JPS62252790A - ピリドベンゾオキサジン誘導体 - Google Patents

ピリドベンゾオキサジン誘導体

Info

Publication number
JPS62252790A
JPS62252790A JP61144640A JP14464086A JPS62252790A JP S62252790 A JPS62252790 A JP S62252790A JP 61144640 A JP61144640 A JP 61144640A JP 14464086 A JP14464086 A JP 14464086A JP S62252790 A JPS62252790 A JP S62252790A
Authority
JP
Japan
Prior art keywords
formula
compound
methyl
lower alkyl
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP61144640A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0327534B2 (en, 2012
Inventor
Isao Hayakawa
勇夫 早川
Seigo Shinko
新子　省悟
Shuichi Yokohama
横浜　秀一
Masazumi Imamura
今村　正純
Katsuichi Sakano
坂野　勝一
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Daiichi Pharmaceutical Co Ltd
Original Assignee
Daiichi Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=15134834&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JPS62252790(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Daiichi Pharmaceutical Co Ltd filed Critical Daiichi Pharmaceutical Co Ltd
Publication of JPS62252790A publication Critical patent/JPS62252790A/ja
Publication of JPH0327534B2 publication Critical patent/JPH0327534B2/ja
Priority to MX9203658A priority Critical patent/MX9203658A/es
Granted legal-status Critical Current

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
JP61144640A 1985-06-20 1986-06-20 ピリドベンゾオキサジン誘導体 Granted JPS62252790A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
MX9203658A MX9203658A (es) 1985-06-20 1992-06-26 Derivados de piridobenzoxazina opticamente activos, y su uso antimicrobiano.

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP60-134712 1985-06-20
JP13471285 1985-06-20
JP61-16496 1986-01-28

Related Child Applications (2)

Application Number Title Priority Date Filing Date
JP11455888A Division JPH0714945B2 (ja) 1988-05-13 1988-05-13 ピリドベンゾオキサジン類
JP7814191A Division JPH0747592B2 (ja) 1985-06-20 1991-01-18 ピリドベンゾオキサジン誘導体

Publications (2)

Publication Number Publication Date
JPS62252790A true JPS62252790A (ja) 1987-11-04
JPH0327534B2 JPH0327534B2 (en, 2012) 1991-04-16

Family

ID=15134834

Family Applications (1)

Application Number Title Priority Date Filing Date
JP61144640A Granted JPS62252790A (ja) 1985-06-20 1986-06-20 ピリドベンゾオキサジン誘導体

Country Status (3)

Country Link
JP (1) JPS62252790A (en, 2012)
PH (1) PH24486A (en, 2012)
ZA (1) ZA864518B (en, 2012)

Cited By (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6287577A (ja) * 1985-10-11 1987-04-22 Dai Ichi Seiyaku Co Ltd 光学活性３−メチルベンゾオキサジン誘導体およびその製法
JPS62145088A (ja) * 1985-12-10 1987-06-29 バイエル・アクチエンゲゼルシヤフト 鏡像異性体的に純粋な１，８−橋かけされた４−キノロン−３−カルボン酸
JPH01175975A (ja) * 1987-12-29 1989-07-12 Dai Ichi Seiyaku Co Ltd （ｓ）−ベンゾオキサジン誘導体の製法
JPH01228974A (ja) * 1988-03-09 1989-09-12 Dai Ichi Seiyaku Co Ltd ベンゾオキサジニルメチレンマロネート
US5185337A (en) * 1989-03-29 1993-02-09 Otsuka Pharmaceutical Co., Ltd. Pyrroloquinoline derivatives and pharmaceutical compositions for antimicrobial use
US5545737A (en) * 1990-03-01 1996-08-13 Daiichi Pharmaceutical Co., Ltd. Process for selectively producing an (S)-9-fluoro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-2,3-dihydro-7h-pyrido (1,2,3, -de) (1,4) benzoxazine-6-carboxylic acid hemihydrate or monohydrate
EP1211254A4 (en) * 1999-09-08 2006-05-03 Daiichi Seiyaku Co PROCESS FOR THE PREPARATION OF BENZOXAZINE DERIVATIVES AND THEIR INTERMEDIATES
EP2275141A1 (en) 1999-03-17 2011-01-19 Daiichi Pharmaceutical Co., Ltd. Tastemasked pharmaceutical compositions
US7964723B2 (en) 2008-08-02 2011-06-21 Apeloa-Kangyu And practical process for exclusively producing (S)-9-fluoro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-2,3-dihydro-7H-pyrido-[1,2,3,de][1,4]benzoxazine-6-carboxylic acid hemihydrate

