AU2019220997B2 - Novel crystalline forms - Google Patents

Novel crystalline forms Download PDF

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Publication number
AU2019220997B2
AU2019220997B2 AU2019220997A AU2019220997A AU2019220997B2 AU 2019220997 B2 AU2019220997 B2 AU 2019220997B2 AU 2019220997 A AU2019220997 A AU 2019220997A AU 2019220997 A AU2019220997 A AU 2019220997A AU 2019220997 B2 AU2019220997 B2 AU 2019220997B2
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AU
Australia
Prior art keywords
methyl
plant
crystalline form
formulations
dichlorophenyl
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AU2019220997A
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English (en)
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AU2019220997A1 (en
Inventor
John Hone
Ian Kevin Jones
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Syngenta Crop Protection AG Switzerland
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Syngenta Crop Protection AG Switzerland
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Publication of AU2019220997A1 publication Critical patent/AU2019220997A1/en
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Assigned to SYNGENTA CROP PROTECTION AG reassignment SYNGENTA CROP PROTECTION AG Request to Amend Deed and Register Assignors: SYNGENTA PARTICIPATIONS AG
Active legal-status Critical Current
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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81Amides; Imides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81Amides; Imides
    • C07D213/82Amides; Imides in position 3
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01PBIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P3/00Fungicides
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01PBIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P5/00Nematocides
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01PBIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P7/00Arthropodicides
    • A01P7/04Insecticides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Insects & Arthropods (AREA)
  • Mycology (AREA)
  • Microbiology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyridine Compounds (AREA)
  • Liquid Crystal Substances (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2019220997A 2018-02-13 2019-02-11 Novel crystalline forms Active AU2019220997B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP18156463.4 2018-02-13
EP18156463 2018-02-13
PCT/EP2019/053292 WO2019158476A1 (en) 2018-02-13 2019-02-11 Novel crystalline forms

Publications (2)

Publication Number Publication Date
AU2019220997A1 AU2019220997A1 (en) 2020-09-03
AU2019220997B2 true AU2019220997B2 (en) 2024-03-28

Family

ID=61198760

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2019220997A Active AU2019220997B2 (en) 2018-02-13 2019-02-11 Novel crystalline forms

Country Status (24)

Country Link
US (1) US11053201B2 (https=)
EP (2) EP3752489A1 (https=)
JP (1) JP7348904B2 (https=)
KR (2) KR102812896B1 (https=)
CN (1) CN111741945B (https=)
AR (1) AR114251A1 (https=)
AU (1) AU2019220997B2 (https=)
CA (2) CA3286688A1 (https=)
CL (2) CL2020002056A1 (https=)
CO (1) CO2020009901A2 (https=)
EA (1) EA202091893A1 (https=)
EC (1) ECSP20048382A (https=)
IL (1) IL276644B2 (https=)
JO (2) JOP20200194A1 (https=)
MA (1) MA51819A (https=)
MX (1) MX2020008367A (https=)
MY (1) MY205650A (https=)
PE (2) PE20211478A1 (https=)
PH (1) PH12020551304A1 (https=)
TW (1) TWI815859B (https=)
UA (1) UA129535C2 (https=)
UY (1) UY38085A (https=)
WO (1) WO2019158476A1 (https=)
ZA (1) ZA202004700B (https=)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL3019476T3 (pl) * 2013-07-08 2018-05-30 Syngenta Participations Ag Związki karboksyamidowe o 4-członowym pierścieniu jako nematocydy
AU2018390864B9 (en) * 2017-12-20 2024-12-12 Syngenta Crop Protection Ag Methods of controlling or preventing infestation of vegetable, tomato and potato plants by phytopathogenic microorganisms
AU2019342401A1 (en) * 2018-09-19 2021-04-15 Syngenta Crop Protection Ag Methods of controlling or preventing infestation of cereal plants by the phytopathogenic microorganism fusarium pseudograminearum
JP7758669B2 (ja) * 2019-12-10 2025-10-22 シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト マクロホミナ(macrophomina)属の種の植物病原性微生物による植物の被害を防除するか又は防止する方法
CN115397243B (zh) * 2020-01-30 2025-03-28 先正达农作物保护股份公司 控制或预防香蕉植物中的巴拿马病的方法
WO2022073797A1 (en) 2020-10-08 2022-04-14 Basf Se Mixtures containing cyclobutrifluram
AR123899A1 (es) 2020-10-23 2023-01-25 Vertellus Holdings Llc Métodos para elaborar derivados de ácido nicotínico
US20240016150A1 (en) 2020-12-01 2024-01-18 Basf Se Mixtures containing metarylpicoxamid
CN112602721A (zh) * 2020-12-15 2021-04-06 美丰农业科技(上海)有限公司 一种杀线虫农用组合物
CN112602718A (zh) * 2020-12-15 2021-04-06 美丰农业科技(上海)有限公司 一种含氟唑菌酰羟胺和Cyclobutrifluram的杀线虫农用组合物
EP4262393A1 (en) * 2020-12-17 2023-10-25 Syngenta Crop Protection AG Methods for controlling or preventing infestation of plants by a phytopathogenic microorganism of the genus aspergillus
CN115067343B (zh) * 2021-03-15 2023-09-29 江苏龙灯化学有限公司 一种杀线虫组合物
CN115067341B (zh) * 2021-03-15 2024-03-01 江苏龙灯化学有限公司 一种杀线虫组合物
CN113615698B (zh) * 2021-08-26 2023-09-15 青岛海利尔生物科技有限公司 一种杀线虫组合物及其用途
CN114208839A (zh) * 2021-12-23 2022-03-22 青岛海利尔生物科技有限公司 一种杀线虫组合物及其用途
CN114271281B (zh) * 2022-01-13 2023-05-30 青岛海利尔生物科技有限公司 一种杀线虫组合物及其应用
CN117546850B (zh) * 2022-01-24 2025-08-19 青岛海利尔生物科技有限公司 一种含Cyclobutrifluram的杀线虫组合物及其应用
KR20250129055A (ko) 2022-12-30 2025-08-28 신젠타 크롭 프로텍션 아게 4-원 고리 카르복사미드 화합물을 포함하는 조성물
WO2026032774A1 (en) 2024-08-08 2026-02-12 Basf Se Fungicidal compositions comprising strobilurins

