CN111741945B - 晶形 - Google Patents

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Publication number
CN111741945B
CN111741945B CN201980013098.5A CN201980013098A CN111741945B CN 111741945 B CN111741945 B CN 111741945B CN 201980013098 A CN201980013098 A CN 201980013098A CN 111741945 B CN111741945 B CN 111741945B
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CN
China
Prior art keywords
methyl
nematodes
species
plants
pyridine
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CN201980013098.5A
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English (en)
Chinese (zh)
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CN111741945A (zh
Inventor
J·霍恩
I·K·琼斯
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Syngenta Crop Protection AG Switzerland
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Syngenta Participations AG
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Publication of CN111741945A publication Critical patent/CN111741945A/zh
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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C07D213/82—Amides; Imides in position 3
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P3/00—Fungicides
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P5/00—Nematocides
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P7/00—Arthropodicides
    • A01P7/04—Insecticides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Insects & Arthropods (AREA)
  • Mycology (AREA)
  • Microbiology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyridine Compounds (AREA)
  • Liquid Crystal Substances (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CN201980013098.5A 2018-02-13 2019-02-11 晶形 Active CN111741945B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP18156463.4 2018-02-13
EP18156463 2018-02-13
PCT/EP2019/053292 WO2019158476A1 (en) 2018-02-13 2019-02-11 Novel crystalline forms

Publications (2)

Publication Number Publication Date
CN111741945A CN111741945A (zh) 2020-10-02
CN111741945B true CN111741945B (zh) 2024-01-09

Family

ID=61198760

Family Applications (1)

Application Number Title Priority Date Filing Date
CN201980013098.5A Active CN111741945B (zh) 2018-02-13 2019-02-11 晶形

Country Status (24)

Country Link
US (1) US11053201B2 (https=)
EP (2) EP3752489A1 (https=)
JP (1) JP7348904B2 (https=)
KR (2) KR102812896B1 (https=)
CN (1) CN111741945B (https=)
AR (1) AR114251A1 (https=)
AU (1) AU2019220997B2 (https=)
CA (2) CA3286688A1 (https=)
CL (2) CL2020002056A1 (https=)
CO (1) CO2020009901A2 (https=)
EA (1) EA202091893A1 (https=)
EC (1) ECSP20048382A (https=)
IL (1) IL276644B2 (https=)
JO (2) JOP20200194A1 (https=)
MA (1) MA51819A (https=)
MX (1) MX2020008367A (https=)
MY (1) MY205650A (https=)
PE (2) PE20211478A1 (https=)
PH (1) PH12020551304A1 (https=)
TW (1) TWI815859B (https=)
UA (1) UA129535C2 (https=)
UY (1) UY38085A (https=)
WO (1) WO2019158476A1 (https=)
ZA (1) ZA202004700B (https=)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL3019476T3 (pl) * 2013-07-08 2018-05-30 Syngenta Participations Ag Związki karboksyamidowe o 4-członowym pierścieniu jako nematocydy
AU2018390864B9 (en) * 2017-12-20 2024-12-12 Syngenta Crop Protection Ag Methods of controlling or preventing infestation of vegetable, tomato and potato plants by phytopathogenic microorganisms
AU2019342401A1 (en) * 2018-09-19 2021-04-15 Syngenta Crop Protection Ag Methods of controlling or preventing infestation of cereal plants by the phytopathogenic microorganism fusarium pseudograminearum
JP7758669B2 (ja) * 2019-12-10 2025-10-22 シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト マクロホミナ（ｍａｃｒｏｐｈｏｍｉｎａ）属の種の植物病原性微生物による植物の被害を防除するか又は防止する方法
CN115397243B (zh) * 2020-01-30 2025-03-28 先正达农作物保护股份公司 控制或预防香蕉植物中的巴拿马病的方法
WO2022073797A1 (en) 2020-10-08 2022-04-14 Basf Se Mixtures containing cyclobutrifluram
AR123899A1 (es) 2020-10-23 2023-01-25 Vertellus Holdings Llc Métodos para elaborar derivados de ácido nicotínico
US20240016150A1 (en) 2020-12-01 2024-01-18 Basf Se Mixtures containing metarylpicoxamid
CN112602721A (zh) * 2020-12-15 2021-04-06 美丰农业科技(上海)有限公司 一种杀线虫农用组合物
CN112602718A (zh) * 2020-12-15 2021-04-06 美丰农业科技(上海)有限公司 一种含氟唑菌酰羟胺和Cyclobutrifluram的杀线虫农用组合物
EP4262393A1 (en) * 2020-12-17 2023-10-25 Syngenta Crop Protection AG Methods for controlling or preventing infestation of plants by a phytopathogenic microorganism of the genus aspergillus
CN115067343B (zh) * 2021-03-15 2023-09-29 江苏龙灯化学有限公司 一种杀线虫组合物
CN115067341B (zh) * 2021-03-15 2024-03-01 江苏龙灯化学有限公司 一种杀线虫组合物
CN113615698B (zh) * 2021-08-26 2023-09-15 青岛海利尔生物科技有限公司 一种杀线虫组合物及其用途
CN114208839A (zh) * 2021-12-23 2022-03-22 青岛海利尔生物科技有限公司 一种杀线虫组合物及其用途
CN114271281B (zh) * 2022-01-13 2023-05-30 青岛海利尔生物科技有限公司 一种杀线虫组合物及其应用
CN117546850B (zh) * 2022-01-24 2025-08-19 青岛海利尔生物科技有限公司 一种含Cyclobutrifluram的杀线虫组合物及其应用
KR20250129055A (ko) 2022-12-30 2025-08-28 신젠타 크롭 프로텍션 아게 4-원 고리 카르복사미드 화합물을 포함하는 조성물
WO2026032774A1 (en) 2024-08-08 2026-02-12 Basf Se Fungicidal compositions comprising strobilurins

