication of JP2022512676A publication Critical patent/JP2022512676A/ja
Publication of JP2022512676A5 publication Critical patent/JP2022512676A5/ja
Publication of JPWO2020075080A5 publication Critical patent/JPWO2020075080A5/ja
Withdrawn legal-status Critical Current

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JP2021519876A 2018-10-10 2019-10-09 大環状インフルエンザエンドヌクレアーゼ阻害剤 Withdrawn JP2022512676A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862744060P 2018-10-10 2018-10-10
US62/744,060 2018-10-10
PCT/IB2019/058591 WO2020075080A1 (en) 2018-10-10 2019-10-09 Macrocyclic flu endonuclease inhibitors

Publications (3)

Publication Number Publication Date
JP2022512676A JP2022512676A (ja) 2022-02-07
JP2022512676A5 JP2022512676A5 (https=) 2022-10-17
JPWO2020075080A5 true JPWO2020075080A5 (https=) 2022-10-17

Family

ID=68242803

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021519876A Withdrawn JP2022512676A (ja) 2018-10-10 2019-10-09 大環状インフルエンザエンドヌクレアーゼ阻害剤

Country Status (10)

Country Link
US (2) US11312727B1 (https=)
EP (1) EP3864020A1 (https=)
JP (1) JP2022512676A (https=)
KR (1) KR20210074329A (https=)
CN (1) CN113195502A (https=)
AU (1) AU2019359539A1 (https=)
CA (1) CA3115792A1 (https=)
MX (1) MX2021004182A (https=)
TW (1) TW202035424A (https=)
WO (1) WO2020075080A1 (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2020197991A1 (en) 2019-03-22 2020-10-01 Gilead Sciences, Inc. Bridged tricyclic carbamoylpyridone compounds and their pharmaceutical use
WO2021191872A1 (en) * 2020-03-26 2021-09-30 Janssen Biopharma, Inc. Heteroaryl-substituted macrocyclic flu endonuclease inhibitors
CN113444010B (zh) * 2020-03-28 2023-09-05 南京正大天晴制药有限公司 一种沙芬酰胺有关物质的制备方法
US12516070B2 (en) 2020-05-21 2026-01-06 Cisen Pharmaceutical Co., Ltd Fused ring derivatives and use thereof in pharmacy
TW202146413A (zh) * 2020-06-12 2021-12-16 大陸商上海翰森生物醫藥科技有限公司 含吡啶酮稠環類衍生物抑制劑、其製備方法和應用
CA3192145A1 (en) 2020-09-30 2022-04-07 Gilead Sciences, Inc. Bridged tricyclic carbamoylpyridone compounds and uses thereof
WO2022105669A1 (zh) * 2020-11-17 2022-05-27 南京明德新药研发有限公司 含Se大环类化合物
FI4196479T3 (fi) * 2021-01-19 2024-01-17 Gilead Sciences Inc Substituoituja pyridotriatsiiniyhdisteitä ja niiden käyttöjä
EP4384178A4 (en) * 2021-08-11 2025-07-02 Merck Sharp & Dohme Llc POLYCYCLIC CAP-DEPENDENT ENDONUCLEASE INHIBITORS FOR THE TREATMENT OR PREVENTION OF INFLUENZA
CN118317964A (zh) * 2021-11-17 2024-07-09 辰欣药业股份有限公司 一种稠环衍生物的晶型及其制备方法
WO2025015300A2 (en) * 2023-07-12 2025-01-16 Apac Pharma, Llc Hepoxilin analogs, methods, uses, and processes for preparation thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LT2444400T (lt) * 2009-06-15 2018-06-11 Shionogi & Co., Ltd. Pakeistasis policiklinis karbamoilpiridono darinys
MX2013003139A (es) * 2010-09-24 2013-06-18 Shionogi & Co Profarmaco de derivado de carbamoilpiridona policiclica substituida.
ES2724581T3 (es) * 2013-09-12 2019-09-12 Janssen Biopharma Inc Compuestos de piridazinona y usos de los mismos
JOP20170169A1 (ar) * 2016-08-29 2019-01-30 Novartis Ag مركبات بيريدازين ثلاثية الحلقة مندمجة تفيد في علاج العدوى بفيروس أورثوميكسو

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