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015003951A1 (en) * 2013-07-08 2015-01-15 Syngenta Participations Ag 4-membered ring carboxamides used as nematicides

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101125932B1 (ko) * 2006-12-06 2012-03-22 아이디유엔 파마슈티칼즈, 인코포레이티드 (3s)-3-[n-(n'-(2-tert-부틸페닐)옥사밀)알라니닐]아미노-5-(2',3',5',6'-테트라플루오로페녹시)-4-옥소펜탄산의 결정 형태
EP2644595A1 (en) * 2012-03-26 2013-10-02 Syngenta Participations AG. N-Cyclylamides as nematicides
UY35543A (es) 2013-04-30 2014-11-28 Bayer Cropscience Ag N-(fenilcicloalquil)carboxamidas y n-(fenilcicloalquil)tiocarboxamidas nematicidas
WO2016066644A1 (en) 2014-10-29 2016-05-06 Bayer Cropscience Aktiengesellschaft N-(phenylcycloalkyl)carboxamides and n-(phenylcycloalkyl)thiocarboxamides as fungicides

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015003951A1 (en) * 2013-07-08 2015-01-15 Syngenta Participations Ag 4-membered ring carboxamides used as nematicides

Also Published As

Publication number Publication date
CA3286688A1 (en) 2025-11-29
US11053201B2 (en) 2021-07-06
EP4480542A2 (en) 2024-12-25
CL2022003528A1 (es) 2023-06-02
MA51819A (fr) 2021-05-19
CL2020002056A1 (es) 2020-10-23
AR114251A1 (es) 2020-08-12
CA3090960A1 (en) 2019-08-22
TWI815859B (zh) 2023-09-21
WO2019158476A1 (en) 2019-08-22
PE20211478A1 (es) 2021-08-05
MX2020008367A (es) 2020-09-25
EP4480542A3 (en) 2025-03-26
US20200369614A1 (en) 2020-11-26
EP3752489A1 (en) 2020-12-23
JOP20200194A1 (ar) 2020-08-11
EA202091893A1 (ru) 2020-12-22
TW202003468A (zh) 2020-01-16
ECSP20048382A (es) 2020-09-30
CO2020009901A2 (es) 2020-08-21
KR20250079046A (ko) 2025-06-04
UY38085A (es) 2019-10-01
AU2019220997A1 (en) 2020-09-03
UA129535C2 (uk) 2025-05-28
JP7348904B2 (ja) 2023-09-21
BR112020016431A2 (pt) 2020-12-15
JOP20250289A1 (ar) 2025-11-18
PE20250001A1 (es) 2025-01-07
KR20200120933A (ko) 2020-10-22
ZA202004700B (en) 2021-09-29
CN111741945A (zh) 2020-10-02
KR102812896B1 (ko) 2025-05-23
IL276644B2 (en) 2023-11-01
CN111741945B (zh) 2024-01-09
IL276644B1 (en) 2023-07-01
MY205650A (en) 2024-11-02
JP2021514356A (ja) 2021-06-10
IL276644A (en) 2020-09-30
PH12020551304A1 (en) 2021-08-16

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HB Alteration of name in register

Owner name: SYNGENTA CROP PROTECTION AG

Free format text: FORMER NAME(S): SYNGENTA PARTICIPATIONS AG