JPS60233076A - 新規なβ−ラクタム化合物およびその製造法 - Google Patents
新規なβ−ラクタム化合物およびその製造法Info
- Publication number
- JPS60233076A JPS60233076A JP59191167A JP19116784A JPS60233076A JP S60233076 A JPS60233076 A JP S60233076A JP 59191167 A JP59191167 A JP 59191167A JP 19116784 A JP19116784 A JP 19116784A JP S60233076 A JPS60233076 A JP S60233076A
- Authority
- JP
- Japan
- Prior art keywords
- group
- general formula
- lower alkyl
- hydrogen atom
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CA000453478A CA1283906C (en) | 1983-05-09 | 1984-05-03 | .beta.-LACTAM COMPOUNDS AND PRODUCTION THEREOF |
CA453478 | 1984-05-03 |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS60233076A true JPS60233076A (ja) | 1985-11-19 |
JPH0463878B2 JPH0463878B2 (enrdf_load_stackoverflow) | 1992-10-13 |
Family
ID=4127789
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP59191167A Granted JPS60233076A (ja) | 1984-05-03 | 1984-09-12 | 新規なβ−ラクタム化合物およびその製造法 |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS60233076A (enrdf_load_stackoverflow) |
Cited By (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS6363680A (ja) * | 1986-09-05 | 1988-03-22 | Nippon Redarii Kk | (1r)−1−メチルカルバペネム−3−カルボン酸誘導体 |
JPH01104076A (ja) * | 1986-03-27 | 1989-04-21 | Sumitomo Pharmaceut Co Ltd | 新規なβ−ラクタム化合物 |
WO1993000344A1 (fr) * | 1991-06-20 | 1993-01-07 | Daiichi Pharmaceutical Co., Ltd. | Derive de carbapenem |
JPH05339269A (ja) * | 1991-06-04 | 1993-12-21 | Sankyo Co Ltd | 1−メチルカルバペネム誘導体 |
US5317016A (en) * | 1991-08-20 | 1994-05-31 | Shionogi Seiyaku Kabushiki Kaisha | Pyrrolidylthiocarbapenem derivative |
JPH06345766A (ja) * | 1993-06-15 | 1994-12-20 | Dong Kook Pharmaceut Co Ltd | 1−β−メチル−2−チオール系カルバペネム誘導体およびその製造方法 |
US5441949A (en) * | 1992-07-21 | 1995-08-15 | Zeneca Limited | Carbapenem antibiotic compounds |
US5444057A (en) * | 1992-07-21 | 1995-08-22 | Zeneca Limited | Carbapenem-antibiotic compounds |
US5478820A (en) * | 1992-02-04 | 1995-12-26 | Zeneca Ltd. | Antibiotic compounds |
US5519015A (en) * | 1992-03-26 | 1996-05-21 | Zeneca Limited | Carbapenem antibiotic compounds |
US5527791A (en) * | 1992-09-28 | 1996-06-18 | Zeneca Limited | Carbapenem antibiotic compounds |
US5527793A (en) * | 1992-07-21 | 1996-06-18 | Zeneca Limited | Antibiotic carbapenem compounds |
US5541178A (en) * | 1991-04-08 | 1996-07-30 | Zeneca Limited | Carbapenem antibiotic compounds |
WO1999057121A1 (fr) * | 1998-05-01 | 1999-11-11 | Kyoto Pharmaceutical Industries, Ltd. | Derives de carbapenem, son utilisation et composes intermediaires a base de carbapenem |
US6232338B1 (en) | 1995-08-04 | 2001-05-15 | Zeneca Limited | 4-Mercaptopyrrolidine derivatives as farnesyl transferase inhibitors |
US6777438B2 (en) | 1999-12-22 | 2004-08-17 | Astrazeneca Ab | Inhibitors of farnesyl protein transferase |
US6946468B1 (en) | 1996-08-17 | 2005-09-20 | Zeneca Limited | 3-mercaptopyrrolidines as farnesyl protein transferase inhibitors |
JP2006001841A (ja) * | 2004-06-15 | 2006-01-05 | Sumitomo Chemical Co Ltd | 含窒素へテロ環化合物の製造方法 |
US7101897B2 (en) | 1999-12-22 | 2006-09-05 | Astrazeneca Ab | Farnesyl transferase inhibitors |
JP2007532693A (ja) * | 2004-08-31 | 2007-11-15 | コリア リサーチ インスティチュート オブ ケミカル テクノロジー | 2−アリールメチルアゼチジン・カルバペネム誘導体及びその製造方法 |
JP2008501657A (ja) * | 2004-06-02 | 2008-01-24 | サンド・アクチエンゲゼルシヤフト | 結晶形態のメロペネム中間体 |
JP2019512547A (ja) * | 2016-03-16 | 2019-05-16 | オーキッド ファーマ リミテッド | カルバペネム化合物 |
CN111960984A (zh) * | 2020-09-11 | 2020-11-20 | 江西如益科技发展有限公司 | 一种合成多尼培南侧链中间体的制备方法 |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5287387U (enrdf_load_stackoverflow) * | 1975-12-23 | 1977-06-29 | ||
JPS6019787A (ja) * | 1983-07-12 | 1985-01-31 | Sumitomo Chem Co Ltd | 新規なβ−ラクタム化合物及びその製造法 |
-
1984
- 1984-09-12 JP JP59191167A patent/JPS60233076A/ja active Granted
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5287387U (enrdf_load_stackoverflow) * | 1975-12-23 | 1977-06-29 | ||