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN115381840A (zh) 2014-11-07 2022-11-25 参天制药株式会社 眼科用水性组合物

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5746986A (en) * 1980-09-02 1982-03-17 Dai Ichi Seiyaku Co Ltd Pyrido(1,2,3-de)(1,4)benzoxazine derivative
JPS6078986A (ja) * 1983-10-07 1985-05-04 Dai Ichi Seiyaku Co Ltd オキサジン誘導体の製法

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5746986A (en) * 1980-09-02 1982-03-17 Dai Ichi Seiyaku Co Ltd Pyrido(1,2,3-de)(1,4)benzoxazine derivative
JPS6078986A (ja) * 1983-10-07 1985-05-04 Dai Ichi Seiyaku Co Ltd オキサジン誘導体の製法

Cited By (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6287577A (ja) * 1985-10-11 1987-04-22 Dai Ichi Seiyaku Co Ltd 光学活性３−メチルベンゾオキサジン誘導体およびその製法
JPS62145088A (ja) * 1985-12-10 1987-06-29 バイエル・アクチエンゲゼルシヤフト 鏡像異性体的に純粋な１，８−橋かけされた４−キノロン−３−カルボン酸
JPH01175975A (ja) * 1987-12-29 1989-07-12 Dai Ichi Seiyaku Co Ltd （ｓ）−ベンゾオキサジン誘導体の製法
JPH01228974A (ja) * 1988-03-09 1989-09-12 Dai Ichi Seiyaku Co Ltd ベンゾオキサジニルメチレンマロネート
US5185337A (en) * 1989-03-29 1993-02-09 Otsuka Pharmaceutical Co., Ltd. Pyrroloquinoline derivatives and pharmaceutical compositions for antimicrobial use
US5545737A (en) * 1990-03-01 1996-08-13 Daiichi Pharmaceutical Co., Ltd. Process for selectively producing an (S)-9-fluoro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-2,3-dihydro-7h-pyrido (1,2,3, -de) (1,4) benzoxazine-6-carboxylic acid hemihydrate or monohydrate
EP2275141A1 (en) 1999-03-17 2011-01-19 Daiichi Pharmaceutical Co., Ltd. Tastemasked pharmaceutical compositions
JP2009221209A (ja) * 1999-09-08 2009-10-01 Daiichi Sankyo Co Ltd ベンゾオキサジン誘導体の製造法およびその製造中間体
US7189847B2 (en) 1999-09-08 2007-03-13 Daiichi Pharmaceutical Co., Ltd. Process for producing benzoxazine derivative and production intermediate thereof
JP2009235077A (ja) * 1999-09-08 2009-10-15 Daiichi Sankyo Co Ltd ベンゾオキサジン誘導体の製造法およびその製造中間体
EP2218722A2 (en) 1999-09-08 2010-08-18 Daiichi Sankyo Company, Limited Process for producing benzoxazine derivative and production intermediate thereof
EP1211254A4 (en) * 1999-09-08 2006-05-03 Daiichi Seiyaku Co PROCESS FOR THE PREPARATION OF BENZOXAZINE DERIVATIVES AND THEIR INTERMEDIATES
EP2284174A1 (en) 1999-09-08 2011-02-16 Daiichi Sankyo Company, Limited Intermediates for the preparation of benzoxazine derivatives and process for their preparation
EP2218722A3 (en) * 1999-09-08 2011-05-11 Daiichi Sankyo Company, Limited Process for producing benzoxazine derivative and production intermediate thereof
EP2360160A1 (en) 1999-09-08 2011-08-24 Daiichi Sankyo Company, Limited Intermediates and their use for producing benzoxazine derivative
US7964723B2 (en) 2008-08-02 2011-06-21 Apeloa-Kangyu And practical process for exclusively producing (S)-9-fluoro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-2,3-dihydro-7H-pyrido-[1,2,3,de][1,4]benzoxazine-6-carboxylic acid hemihydrate

