JP7348904B2 - 新規な結晶形態 - Google Patents

新規な結晶形態 Download PDF

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Publication number
JP7348904B2
JP7348904B2 JP2020543281A JP2020543281A JP7348904B2 JP 7348904 B2 JP7348904 B2 JP 7348904B2 JP 2020543281 A JP2020543281 A JP 2020543281A JP 2020543281 A JP2020543281 A JP 2020543281A JP 7348904 B2 JP7348904 B2 JP 7348904B2
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plants
methyl
dichlorophenyl
species
trifluoromethyl
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Japanese (ja)
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JP2021514356A5 (https=
JPWO2019158476A5 (https=
JP2021514356A (ja
Inventor
ジョン ホーン
イアン ケヴィン ジョーンズ
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シンジェンタ パーティシペーションズ アーゲー
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C07D213/82—Amides; Imides in position 3
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P3/00—Fungicides
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P5/00—Nematocides
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P7/00—Arthropodicides
    • A01P7/04—Insecticides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Insects & Arthropods (AREA)
  • Mycology (AREA)
  • Microbiology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyridine Compounds (AREA)
  • Liquid Crystal Substances (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2020543281A 2018-02-13 2019-02-11 新規な結晶形態 Active JP7348904B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP18156463.4 2018-02-13
EP18156463 2018-02-13
PCT/EP2019/053292 WO2019158476A1 (en) 2018-02-13 2019-02-11 Novel crystalline forms

Publications (4)

Publication Number Publication Date
JP2021514356A JP2021514356A (ja) 2021-06-10
JP2021514356A5 JP2021514356A5 (https=) 2022-02-22
JPWO2019158476A5 JPWO2019158476A5 (https=) 2022-02-22
JP7348904B2 true JP7348904B2 (ja) 2023-09-21

Family

ID=61198760

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Application Number Title Priority Date Filing Date
JP2020543281A Active JP7348904B2 (ja) 2018-02-13 2019-02-11 新規な結晶形態

Country Status (24)

Country Link
US (1) US11053201B2 (https=)
EP (2) EP3752489A1 (https=)
JP (1) JP7348904B2 (https=)
KR (2) KR102812896B1 (https=)
CN (1) CN111741945B (https=)
AR (1) AR114251A1 (https=)
AU (1) AU2019220997B2 (https=)
CA (2) CA3286688A1 (https=)
CL (2) CL2020002056A1 (https=)
CO (1) CO2020009901A2 (https=)
EA (1) EA202091893A1 (https=)
EC (1) ECSP20048382A (https=)
IL (1) IL276644B2 (https=)
JO (2) JOP20200194A1 (https=)
MA (1) MA51819A (https=)
MX (1) MX2020008367A (https=)
MY (1) MY205650A (https=)
PE (2) PE20211478A1 (https=)
PH (1) PH12020551304A1 (https=)
TW (1) TWI815859B (https=)
UA (1) UA129535C2 (https=)
UY (1) UY38085A (https=)
WO (1) WO2019158476A1 (https=)
ZA (1) ZA202004700B (https=)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL3019476T3 (pl) * 2013-07-08 2018-05-30 Syngenta Participations Ag Związki karboksyamidowe o 4-członowym pierścieniu jako nematocydy
AU2018390864B9 (en) * 2017-12-20 2024-12-12 Syngenta Crop Protection Ag Methods of controlling or preventing infestation of vegetable, tomato and potato plants by phytopathogenic microorganisms
AU2019342401A1 (en) * 2018-09-19 2021-04-15 Syngenta Crop Protection Ag Methods of controlling or preventing infestation of cereal plants by the phytopathogenic microorganism fusarium pseudograminearum
JP7758669B2 (ja) * 2019-12-10 2025-10-22 シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト マクロホミナ（ｍａｃｒｏｐｈｏｍｉｎａ）属の種の植物病原性微生物による植物の被害を防除するか又は防止する方法
CN115397243B (zh) * 2020-01-30 2025-03-28 先正达农作物保护股份公司 控制或预防香蕉植物中的巴拿马病的方法
WO2022073797A1 (en) 2020-10-08 2022-04-14 Basf Se Mixtures containing cyclobutrifluram
AR123899A1 (es) 2020-10-23 2023-01-25 Vertellus Holdings Llc Métodos para elaborar derivados de ácido nicotínico
US20240016150A1 (en) 2020-12-01 2024-01-18 Basf Se Mixtures containing metarylpicoxamid
CN112602721A (zh) * 2020-12-15 2021-04-06 美丰农业科技(上海)有限公司 一种杀线虫农用组合物
CN112602718A (zh) * 2020-12-15 2021-04-06 美丰农业科技(上海)有限公司 一种含氟唑菌酰羟胺和Cyclobutrifluram的杀线虫农用组合物
EP4262393A1 (en) * 2020-12-17 2023-10-25 Syngenta Crop Protection AG Methods for controlling or preventing infestation of plants by a phytopathogenic microorganism of the genus aspergillus
CN115067343B (zh) * 2021-03-15 2023-09-29 江苏龙灯化学有限公司 一种杀线虫组合物
CN115067341B (zh) * 2021-03-15 2024-03-01 江苏龙灯化学有限公司 一种杀线虫组合物
CN113615698B (zh) * 2021-08-26 2023-09-15 青岛海利尔生物科技有限公司 一种杀线虫组合物及其用途
CN114208839A (zh) * 2021-12-23 2022-03-22 青岛海利尔生物科技有限公司 一种杀线虫组合物及其用途
CN114271281B (zh) * 2022-01-13 2023-05-30 青岛海利尔生物科技有限公司 一种杀线虫组合物及其应用
CN117546850B (zh) * 2022-01-24 2025-08-19 青岛海利尔生物科技有限公司 一种含Cyclobutrifluram的杀线虫组合物及其应用
KR20250129055A (ko) 2022-12-30 2025-08-28 신젠타 크롭 프로텍션 아게 4-원 고리 카르복사미드 화합물을 포함하는 조성물
WO2026032774A1 (en) 2024-08-08 2026-02-12 Basf Se Fungicidal compositions comprising strobilurins

