JPS58154584A - ５位ヒドロキシ置換カンプトテシン誘導体の製造法 - Google Patents

５位ヒドロキシ置換カンプトテシン誘導体の製造法

Info

Publication number
JPS58154584A
JPS58154584A JP3634682A JP3634682A JPS58154584A JP S58154584 A JPS58154584 A JP S58154584A JP 3634682 A JP3634682 A JP 3634682A JP 3634682 A JP3634682 A JP 3634682A JP S58154584 A JPS58154584 A JP S58154584A
Authority
JP
Japan
Prior art keywords
group
camptothecin
substituted
substituent
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP3634682A
Other languages
English (en)
Japanese (ja)
Other versions
JPS6247873B2 (enExample
Inventor
Sada Miyasaka
宮坂　貞
Seigo Sawada
誠吾 沢田
Kenichiro Nogata
野方　健一郎
Masahiko Mutai
務台　方彦
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Yakult Honsha Co Ltd
Original Assignee
Yakult Honsha Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yakult Honsha Co Ltd filed Critical Yakult Honsha Co Ltd
Priority to JP3634682A priority Critical patent/JPS58154584A/ja
Publication of JPS58154584A publication Critical patent/JPS58154584A/ja
Publication of JPS6247873B2 publication Critical patent/JPS6247873B2/ja
Granted legal-status Critical Current

Links

Landscapes

  • Nitrogen Condensed Heterocyclic Rings (AREA)
JP3634682A 1982-03-10 1982-03-10 ５位ヒドロキシ置換カンプトテシン誘導体の製造法 Granted JPS58154584A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP3634682A JPS58154584A (ja) 1982-03-10 1982-03-10 ５位ヒドロキシ置換カンプトテシン誘導体の製造法

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP3634682A JPS58154584A (ja) 1982-03-10 1982-03-10 ５位ヒドロキシ置換カンプトテシン誘導体の製造法

Publications (2)

Publication Number Publication Date
JPS58154584A true JPS58154584A (ja) 1983-09-14
JPS6247873B2 JPS6247873B2 (enExample) 1987-10-09

Family

ID=12467268

Family Applications (1)

Application Number Title Priority Date Filing Date
JP3634682A Granted JPS58154584A (ja) 1982-03-10 1982-03-10 ５位ヒドロキシ置換カンプトテシン誘導体の製造法

Country Status (1)

Country Link
JP (1) JPS58154584A (enExample)

Cited By (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4604463A (en) * 1983-07-14 1986-08-05 Kabushiki Kaisha Yakult Honsha Camptothecin derivatives and process for preparing same
JPH01186892A (ja) * 1988-01-20 1989-07-26 Yakult Honsha Co Ltd 新規なカンプトテシン誘導体
JPH01186893A (ja) * 1987-12-01 1989-07-26 Smithkline Beckman Corp 水溶性カンプトテシン類似体
US5447936A (en) * 1993-12-22 1995-09-05 Bionumerik Pharmaceuticals, Inc. Lactone stable formulation of 10-hydroxy 7-ethyl camptothecin and methods for uses thereof
US5468754A (en) * 1994-04-19 1995-11-21 Bionumerik Pharmaceuticals, Inc. 11,7 substituted camptothecin derivatives and formulations of 11,7 substituted camptothecin derivatives and methods for uses thereof
WO1997046563A1 (en) * 1996-06-05 1997-12-11 Dr. Reddy's Research Foundation Novel water-soluble c-ring analogues of 20 (s)-camptothecin
US5972955A (en) * 1995-06-06 1999-10-26 Dr. Reddy's Research Foundation Water soluble C-ring analogues of 20(S)-camptothecin
US6177439B1 (en) 1995-06-06 2001-01-23 Reddy's Research Foundation Water soluble analogues of 20(S)-camptothecin
US6214836B1 (en) 1995-06-06 2001-04-10 Dr. Reddy's Research Foundation Water soluble analogues of 20(S)-camptothecin
EP1138682A1 (en) * 1996-12-19 2001-10-04 Dr. Reddy's Research Foundation Novel water soluble c-ring analogues of 20 (s)-camptothecin

