JPH07507811A - 鏡像異性のシス−3−(4,6−ジヒドロキシクロマン−3−イル−メチル)安息香酸 - Google Patents

鏡像異性のシス−3−(4,6−ジヒドロキシクロマン−3−イル−メチル)安息香酸

Info

Publication number
JPH07507811A
JPH07507811A JP6509963A JP50996393A JPH07507811A JP H07507811 A JPH07507811 A JP H07507811A JP 6509963 A JP6509963 A JP 6509963A JP 50996393 A JP50996393 A JP 50996393A JP H07507811 A JPH07507811 A JP H07507811A
Authority
JP
Japan
Prior art keywords
reducing agent
cis
salt
ylmethyl
dihydroxychroman
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP6509963A
Other languages
English (en)
Japanese (ja)
Inventor
マーチアショー,チャールズ ダブリュ.ザ・サード
ヴァンダープラス,ブライアン シー.
Original Assignee
ファイザー・インク.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ファイザー・インク. filed Critical ファイザー・インク.
Publication of JPH07507811A publication Critical patent/JPH07507811A/ja
Pending legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/22Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP6509963A 1992-10-21 1993-06-30 鏡像異性のシス−3−(4,6−ジヒドロキシクロマン−3−イル−メチル)安息香酸 Pending JPH07507811A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US96433692A 1992-10-21 1992-10-21
US964,336 1992-10-21
PCT/US1993/006061 WO1994008986A1 (en) 1992-10-21 1993-06-30 Enantiomeric cis-3-(4,6-dihydroxychroman-3-yl-methyl)benzoic acids

Publications (1)

Publication Number Publication Date
JPH07507811A true JPH07507811A (ja) 1995-08-31

Family

ID=25508434

Family Applications (1)

Application Number Title Priority Date Filing Date
JP6509963A Pending JPH07507811A (ja) 1992-10-21 1993-06-30 鏡像異性のシス−3−(4,6−ジヒドロキシクロマン−3−イル−メチル)安息香酸

Country Status (16)

Country Link
EP (1) EP0665839A1 (fi)
JP (1) JPH07507811A (fi)
KR (1) KR950704291A (fi)
CN (1) CN1090577A (fi)
AU (1) AU4650493A (fi)
CA (1) CA2146005A1 (fi)
CZ (1) CZ100895A3 (fi)
FI (1) FI934624A (fi)
HU (1) HUT65128A (fi)
IL (1) IL107293A0 (fi)
MX (1) MX9306526A (fi)
MY (1) MY131378A (fi)
NO (1) NO951507L (fi)
PL (1) PL308473A1 (fi)
WO (1) WO1994008986A1 (fi)
ZA (1) ZA937737B (fi)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU713701B2 (en) * 1996-09-16 1999-12-09 Pfizer Inc. Processes and intermediates for preparing substituted chromanol derivatives
MXPA02004225A (es) * 1999-10-27 2002-10-17 Nobex Corp Resolucion de intermediarios en la sintesis de bicalutamida sustancialmente pura.
TWI270545B (en) 2000-05-24 2007-01-11 Sugen Inc Mannich base prodrugs of 3-(pyrrol-2-ylmethylidene)-2-indolinone derivatives
US6479692B1 (en) 2001-05-02 2002-11-12 Nobex Corporation Methods of synthesizing acylanilides including bicalutamide and derivatives thereof
US8080675B2 (en) 2004-09-21 2011-12-20 Marshall Edwards, Inc. Chroman derivatives, medicaments and use in therapy
ATE532777T1 (de) 2004-09-21 2011-11-15 Marshall Edwards Inc Substituierte chromanderivate, medikamente und anwendungen in der therapie
CA2816322A1 (en) 2010-11-01 2012-05-10 Marshall Edwards, Inc. Isoflavonoid compositions and methods for the treatment of cancer
AU2016215515B2 (en) 2015-02-02 2020-04-30 Mei Pharma, Inc. Combination therapies

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5059609A (en) * 1987-10-19 1991-10-22 Pfizer Inc. Substituted tetralins, chromans and related compounds in the treatment of asthma, arthritis and related diseases

Also Published As

Publication number Publication date
FI934624A0 (fi) 1993-10-20
NO951507D0 (no) 1995-04-20
MX9306526A (es) 1994-04-29
PL308473A1 (en) 1995-08-07
EP0665839A1 (en) 1995-08-09
KR950704291A (ko) 1995-11-17
MY131378A (en) 2007-08-30
FI934624A (fi) 1994-04-22
CZ100895A3 (en) 1995-10-18
IL107293A0 (en) 1994-01-25
AU4650493A (en) 1994-05-09
HUT65128A (en) 1994-04-28
CN1090577A (zh) 1994-08-10
WO1994008986A1 (en) 1994-04-28
NO951507L (no) 1995-04-20
ZA937737B (en) 1995-04-19
HU9302973D0 (en) 1993-12-28
CA2146005A1 (en) 1994-04-28

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