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010511689A (ja) 2006-12-06 2010-04-15 ファイザー・インク （３Ｓ）−３−［Ｎ−（Ｎ’−（２−ｔｅｒｔ−ブチルフェニル）オキサミル）アラニニル］アミノ−５−（２’，３’，５’，６’−テトラフルオロフェノキシ）−４−オキソペンタン酸の結晶形態
JP2016528201A (ja) 2013-07-08 2016-09-15 シンジェンタ パーティシペーションズ アーゲー 殺線虫剤として使用される４員環カルボキサミド

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EP2644595A1 (en) * 2012-03-26 2013-10-02 Syngenta Participations AG. N-Cyclylamides as nematicides
UY35543A (es) 2013-04-30 2014-11-28 Bayer Cropscience Ag N-(fenilcicloalquil)carboxamidas y n-(fenilcicloalquil)tiocarboxamidas nematicidas
WO2016066644A1 (en) 2014-10-29 2016-05-06 Bayer Cropscience Aktiengesellschaft N-(phenylcycloalkyl)carboxamides and n-(phenylcycloalkyl)thiocarboxamides as fungicides

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010511689A (ja) 2006-12-06 2010-04-15 ファイザー・インク （３Ｓ）−３−［Ｎ−（Ｎ’−（２−ｔｅｒｔ−ブチルフェニル）オキサミル）アラニニル］アミノ−５−（２’，３’，５’，６’−テトラフルオロフェノキシ）−４−オキソペンタン酸の結晶形態
JP2016528201A (ja) 2013-07-08 2016-09-15 シンジェンタ パーティシペーションズ アーゲー 殺線虫剤として使用される４員環カルボキサミド

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
平山令明，有機化合物結晶作製ハンドブック，2008年，p.17-23,37-40,45-51,57-65

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Publication number Publication date
CA3286688A1 (en) 2025-11-29
US11053201B2 (en) 2021-07-06
EP4480542A2 (en) 2024-12-25
CL2022003528A1 (es) 2023-06-02
MA51819A (fr) 2021-05-19
CL2020002056A1 (es) 2020-10-23
AR114251A1 (es) 2020-08-12
CA3090960A1 (en) 2019-08-22
TWI815859B (zh) 2023-09-21
AU2019220997B2 (en) 2024-03-28
WO2019158476A1 (en) 2019-08-22
PE20211478A1 (es) 2021-08-05
MX2020008367A (es) 2020-09-25
EP4480542A3 (en) 2025-03-26
US20200369614A1 (en) 2020-11-26
EP3752489A1 (en) 2020-12-23
JOP20200194A1 (ar) 2020-08-11
EA202091893A1 (ru) 2020-12-22
TW202003468A (zh) 2020-01-16
ECSP20048382A (es) 2020-09-30
CO2020009901A2 (es) 2020-08-21
KR20250079046A (ko) 2025-06-04
UY38085A (es) 2019-10-01
AU2019220997A1 (en) 2020-09-03
UA129535C2 (uk) 2025-05-28
BR112020016431A2 (pt) 2020-12-15
JOP20250289A1 (ar) 2025-11-18
PE20250001A1 (es) 2025-01-07
KR20200120933A (ko) 2020-10-22
ZA202004700B (en) 2021-09-29
CN111741945A (zh) 2020-10-02
KR102812896B1 (ko) 2025-05-23
IL276644B2 (en) 2023-11-01
CN111741945B (zh) 2024-01-09
IL276644B1 (en) 2023-07-01
MY205650A (en) 2024-11-02
JP2021514356A (ja) 2021-06-10
IL276644A (en) 2020-09-30
PH12020551304A1 (en) 2021-08-16

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