Cited By (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4604463A (en) * 1983-07-14 1986-08-05 Kabushiki Kaisha Yakult Honsha Camptothecin derivatives and process for preparing same
JPH01186893A (ja) * 1987-12-01 1989-07-26 Smithkline Beckman Corp 水溶性カンプトテシン類似体
JPH01186892A (ja) * 1988-01-20 1989-07-26 Yakult Honsha Co Ltd 新規なカンプトテシン誘導体
US5447936A (en) * 1993-12-22 1995-09-05 Bionumerik Pharmaceuticals, Inc. Lactone stable formulation of 10-hydroxy 7-ethyl camptothecin and methods for uses thereof
US5468754A (en) * 1994-04-19 1995-11-21 Bionumerik Pharmaceuticals, Inc. 11,7 substituted camptothecin derivatives and formulations of 11,7 substituted camptothecin derivatives and methods for uses thereof
US5633260A (en) * 1994-04-19 1997-05-27 Bionumerik Pharmaceuticals, Inc. 11,7 Substituted camptothecin derivatives and formulations of 11,7 substituted camptothecin derivatives and methods for uses thereof
US5972955A (en) * 1995-06-06 1999-10-26 Dr. Reddy's Research Foundation Water soluble C-ring analogues of 20(S)-camptothecin
US6177439B1 (en) 1995-06-06 2001-01-23 Reddy's Research Foundation Water soluble analogues of 20(S)-camptothecin
US6214836B1 (en) 1995-06-06 2001-04-10 Dr. Reddy's Research Foundation Water soluble analogues of 20(S)-camptothecin
WO1997046563A1 (en) * 1996-06-05 1997-12-11 Dr. Reddy's Research Foundation Novel water-soluble c-ring analogues of 20 (s)-camptothecin
EP1138682A1 (en) * 1996-12-19 2001-10-04 Dr. Reddy's Research Foundation Novel water soluble c-ring analogues of 20 (s)-camptothecin

Also Published As

Publication number Publication date
JPS6247873B2 (enExample) 1987-10-09

Similar Documents

Publication Publication Date Title
JPH0329791B2 (enExample)
JP3523267B2 (ja) ベンゾイミダゾール化合物の合成法
JPS6247195B2 (enExample)
JPS58154584A (ja) ５位ヒドロキシ置換カンプトテシン誘導体の製造法
JPS59122470A (ja) キノリン−３−カルボン酸誘導体の製造法
SU1321376A3 (ru) Способ получени производных хинолинкарбоновой кислоты
JPS5839683A (ja) 新規なカンプトテシン誘導体
JPH029032B2 (enExample)
RU2145325C1 (ru) Способы получения 9-аминокамптотецина, промежуточные продукты и способ их получения
JPS636072B2 (enExample)
CN116969881A (zh) 一种吡仑帕奈的合成方法
JPS6045196B2 (ja) １−（２−テトラヒドロフリル）ウラシル類の製造方法
JP2726653B2 (ja) ジアミノピリミジン誘導体
JPS63162689A (ja) ７―ブロモ―β―カルボリン誘導体の製造方法
JP3814742B2 (ja) ４−フルオロサリチル酸類
JPH03176473A (ja) ピリジン―ｎ―オキシド誘導体及びその製法
JP3037816B2 (ja) ピラノインドリジンジオン誘導体の製法
JP2803140B2 (ja) ベンゾキノンジカルボキシミド誘導体、その中間体、この中間体の製造方法、この誘導体を用いた酸化剤
JP3328694B2 (ja) 含窒素複素環化合物の製造方法
JPH0429674B2 (enExample)
JPH0532629A (ja) 高純度メチルチオカーバメイト類の製造方法
CN120112512A (zh) 制备(z)-3-(2-(5-溴-1h-吲哚-3-基)-2-氰基乙烯基)-4-甲氧基苯甲腈的方法
JP3023773B2 (ja) 含窒素複素環化合物
JPH0144718B2 (enExample)
JPH02111761A (ja) ウラシルの製造法