JPS6019787A (ja) * | 1983-07-12 | 1985-01-31 | Sumitomo Chem Co Ltd | 新規なβ−ラクタム化合物及びその製造法 |
Cited By (33)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH01104076A (ja) * | 1986-03-27 | 1989-04-21 | Sumitomo Pharmaceut Co Ltd | 新規なβ−ラクタム化合物 |
JPS6363680A (ja) * | 1986-09-05 | 1988-03-22 | Nippon Redarii Kk | (1r)−1−メチルカルバペネム−3−カルボン酸誘導体 |
US5541178A (en) * | 1991-04-08 | 1996-07-30 | Zeneca Limited | Carbapenem antibiotic compounds |
JPH05339269A (ja) * | 1991-06-04 | 1993-12-21 | Sankyo Co Ltd | 1−メチルカルバペネム誘導体 |
WO1993000344A1 (fr) * | 1991-06-20 | 1993-01-07 | Daiichi Pharmaceutical Co., Ltd. | Derive de carbapenem |
US5317016A (en) * | 1991-08-20 | 1994-05-31 | Shionogi Seiyaku Kabushiki Kaisha | Pyrrolidylthiocarbapenem derivative |
US5703243A (en) * | 1991-08-20 | 1997-12-30 | Shionogi Seiyaku Kabushiki Kaisha | Intermediates for pyrrolidylthiocarbapenem derivative |
US5478820A (en) * | 1992-02-04 | 1995-12-26 | Zeneca Ltd. | Antibiotic compounds |
US7041836B2 (en) | 1992-02-04 | 2006-05-09 | Astrazeneca Uk Limited | Antibiotic compounds |
US6521612B2 (en) | 1992-02-04 | 2003-02-18 | Zeneca Ltd. | Antibiotic compounds |
US5652233A (en) * | 1992-02-04 | 1997-07-29 | Zeneca Limited | Antibiotic compounds |
US5856321A (en) * | 1992-02-04 | 1999-01-05 | Zeneca Limited | Antibiotic compounds |
US7342005B2 (en) | 1992-02-04 | 2008-03-11 | Astrazeneca Uk Limited | Antibiotic compounds |
US6187804B1 (en) | 1992-02-04 | 2001-02-13 | Zeneca Limited | Antibiotic compounds |
US5519015A (en) * | 1992-03-26 | 1996-05-21 | Zeneca Limited | Carbapenem antibiotic compounds |
US5441949A (en) * | 1992-07-21 | 1995-08-15 | Zeneca Limited | Carbapenem antibiotic compounds |
US5444057A (en) * | 1992-07-21 | 1995-08-22 | Zeneca Limited | Carbapenem-antibiotic compounds |
US5527793A (en) * | 1992-07-21 | 1996-06-18 | Zeneca Limited | Antibiotic carbapenem compounds |
US5527791A (en) * | 1992-09-28 | 1996-06-18 | Zeneca Limited | Carbapenem antibiotic compounds |
JPH06345766A (ja) * | 1993-06-15 | 1994-12-20 | Dong Kook Pharmaceut Co Ltd | 1−β−メチル−2−チオール系カルバペネム誘導体およびその製造方法 |
US6232338B1 (en) | 1995-08-04 | 2001-05-15 | Zeneca Limited | 4-Mercaptopyrrolidine derivatives as farnesyl transferase inhibitors |
US6946468B1 (en) | 1996-08-17 | 2005-09-20 | Zeneca Limited | 3-mercaptopyrrolidines as farnesyl protein transferase inhibitors |
WO1999057121A1 (fr) * | 1998-05-01 | 1999-11-11 | Kyoto Pharmaceutical Industries, Ltd. | Derives de carbapenem, son utilisation et composes intermediaires a base de carbapenem |
EP1078927A4 (en) * | 1998-05-01 | 2003-01-08 | Kyoto Pharma Ind | CABAPEN DERIVATIVES, YOUR APPLICATION AND YOUR INTERMEDIATE PRODUCTS |
US6410525B1 (en) | 1998-05-01 | 2002-06-25 | Kyoto Pharmaceutical Industries, Ltd. | Carbapenem derivatives, utilization thereof and intermediate compounds of the same |
US6777438B2 (en) | 1999-12-22 | 2004-08-17 | Astrazeneca Ab | Inhibitors of farnesyl protein transferase |
US7101897B2 (en) | 1999-12-22 | 2006-09-05 | Astrazeneca Ab | Farnesyl transferase inhibitors |
JP2008501657A (ja) * | 2004-06-02 | 2008-01-24 | サンド・アクチエンゲゼルシヤフト | 結晶形態のメロペネム中間体 |
JP2006001841A (ja) * | 2004-06-15 | 2006-01-05 | Sumitomo Chemical Co Ltd | 含窒素へテロ環化合物の製造方法 |
JP2007532693A (ja) * | 2004-08-31 | 2007-11-15 | コリア リサーチ インスティチュート オブ ケミカル テクノロジー | 2−アリールメチルアゼチジン・カルバペネム誘導体及びその製造方法 |
JP2019512547A (ja) * | 2016-03-16 | 2019-05-16 | オーキッド ファーマ リミテッド | カルバペネム化合物 |
CN111960984A (zh) * | 2020-09-11 | 2020-11-20 | 江西如益科技发展有限公司 | 一种合成多尼培南侧链中间体的制备方法 |
CN111960984B (zh) * | 2020-09-11 | 2023-04-28 | 江西如益科技发展有限公司 | 一种合成多尼培南侧链中间体的制备方法 |
Also Published As
Publication number | Publication date |
---|---|
JPH0463878B2 (enrdf_load_stackoverflow) | 1992-10-13 |
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