JPS57203085A - 1,8-cyclic substituted quinoline derivative - Google Patents
1,8-cyclic substituted quinoline derivativeInfo
- Publication number
- JPS57203085A JPS57203085A JP8845781A JP8845781A JPS57203085A JP S57203085 A JPS57203085 A JP S57203085A JP 8845781 A JP8845781 A JP 8845781A JP 8845781 A JP8845781 A JP 8845781A JP S57203085 A JPS57203085 A JP S57203085A
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formulai
- lower alkyl
- quinoline derivative
- substituted quinoline
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 125000002943 quinolinyl group Chemical class N1=C(C=CC2=CC=CC=C12)* 0.000 title 1
- IAZDPXIOMUYVGZ-UHFFFAOYSA-N Dimethylsulphoxide Chemical compound CS(C)=O IAZDPXIOMUYVGZ-UHFFFAOYSA-N 0.000 abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 230000000844 anti-bacterial effect Effects 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- -1 10-Fluoro-11-( 4-methyl-1-piperazinyl )-8-oxo-2, 3-dihydro-4H, 8H-pyrido [1,2,3-ef][1,5]benzoxazepin-7-carboxylic acid Chemical compound 0.000 abstract 1
- 241000894006 Bacteria Species 0.000 abstract 1
- 241000589517 Pseudomonas aeruginosa Species 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- 239000000463 material Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
- 238000001228 spectrum Methods 0.000 abstract 1
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP8845781A JPS57203085A (en) | 1981-06-09 | 1981-06-09 | 1,8-cyclic substituted quinoline derivative |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP8845781A JPS57203085A (en) | 1981-06-09 | 1981-06-09 | 1,8-cyclic substituted quinoline derivative |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS57203085A true JPS57203085A (en) | 1982-12-13 |
| JPH0215551B2 JPH0215551B2 (enrdf_load_stackoverflow) | 1990-04-12 |
Family
ID=13943316
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP8845781A Granted JPS57203085A (en) | 1981-06-09 | 1981-06-09 | 1,8-cyclic substituted quinoline derivative |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JPS57203085A (enrdf_load_stackoverflow) |
Cited By (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5976091A (ja) * | 1982-10-22 | 1984-04-28 | Otsuka Pharmaceut Co Ltd | ピリド〔１，２，３−ｄｅ〕〔１，４〕ベンゾチアジン誘導体 |
| JPS60208987A (ja) * | 1984-02-24 | 1985-10-21 | メデイオラヌム・フアルマセウテイシ・エス．ア−ル．エル． | ピリドベンゾチアジン誘導体の製造法 |
| US4571396A (en) * | 1984-04-16 | 1986-02-18 | Warner-Lambert Company | Antibacterial agents |
| JPS62145088A (ja) * | 1985-12-10 | 1987-06-29 | バイエル・アクチエンゲゼルシヤフト | 鏡像異性体的に純粋な１，８−橋かけされた４−キノロン−３−カルボン酸 |
| JPS6322590A (ja) * | 1986-07-01 | 1988-01-30 | メディオラヌム・ファルマセウティシ・エス．ア−ル．エル． | 高度溶解性、抗菌活性のピリド−ベンゾチアジン類の有機塩類及びその製法 |
| JPH01128988A (ja) * | 1987-10-06 | 1989-05-22 | Mediolanum Farmaceut Srl | 高抗菌活性及び組織に対する高生物学的利用能をもつピリドベンゾチアジン誘導体 |
| WO1991016894A1 (en) * | 1990-05-02 | 1991-11-14 | Abbott Laboratories | Quinolizinone type compounds |
| US5175160A (en) * | 1988-08-09 | 1992-12-29 | Daiichi Pharmaceutical Co., Ltd. | Antimicrobial agent for animals |
| CN111170941A (zh) * | 2018-11-12 | 2020-05-19 | 江西农业大学 | 1-环丙基-6,7-二氟-8-甲氧基氟喹诺酮-3-羧酸酯的制备方法 |
-
1981
- 1981-06-09 JP JP8845781A patent/JPS57203085A/ja active Granted
Cited By (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5976091A (ja) * | 1982-10-22 | 1984-04-28 | Otsuka Pharmaceut Co Ltd | ピリド〔１，２，３−ｄｅ〕〔１，４〕ベンゾチアジン誘導体 |
| AU573780B2 (en) * | 1984-02-24 | 1988-06-23 | Mediolanum Farmaceutici S.P.A. | Pyrido-benzothiazine derivatives |
| US4668784A (en) * | 1984-02-24 | 1987-05-26 | Mediolanum Farmaceutici S.R.L. | Derivatives of pyrido-benzothiazine with high anti-microbial activity |
| JPS60208987A (ja) * | 1984-02-24 | 1985-10-21 | メデイオラヌム・フアルマセウテイシ・エス．ア−ル．エル． | ピリドベンゾチアジン誘導体の製造法 |
| JPH0327389A (ja) * | 1984-02-24 | 1991-02-05 | Mediolanum Farmaceut Srl | 抗菌剤 |
| US4571396A (en) * | 1984-04-16 | 1986-02-18 | Warner-Lambert Company | Antibacterial agents |
| JPS62145088A (ja) * | 1985-12-10 | 1987-06-29 | バイエル・アクチエンゲゼルシヤフト | 鏡像異性体的に純粋な１，８−橋かけされた４−キノロン−３−カルボン酸 |
| JPS6322590A (ja) * | 1986-07-01 | 1988-01-30 | メディオラヌム・ファルマセウティシ・エス．ア−ル．エル． | 高度溶解性、抗菌活性のピリド−ベンゾチアジン類の有機塩類及びその製法 |
| US4923859A (en) * | 1987-10-06 | 1990-05-08 | Mediolanum Farmaceutici, S.R.L. | Pyrido-benzothiazine derivatives having high antibacterial activity and high bioavailability to tissues |
| JPH01128988A (ja) * | 1987-10-06 | 1989-05-22 | Mediolanum Farmaceut Srl | 高抗菌活性及び組織に対する高生物学的利用能をもつピリドベンゾチアジン誘導体 |
| US5066802A (en) * | 1987-10-06 | 1991-11-19 | Mediolanum Farmaceutici Srl. | Process for preparing pyrido-benzothiazine derivatives having high antibacterial activity and high bioavailability to tissues |
| US5175160A (en) * | 1988-08-09 | 1992-12-29 | Daiichi Pharmaceutical Co., Ltd. | Antimicrobial agent for animals |
| WO1991016894A1 (en) * | 1990-05-02 | 1991-11-14 | Abbott Laboratories | Quinolizinone type compounds |
| CN111170941A (zh) * | 2018-11-12 | 2020-05-19 | 江西农业大学 | 1-环丙基-6,7-二氟-8-甲氧基氟喹诺酮-3-羧酸酯的制备方法 |
| CN111170941B (zh) * | 2018-11-12 | 2023-07-25 | 江西农业大学 | 1-环丙基-6,7-二氟-8-甲氧基氟喹诺酮-3-羧酸酯的制备方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| JPH0215551B2 (enrdf_load_stackoverflow) | 1990-04-12 |
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