TWI815859B - 新穎晶型 - Google Patents

新穎晶型 Download PDF

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Publication number
TWI815859B
TWI815859B TW108104399A TW108104399A TWI815859B TW I815859 B TWI815859 B TW I815859B TW 108104399 A TW108104399 A TW 108104399A TW 108104399 A TW108104399 A TW 108104399A TW I815859 B TWI815859 B TW I815859B
Authority
TW
Taiwan
Prior art keywords
methyl
diffraction pattern
plants
dichlorophenyl
formulations
Prior art date
Application number
TW108104399A
Other languages
English (en)
Chinese (zh)
Other versions
TW202003468A (zh
Inventor
約翰 侯尼
伊恩 凱文 瓊斯
Original Assignee
瑞士商先正達合夥公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 瑞士商先正達合夥公司 filed Critical 瑞士商先正達合夥公司
Publication of TW202003468A publication Critical patent/TW202003468A/zh
Application granted granted Critical
Publication of TWI815859B publication Critical patent/TWI815859B/zh

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C07D213/82—Amides; Imides in position 3
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P3/00—Fungicides
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P5/00—Nematocides
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P7/00—Arthropodicides
    • A01P7/04—Insecticides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Insects & Arthropods (AREA)
  • Mycology (AREA)
  • Microbiology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyridine Compounds (AREA)
  • Liquid Crystal Substances (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
TW108104399A 2018-02-13 2019-02-11 新穎晶型 TWI815859B (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP18156463.4 2018-02-13
EP18156463 2018-02-13

Publications (2)

Publication Number Publication Date
TW202003468A TW202003468A (zh) 2020-01-16
TWI815859B true TWI815859B (zh) 2023-09-21

Family

ID=61198760

Family Applications (1)

Application Number Title Priority Date Filing Date
TW108104399A TWI815859B (zh) 2018-02-13 2019-02-11 新穎晶型

Country Status (24)

Country Link
US (1) US11053201B2 (https=)
EP (2) EP3752489A1 (https=)
JP (1) JP7348904B2 (https=)
KR (2) KR102812896B1 (https=)
CN (1) CN111741945B (https=)
AR (1) AR114251A1 (https=)
AU (1) AU2019220997B2 (https=)
CA (2) CA3286688A1 (https=)
CL (2) CL2020002056A1 (https=)
CO (1) CO2020009901A2 (https=)
EA (1) EA202091893A1 (https=)
EC (1) ECSP20048382A (https=)
IL (1) IL276644B2 (https=)
JO (2) JOP20200194A1 (https=)
MA (1) MA51819A (https=)
MX (1) MX2020008367A (https=)
MY (1) MY205650A (https=)
PE (2) PE20211478A1 (https=)
PH (1) PH12020551304A1 (https=)
TW (1) TWI815859B (https=)
UA (1) UA129535C2 (https=)
UY (1) UY38085A (https=)
WO (1) WO2019158476A1 (https=)
ZA (1) ZA202004700B (https=)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL3019476T3 (pl) * 2013-07-08 2018-05-30 Syngenta Participations Ag Związki karboksyamidowe o 4-członowym pierścieniu jako nematocydy
AU2018390864B9 (en) * 2017-12-20 2024-12-12 Syngenta Crop Protection Ag Methods of controlling or preventing infestation of vegetable, tomato and potato plants by phytopathogenic microorganisms
AU2019342401A1 (en) * 2018-09-19 2021-04-15 Syngenta Crop Protection Ag Methods of controlling or preventing infestation of cereal plants by the phytopathogenic microorganism fusarium pseudograminearum
JP7758669B2 (ja) * 2019-12-10 2025-10-22 シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト マクロホミナ（ｍａｃｒｏｐｈｏｍｉｎａ）属の種の植物病原性微生物による植物の被害を防除するか又は防止する方法
CN115397243B (zh) * 2020-01-30 2025-03-28 先正达农作物保护股份公司 控制或预防香蕉植物中的巴拿马病的方法
WO2022073797A1 (en) 2020-10-08 2022-04-14 Basf Se Mixtures containing cyclobutrifluram
AR123899A1 (es) 2020-10-23 2023-01-25 Vertellus Holdings Llc Métodos para elaborar derivados de ácido nicotínico
US20240016150A1 (en) 2020-12-01 2024-01-18 Basf Se Mixtures containing metarylpicoxamid
CN112602721A (zh) * 2020-12-15 2021-04-06 美丰农业科技(上海)有限公司 一种杀线虫农用组合物
CN112602718A (zh) * 2020-12-15 2021-04-06 美丰农业科技(上海)有限公司 一种含氟唑菌酰羟胺和Cyclobutrifluram的杀线虫农用组合物
EP4262393A1 (en) * 2020-12-17 2023-10-25 Syngenta Crop Protection AG Methods for controlling or preventing infestation of plants by a phytopathogenic microorganism of the genus aspergillus
CN115067343B (zh) * 2021-03-15 2023-09-29 江苏龙灯化学有限公司 一种杀线虫组合物
CN115067341B (zh) * 2021-03-15 2024-03-01 江苏龙灯化学有限公司 一种杀线虫组合物
CN113615698B (zh) * 2021-08-26 2023-09-15 青岛海利尔生物科技有限公司 一种杀线虫组合物及其用途
CN114208839A (zh) * 2021-12-23 2022-03-22 青岛海利尔生物科技有限公司 一种杀线虫组合物及其用途
CN114271281B (zh) * 2022-01-13 2023-05-30 青岛海利尔生物科技有限公司 一种杀线虫组合物及其应用
CN117546850B (zh) * 2022-01-24 2025-08-19 青岛海利尔生物科技有限公司 一种含Cyclobutrifluram的杀线虫组合物及其应用
KR20250129055A (ko) 2022-12-30 2025-08-28 신젠타 크롭 프로텍션 아게 4-원 고리 카르복사미드 화합물을 포함하는 조성물
WO2026032774A1 (en) 2024-08-08 2026-02-12 Basf Se Fungicidal compositions comprising strobilurins