Also Published As

Publication number Publication date
JPH0327534B2 (en, 2012) 1991-04-16
PH24486A (en) 1990-07-18
ZA864518B (en) 1987-03-25

Similar Documents

Publication Publication Date Title
KR940003757B1 (ko) 광학 활성 피리도벤즈옥사진 유도체의 제조방법
JPH0737460B2 (ja) ピラノインドリジン誘導体及びその製造法
JPS62252790A (ja) ピリドベンゾオキサジン誘導体
KR0125115B1 (ko) (-)피페라진 벤즈옥사진 유도체의 제조방법
SU936815A3 (ru) Способ получени 4,1-бензоксазепинов или их тиааналогов
JPH0256358B2 (en, 2012)
Chupp et al. Heterocycles from substituted amides. VI. A new carbostyril synthesis from alpha‐substituted acetamides and the vilsmeier reagent
KR900004145B1 (ko) 트리사이클릭 화합물의 제조방법
KR950012563B1 (ko) 광학 활성 2,3-디하이드로벤즈옥사진 유도체 및 이의 제조방법
JPH04364185A (ja) ピリドベンゾオキサジン誘導体
JPH0714945B2 (ja) ピリドベンゾオキサジン類
EP0267432A1 (en) Antibacterially active pyrido-benzothiazine derivatives with long term action
KR100248370B1 (ko) (-)-3(s)-메틸피리도 벤즈옥사진 중간 유도체의 제조방법
JPS6335579A (ja) 含硫ベンゾキサジノリフアマイシン誘導体
JP2651658B2 (ja) １，２，３，５−テトラヒドロインドリジン誘導体
JPS58192874A (ja) 新規スピロイソキサゾリン誘導体
DK175312B1 (da) Optisk aktive benzoxazinderivater
JPS61293979A (ja) ３−置換−２−ホルミルチオフエン化合物の製造方法
JPS61236779A (ja) ３環式化合物
JPH04270291A (ja) チアジノ〔６，５−ｂ〕インドリジン誘導体
JPH02138281A (ja) ３‐置換ピリドベンゾオキサジン
JPH02152947A (ja) ジフルオロフェノキシ化合物
JPS6256154B2 (en, 2012)
IE64929B1 (en) Optically active pyridobenzoxazine derivatives and intermediates thereof
JPH0395185A (ja) ペネム―３―カルボン酸エステル誘導体

Legal Events

Date Code Title Description
R153 Grant of patent term extension

Free format text: JAPANESE INTERMEDIATE CODE: R153

R153 Grant of patent term extension

Free format text: JAPANESE INTERMEDIATE CODE: R153

R153 Grant of patent term extension

Free format text: JAPANESE INTERMEDIATE CODE: R153

R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

R153 Grant of patent term extension

Free format text: JAPANESE INTERMEDIATE CODE: R153

FPAY Renewal fee payment (event date is renewal date of database)

Free format text: PAYMENT UNTIL: 20120416

Year of fee payment: 21

S111 Request for change of ownership or part of ownership

Free format text: JAPANESE INTERMEDIATE CODE: R313111

FPAY Renewal fee payment (event date is renewal date of database)

Free format text: PAYMENT UNTIL: 20120416

Year of fee payment: 21

R350 Written notification of registration of transfer

Free format text: JAPANESE INTERMEDIATE CODE: R350

FPAY Renewal fee payment (event date is renewal date of database)

Free format text: PAYMENT UNTIL: 20120416

Year of fee payment: 21

FPAY Renewal fee payment (event date is renewal date of database)

Free format text: PAYMENT UNTIL: 20120416

Year of fee payment: 21

EXPY Cancellation because of completion of term
FPAY Renewal fee payment (event date is renewal date of database)

Free format text: PAYMENT UNTIL: 20120416

Year of fee payment: 21