JPS6124580A - アミノチアゾリルグルタル酸誘導体の製造方法 - Google Patents

アミノチアゾリルグルタル酸誘導体の製造方法

Info

Publication number
JPS6124580A
JPS6124580A JP14579484A JP14579484A JPS6124580A JP S6124580 A JPS6124580 A JP S6124580A JP 14579484 A JP14579484 A JP 14579484A JP 14579484 A JP14579484 A JP 14579484A JP S6124580 A JPS6124580 A JP S6124580A
Authority
JP
Japan
Prior art keywords
amino
thiazolyl
ester
formula
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP14579484A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0587512B2 (https=
Inventor
Hiroshi Matsumura
宏 松村
Toshisada Yano
利定 矢野
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Shionogi and Co Ltd
Original Assignee
Shionogi and Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi and Co Ltd filed Critical Shionogi and Co Ltd
Priority to JP14579484A priority Critical patent/JPS6124580A/ja
Priority to US06/746,564 priority patent/US4652652A/en
Priority to GB08515640A priority patent/GB2162514B/en
Priority to KR1019850004645A priority patent/KR920003197B1/ko
Priority to EP85108491A priority patent/EP0168025B1/en
Priority to DE8585108491T priority patent/DE3573252D1/de
Priority to ES545068A priority patent/ES8603849A1/es
Publication of JPS6124580A publication Critical patent/JPS6124580A/ja
Publication of JPH0587512B2 publication Critical patent/JPH0587512B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/40—Unsubstituted amino or imino radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP14579484A 1984-07-12 1984-07-12 アミノチアゾリルグルタル酸誘導体の製造方法 Granted JPS6124580A (ja)

Priority Applications (7)

Application Number Priority Date Filing Date Title
JP14579484A JPS6124580A (ja) 1984-07-12 1984-07-12 アミノチアゾリルグルタル酸誘導体の製造方法
US06/746,564 US4652652A (en) 1984-07-12 1985-06-19 Thiazolylpropenedicarboxylic acid half esters and process for making
GB08515640A GB2162514B (en) 1984-07-12 1985-06-20 Thiazolylpropenedicarboxylic acid half esters
KR1019850004645A KR920003197B1 (ko) 1984-07-12 1985-06-28 티아졸릴프로펜디카르복실산 반 에스테르류의 제조방법
EP85108491A EP0168025B1 (en) 1984-07-12 1985-07-09 Process for producing aminothiazolylpropendicarboxylic acid monoesters
DE8585108491T DE3573252D1 (en) 1984-07-12 1985-07-09 Process for producing aminothiazolylpropendicarboxylic acid monoesters
ES545068A ES8603849A1 (es) 1984-07-12 1985-07-11 Procedimiento para la fabricacion de derivados del acido aminotiazolilpropandicarboxilico

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP14579484A JPS6124580A (ja) 1984-07-12 1984-07-12 アミノチアゾリルグルタル酸誘導体の製造方法

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP5055092A Division JPH0647581B2 (ja) 1993-02-18 1993-02-18 アミノチアゾリルグルタル酸誘導体

Publications (2)

Publication Number Publication Date
JPS6124580A true JPS6124580A (ja) 1986-02-03
JPH0587512B2 JPH0587512B2 (https=) 1993-12-16

Family

ID=15393306

Family Applications (1)

Application Number Title Priority Date Filing Date
JP14579484A Granted JPS6124580A (ja) 1984-07-12 1984-07-12 アミノチアゾリルグルタル酸誘導体の製造方法

Country Status (7)

Country Link
US (1) US4652652A (https=)
EP (1) EP0168025B1 (https=)
JP (1) JPS6124580A (https=)
KR (1) KR920003197B1 (https=)
DE (1) DE3573252D1 (https=)
ES (1) ES8603849A1 (https=)
GB (1) GB2162514B (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6153272A (ja) * 1984-08-24 1986-03-17 Shionogi & Co Ltd グルタル酸誘導体の製法
DE3807232A1 (de) * 1988-03-05 1989-09-14 Bayer Ag Substituierte acrylsaeureester
GB0922204D0 (en) * 2009-12-18 2010-02-03 Givaudan Sa Organic Compounds
CN111116508A (zh) * 2019-12-31 2020-05-08 烟台坤益液晶显示材料有限公司 一种头孢布烯7β位侧链中间体合成方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4298375A (en) * 1979-10-01 1981-11-03 Monsanto Company 2-Substituted-5-phenyl-4-thiazolecarboxylic acids and their derivatives as safening agents
DE3145727A1 (de) * 1981-11-19 1983-05-26 Bayer Ag, 5090 Leverkusen Zwischenprodukte, verfahren zu deren herstellung und verfahren zur herstellung von cephalosporinen
US4426528A (en) * 1982-04-01 1984-01-17 Eli Lilly And Company Purification of syn-(2-aminothiazol-4-yl)methoxyimino)acetic acid
AU575854B2 (en) * 1983-10-04 1988-08-11 Shionogi & Co., Ltd. 7beta-(carboxyalkenamido) cephalosporins
JPS6153272A (ja) * 1984-08-24 1986-03-17 Shionogi & Co Ltd グルタル酸誘導体の製法

Also Published As

Publication number Publication date
ES545068A0 (es) 1986-01-01
ES8603849A1 (es) 1986-01-01
US4652652A (en) 1987-03-24
KR920003197B1 (ko) 1992-04-24
EP0168025B1 (en) 1989-09-27
GB2162514B (en) 1988-04-20
GB2162514A (en) 1986-02-05
DE3573252D1 (en) 1989-11-02
KR860001085A (ko) 1986-02-22
EP0168025A1 (en) 1986-01-15
JPH0587512B2 (https=) 1993-12-16
GB8515640D0 (en) 1985-07-24

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Legal Events

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