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015003951A1 (en) * 2013-07-08 2015-01-15 Syngenta Participations Ag 4-membered ring carboxamides used as nematicides
US9414589B2 (en) * 2012-03-26 2016-08-16 Syngenta Participations Ag N-cyclylamides as nematicides

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101125932B1 (ko) * 2006-12-06 2012-03-22 아이디유엔 파마슈티칼즈, 인코포레이티드 (3ｓ)-3-［ｎ-(ｎ'-(2-ｔｅｒｔ-부틸페닐)옥사밀)알라니닐］아미노-5-(2',3',5',6'-테트라플루오로페녹시)-4-옥소펜탄산의 결정 형태
UY35543A (es) 2013-04-30 2014-11-28 Bayer Cropscience Ag N-(fenilcicloalquil)carboxamidas y n-(fenilcicloalquil)tiocarboxamidas nematicidas
WO2016066644A1 (en) 2014-10-29 2016-05-06 Bayer Cropscience Aktiengesellschaft N-(phenylcycloalkyl)carboxamides and n-(phenylcycloalkyl)thiocarboxamides as fungicides

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9414589B2 (en) * 2012-03-26 2016-08-16 Syngenta Participations Ag N-cyclylamides as nematicides
WO2015003951A1 (en) * 2013-07-08 2015-01-15 Syngenta Participations Ag 4-membered ring carboxamides used as nematicides

Also Published As

Publication number Publication date
CA3286688A1 (en) 2025-11-29
US11053201B2 (en) 2021-07-06
EP4480542A2 (en) 2024-12-25
CL2022003528A1 (es) 2023-06-02
MA51819A (fr) 2021-05-19
CL2020002056A1 (es) 2020-10-23
AR114251A1 (es) 2020-08-12
CA3090960A1 (en) 2019-08-22
AU2019220997B2 (en) 2024-03-28
WO2019158476A1 (en) 2019-08-22
PE20211478A1 (es) 2021-08-05
MX2020008367A (es) 2020-09-25
EP4480542A3 (en) 2025-03-26
US20200369614A1 (en) 2020-11-26
EP3752489A1 (en) 2020-12-23
JOP20200194A1 (ar) 2020-08-11
EA202091893A1 (ru) 2020-12-22
TW202003468A (zh) 2020-01-16
ECSP20048382A (es) 2020-09-30
CO2020009901A2 (es) 2020-08-21
KR20250079046A (ko) 2025-06-04
UY38085A (es) 2019-10-01
AU2019220997A1 (en) 2020-09-03
UA129535C2 (uk) 2025-05-28
JP7348904B2 (ja) 2023-09-21
BR112020016431A2 (pt) 2020-12-15
JOP20250289A1 (ar) 2025-11-18
PE20250001A1 (es) 2025-01-07
KR20200120933A (ko) 2020-10-22
ZA202004700B (en) 2021-09-29
CN111741945A (zh) 2020-10-02
KR102812896B1 (ko) 2025-05-23
IL276644B2 (en) 2023-11-01
CN111741945B (zh) 2024-01-09
IL276644B1 (en) 2023-07-01
MY205650A (en) 2024-11-02
JP2021514356A (ja) 2021-06-10
IL276644A (en) 2020-09-30
PH12020551304A1 (en) 2021-08-16

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