JPS63284169A - フォルスコリンの新規な誘導体、その製造方法及び中間体、医薬としてのその使用、並びにそれを含有する医薬組成物 - Google Patents

フォルスコリンの新規な誘導体、その製造方法及び中間体、医薬としてのその使用、並びにそれを含有する医薬組成物

Info

Publication number
JPS63284169A
JPS63284169A JP63109294A JP10929488A JPS63284169A JP S63284169 A JPS63284169 A JP S63284169A JP 63109294 A JP63109294 A JP 63109294A JP 10929488 A JP10929488 A JP 10929488A JP S63284169 A JPS63284169 A JP S63284169A
Authority
JP
Japan
Prior art keywords
formula
compound
group
treated
tables
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP63109294A
Other languages
English (en)
Japanese (ja)
Inventor
ベルナール・デルペ
ロベール・レ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA
Publication of JPS63284169A publication Critical patent/JPS63284169A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78—Ring systems having three or more relevant rings
    • C07D311/92—Naphthopyrans; Hydrogenated naphthopyrans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Ophthalmology & Optometry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)
JP63109294A 1987-05-04 1988-05-06 フォルスコリンの新規な誘導体、その製造方法及び中間体、医薬としてのその使用、並びにそれを含有する医薬組成物 Pending JPS63284169A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR87-06242 1987-05-04
FR8706242A FR2614891B1 (fr) 1987-05-04 1987-05-04 Nouveaux derives de la forskoline, leur procede de preparation, leur application comme medicaments, les compositions pharmaceutiques les renfermant ainsi que des intermediaires de leur procede de preparation

Publications (1)

Publication Number Publication Date
JPS63284169A true JPS63284169A (ja) 1988-11-21

Family

ID=9350729

Family Applications (1)

Application Number Title Priority Date Filing Date
JP63109294A Pending JPS63284169A (ja) 1987-05-04 1988-05-06 フォルスコリンの新規な誘導体、その製造方法及び中間体、医薬としてのその使用、並びにそれを含有する医薬組成物

Country Status (7)

Country Link
JP (1) JPS63284169A (enrdf_load_stackoverflow)
CH (1) CH676598A5 (enrdf_load_stackoverflow)
DE (1) DE3815213A1 (enrdf_load_stackoverflow)
FR (1) FR2614891B1 (enrdf_load_stackoverflow)
GB (1) GB2205564A (enrdf_load_stackoverflow)
IT (1) IT1219567B (enrdf_load_stackoverflow)
NL (1) NL8801174A (enrdf_load_stackoverflow)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5268471A (en) * 1990-07-24 1993-12-07 Hoechst Aktiengesellschaft Process for the preparation of 6-acyl, 7-acyl, and 6,7-diacyl analogues of forskolin and intermediates thereof
KR920002575A (ko) * 1990-07-24 1992-02-28 이젠브루크, 라피체 포르스콜린의 6-아실,7-아실 및 6,7- 디아실동족체 및 이의 중간체를 제조하는 방법
FI913506A7 (fi) * 1990-07-24 1992-01-25 Hoechst Ag Foerfarande foer framstaellning av 6-(substituerat aminopropionyl)-derivat av forskolin.
CN1089092C (zh) * 1997-10-30 2002-08-14 中国科学院动物研究所 一种促分化抑增殖抗癌药二萜类化合物及其制备方法和用途

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS59152380A (ja) * 1982-12-27 1984-08-31 シエリング・コ−ポレ−シヨン ラブダン誘導体を含む医薬組成物

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE43545B1 (en) * 1975-09-06 1981-03-25 Hoechst Ag Pharmacologically active substance obtainable from plants
AU2717777A (en) * 1976-07-21 1979-01-25 Hoechst Ag Pharmacologically effective substance from plants belonging to the family of labiatae

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS59152380A (ja) * 1982-12-27 1984-08-31 シエリング・コ−ポレ−シヨン ラブダン誘導体を含む医薬組成物

Also Published As

Publication number Publication date
GB2205564A (en) 1988-12-14
FR2614891B1 (fr) 1991-05-24
FR2614891A1 (fr) 1988-11-10
DE3815213A1 (de) 1988-11-17
CH676598A5 (enrdf_load_stackoverflow) 1991-02-15
IT1219567B (it) 1990-05-18
IT8847912A0 (it) 1988-05-03
GB8810463D0 (en) 1988-06-08
NL8801174A (nl) 1988-12-01

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