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101573328A (zh) * 2006-12-06 2009-11-04 辉瑞有限公司 (3s)-3-[n-(n’-(2-叔丁基苯基)草氨酰基)丙氨酰基]氨基-5-(2’,3’,5’,6’-四氟苯氧基)-4-氧代戊酸的结晶形式
EP2644595A1 (en) * 2012-03-26 2013-10-02 Syngenta Participations AG. N-Cyclylamides as nematicides
CN105431414A (zh) * 2013-07-08 2016-03-23 先正达参股股份有限公司 用作杀线虫剂的4元环甲酰胺

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UY35543A (es) 2013-04-30 2014-11-28 Bayer Cropscience Ag N-(fenilcicloalquil)carboxamidas y n-(fenilcicloalquil)tiocarboxamidas nematicidas
WO2016066644A1 (en) 2014-10-29 2016-05-06 Bayer Cropscience Aktiengesellschaft N-(phenylcycloalkyl)carboxamides and n-(phenylcycloalkyl)thiocarboxamides as fungicides

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101573328A (zh) * 2006-12-06 2009-11-04 辉瑞有限公司 (3s)-3-[n-(n’-(2-叔丁基苯基)草氨酰基)丙氨酰基]氨基-5-(2’,3’,5’,6’-四氟苯氧基)-4-氧代戊酸的结晶形式
EP2644595A1 (en) * 2012-03-26 2013-10-02 Syngenta Participations AG. N-Cyclylamides as nematicides
CN105431414A (zh) * 2013-07-08 2016-03-23 先正达参股股份有限公司 用作杀线虫剂的4元环甲酰胺

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
赵桂森等主编.《新药设计与开发基础》.山东大学出版社,2015,第92-93页. *

Also Published As

Publication number Publication date
CA3286688A1 (en) 2025-11-29
US11053201B2 (en) 2021-07-06
EP4480542A2 (en) 2024-12-25
CL2022003528A1 (es) 2023-06-02
MA51819A (fr) 2021-05-19
CL2020002056A1 (es) 2020-10-23
AR114251A1 (es) 2020-08-12
CA3090960A1 (en) 2019-08-22
TWI815859B (zh) 2023-09-21
AU2019220997B2 (en) 2024-03-28
WO2019158476A1 (en) 2019-08-22
PE20211478A1 (es) 2021-08-05
MX2020008367A (es) 2020-09-25
EP4480542A3 (en) 2025-03-26
US20200369614A1 (en) 2020-11-26
EP3752489A1 (en) 2020-12-23
JOP20200194A1 (ar) 2020-08-11
EA202091893A1 (ru) 2020-12-22
TW202003468A (zh) 2020-01-16
ECSP20048382A (es) 2020-09-30
CO2020009901A2 (es) 2020-08-21
KR20250079046A (ko) 2025-06-04
UY38085A (es) 2019-10-01
AU2019220997A1 (en) 2020-09-03
UA129535C2 (uk) 2025-05-28
JP7348904B2 (ja) 2023-09-21
BR112020016431A2 (pt) 2020-12-15
JOP20250289A1 (ar) 2025-11-18
PE20250001A1 (es) 2025-01-07
KR20200120933A (ko) 2020-10-22
ZA202004700B (en) 2021-09-29
CN111741945A (zh) 2020-10-02
KR102812896B1 (ko) 2025-05-23
IL276644B2 (en) 2023-11-01
IL276644B1 (en) 2023-07-01
MY205650A (en) 2024-11-02
JP2021514356A (ja) 2021-06-10
IL276644A (en) 2020-09-30
PH12020551304A1 (en) 2021-08-16

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Patentee before: SYNGENTA PARTICIPATIONS AG

Country or region before: Switzerland